- 专利标题: α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
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申请号: US11110943申请日: 2005-04-21
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公开(公告)号: US07141609B2公开(公告)日: 2006-11-28
- 发明人: Michael L. Vazquez , Richard A. Mueller , John J. Talley , Daniel P. Getman , Gary A. DeCrescenzo , John N. Freskos , Deborah E. Bertenshaw , Robert M. Heintz
- 申请人: Michael L. Vazquez , Richard A. Mueller , John J. Talley , Daniel P. Getman , Gary A. DeCrescenzo , John N. Freskos , Deborah E. Bertenshaw , Robert M. Heintz
- 申请人地址: US IL Chicago
- 专利权人: G.D. Searle & Co.
- 当前专利权人: G.D. Searle & Co.
- 当前专利权人地址: US IL Chicago
- 代理机构: Banner & Witcoff, Ltd.
- 主分类号: A61K31/27
- IPC分类号: A61K31/27 ; A61K31/19
摘要:
α- and β-amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.