Invention Grant
- Patent Title: Fused heterocycles
- Patent Title (中): 融合杂环
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Application No.: US11833903Application Date: 2007-08-03
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Publication No.: US07579370B2Publication Date: 2009-08-25
- Inventor: Michele L. R. Heffernan , James M. Dorsey , Qun Kevin Fang , Robert J. Foglesong , Seth C. Hopkins , Cyprian O. Ogbu , Mustapha Soukri , Kerry L. Spear
- Applicant: Michele L. R. Heffernan , James M. Dorsey , Qun Kevin Fang , Robert J. Foglesong , Seth C. Hopkins , Cyprian O. Ogbu , Mustapha Soukri , Kerry L. Spear
- Applicant Address: US MA Marlborough
- Assignee: Sepracor Inc.
- Current Assignee: Sepracor Inc.
- Current Assignee Address: US MA Marlborough
- Agency: Morgan, Lewis & Bockius, LLP
- Main IPC: A61K31/40
- IPC: A61K31/40 ; A61K31/34 ; A61K31/19 ; A01N43/38 ; A01N43/08 ; A01N37/00

Abstract:
This invention provides fused heterocycles having the formula: in which R1 is a member selected from the group consisting of H, substituted or unsubstituted arylalkyl and substituted or unsubstituted heteroarylalkyl. R2 is a member selected from the group consisting of H substituted or unsubstituted alkenyl, substituted or unsubstituted arylalkyl and substituted or unsubstituted heteroarylalkyl. R3is a member selected from the group consisting of H, C1-C6 substituted or unsubstituted alkyl, substituted or unsubstituted arylalkyl and substituted or unsubstituted heteroarylalkyl. R4 is a member selected from OH and O−X+, in which X+ is positive ion which is a member selected from organic positive ions and inorganic positive ions. Substituted or unsubstituted arylalkyl and substituted or unsubstituted heteroarylalkyl moieties have the formula: in which Ar is a member selected from the group consisting of substituted or unsubstituted aryl and substituted or unsubstituted heteroaryl. The index n is an integer from 1 to 4.
Public/Granted literature
- US20080004328A1 FUSED HETEROCYCLES Public/Granted day:2008-01-03
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