发明授权
- 专利标题: Indolylmaleimide derivatives
- 专利标题(中): 吲哚马来酰亚胺衍生物
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申请号: US10007368申请日: 2001-11-05
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公开(公告)号: US06645970B2公开(公告)日: 2003-11-11
- 发明人: Rainer Albert , Nigel Graham Cooke , Sylvain Cottens , Claus Ehrhardt , Jean-Pierre Evenou , Richard Sedrani , Peter Von Matt , Jürgen Wagner , Gerhard Zenke
- 申请人: Rainer Albert , Nigel Graham Cooke , Sylvain Cottens , Claus Ehrhardt , Jean-Pierre Evenou , Richard Sedrani , Peter Von Matt , Jürgen Wagner , Gerhard Zenke
- 主分类号: A61K31498
- IPC分类号: A61K31498
摘要:
Indolylmaleimide derivatives comprising either a substituted phenyl, naphthyl, tetrahydronaphthyl, quinazolinyl, quinolyl, isoquinolyl or pyrimidinyl residue have interesting pharmaceutical properties, e.g. in the treatment and/or prevention of T-cell mediated acute or chronic inflammatory diseases or disorders, autoimmune diseases, graft rejection or cancer.
公开/授权文献
- US20030069424A1 Indolylmaleimide derivatives 公开/授权日:2003-04-10