发明授权
- 专利标题： Process for preparing glycopeptide phosphonate derivatives
- 专利标题（中）： 制备糖肽膦酸酯衍生物的方法
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申请号： US11437066申请日： 2006-05-19
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公开(公告)号： US07301004B2公开(公告)日： 2007-11-27
- 发明人: Michael R. Leadbetter , Martin S. Linsell , Junning Lee , Jyanwei Liu
- 申请人： Michael R. Leadbetter , Martin S. Linsell , Junning Lee , Jyanwei Liu
- 申请人地址： US CA South San Francisco
- 专利权人： Theravance, Inc.
- 当前专利权人： Theravance, Inc.
- 当前专利权人地址： US CA South San Francisco
- 代理商 Jeffrey A. Hagenah
- 主分类号： A61K38/14
- IPC分类号： A61K38/14 ; C07K9/0014
摘要：
Disclosed are processes for preparing glycopeptide phosphonate derivatives having an amino-containing side chain. Several of the process steps are conducted in a single reaction vessel without isolation of intermediate reaction products, thereby generating less waste and improving the overall efficiency and yield of the process.