1,2,3,4-tetrahydroisoquinoline derivatives

Invention Grant

US06703392B2 1,2,3,4-tetrahydroisoquinoline derivatives 有权

Title translation: 1,2,3,4-四氢异喹啉衍生物

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Patent Title: 1,2,3,4-tetrahydroisoquinoline derivatives
Patent Title (中): 1,2,3,4-四氢异喹啉衍生物
Application No.: US10239693

Application Date: 2003-02-24
Publication No.: US06703392B2

Publication Date: 2004-03-09
Inventor: Hamed Aissaoui , Michael Cappi , Martine Clozel , Walter Fischli , Ralf Koberstein
Applicant: Hamed Aissaoui , Michael Cappi , Martine Clozel , Walter Fischli , Ralf Koberstein
Priority: EPPCT/EP00/02245 20000314
Main IPC: C07D21704
IPC: C07D21704

1,2,3,4-tetrahydroisoquinoline derivatives

Abstract:

The invention relates to novel 1,2,3,4-tetrahydroisochinoline derivatives of formula (I) and their use as active ingredients in the preparation of pharmaceutical compositions. The invention also concerns related aspects including processes for the preparation of the compounds, pharmaceutical compositions containing one or more of those compounds and especially their use as orexin receptor antagonists.

Abstract(Chinese):

本发明涉及式（I）的新型1,2,3,4-四氢异噻唑啉衍生物及其在制备药物组合物中作为活性成分的用途。本发明还涉及包括制备化合物的方法，含有一种或多种这些化合物的药物组合物，特别是其作为食欲素受体拮抗剂的用途的相关方面。

Public/Granted literature

US20030176415A1 1,2,3,4-tetrahydroisoquinoline derivatives Public/Granted day:2003-09-18

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