发明授权
US06613766B1 Pentaaza-cyclopental[a]naphthalene derivatives as ligands for GABAa &agr;5 receptors
失效
Pentaaza-cyclopial [a]萘衍生物作为GABAaα5受体的配体
![Pentaaza-cyclopental[a]naphthalene derivatives as ligands for GABAa &agr;5 receptors](/docs/US/2003-09-02/US06613766B1/abs.jpg.600x600.jpg)
- 专利标题： Pentaaza-cyclopental[a]naphthalene derivatives as ligands for GABAa &agr;5 receptors
- 专利标题（中）： Pentaaza-cyclopial [a]萘衍生物作为GABAaα5受体的配体
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申请号： US09831547申请日： 2001-05-10
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公开(公告)号： US06613766B1公开(公告)日： 2003-09-02
- 发明人: Neil Roy Curtis , Janusz Jozef Kulagowski , Francine Sternfeld
- 申请人： Neil Roy Curtis , Janusz Jozef Kulagowski , Francine Sternfeld
- 优先权： GB9824897 19981112
- 主分类号： A61K3150
- IPC分类号： A61K3150
![Pentaaza-cyclopental[a]naphthalene derivatives as ligands for GABAa &agr;5 receptors](/abs-image/US/2003/09/02/US06613766B1/abs.jpg.150x150.jpg)
摘要：
A class of 1,2,3a,4,x-pentaaza-cyclopenta[a]naphthalene compounds (x=6, 7, 8 or 9) is described. The compounds have a high affinity for the GABAA &agr;5 receptors and show inverse agonist activity thereat. The compounds are useful in therapy where cognition enhancement is required.
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