发明授权
US07220740B2 1,4-diazabicyclo[3.2.2]nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof
有权
1,4-二氮杂双环[3.2.2]壬苯并唑，苯并噻唑和苯并咪唑衍生物，其制备和治疗用途
![1,4-diazabicyclo[3.2.2]nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof](/docs/US/2007-05-22/US07220740B2/abs.jpg.600x600.jpg)
- 专利标题： 1,4-diazabicyclo[3.2.2]nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof
- 专利标题（中）： 1,4-二氮杂双环[3.2.2]壬苯并唑，苯并噻唑和苯并咪唑衍生物，其制备和治疗用途
-
申请号： US10276646申请日： 2001-05-29
-
公开(公告)号： US07220740B2公开(公告)日： 2007-05-22
- 发明人: Frédéric Galli , Alistair Lochead , Axelle Samson
- 申请人： Frédéric Galli , Alistair Lochead , Axelle Samson
- 申请人地址： FR Paris
- 专利权人： Sanofi-aventis
- 当前专利权人： Sanofi-aventis
- 当前专利权人地址： FR Paris
- 代理商 Balaram Gupta
- 优先权： FR0006975 20000531
- 国际申请： PCT/FR01/01651 WO 20010529
- 国际公布： WO01/92261 WO 20011206
- 主分类号： C07D471/08
- IPC分类号： C07D471/08 ; A61K31/55 ; A61P25/00
![1,4-diazabicyclo[3.2.2]nonabenzoxazole, -benzothiazole and benzimidazole derivatives, preparation and therapeutic use thereof](/abs-image/US/2007/05/22/US07220740B2/abs.jpg.150x150.jpg)
摘要：
Compound corresponding to the general formula (I) in which X represents an oxygen or sulphur atom or an NH group and R1, R2, R3 and R4 each represent a hydrogen or halogen atom or a nitro, amino, trifluoromethyl, trifluoroalkoxy, cyano, hydroxyl, (C1–C6)alkyl, (C1–C6)alkoxy or phenyl group. Application in therapeutics.