Invention Grant
US07226924B2 Substituted 3,4-dihydro-pyrimido[1,2a]pyrimidines and 3,4-dihydro-pyrazino[1,2a]pyrimidines, and methods for their preparation and use
失效
取代的3,4-二氢 - 嘧啶并[1,2a]嘧啶和3,4-二氢 - 吡嗪并[1,2a]嘧啶及其制备和使用方法
- Patent Title: Substituted 3,4-dihydro-pyrimido[1,2a]pyrimidines and 3,4-dihydro-pyrazino[1,2a]pyrimidines, and methods for their preparation and use
- Patent Title (中): 取代的3,4-二氢 - 嘧啶并[1,2a]嘧啶和3,4-二氢 - 吡嗪并[1,2a]嘧啶及其制备和使用方法
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Application No.: US10409614Application Date: 2003-04-09
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Publication No.: US07226924B2Publication Date: 2007-06-05
- Inventor: Matthias Gerlach , Corinna Maul , Utz-Peter Jagusch
- Applicant: Matthias Gerlach , Corinna Maul , Utz-Peter Jagusch
- Applicant Address: DE Aachen
- Assignee: Gruenenthal GmbH
- Current Assignee: Gruenenthal GmbH
- Current Assignee Address: DE Aachen
- Agency: Crowell & Moring LLP
- Priority: DE10050661 20001013
- Main IPC: C07D487/04
- IPC: C07D487/04 ; A61K31/519 ; A61P29/00 ; A61P13/02
![Substituted 3,4-dihydro-pyrimido[1,2a]pyrimidines and 3,4-dihydro-pyrazino[1,2a]pyrimidines, and methods for their preparation and use](/abs-image/US/2007/06/05/US07226924B2/abs.jpg.150x150.jpg)
Abstract:
Substituted 3,4-dihydro-pyrimido[1,2a]pyrimidines and 3,4-dihydro-pyrazino[1,2a]pyrimidines of general formula I, the invention also relates to a method for the production thereof, substance libraries containing these compounds, medicaments which contain these compounds in the production of medicaments for treating pain, urinary incontinence, itching, tinnitus aurium and/or diarrhea and to pharmaceutical compositions containing these compounds.
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