发明授权
- 专利标题: Pyrrolopyridine derivative and use thereof
- 专利标题(中): 吡咯并吡啶衍生物及其用途
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申请号: US10520784申请日: 2003-07-10
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公开(公告)号: US07582651B2公开(公告)日: 2009-09-01
- 发明人: Takahiro Matsumoto , Osamu Kurasawa , Tsuneo Oda , Hiroshi Nagabukuro , Manabu Mochizuki
- 申请人: Takahiro Matsumoto , Osamu Kurasawa , Tsuneo Oda , Hiroshi Nagabukuro , Manabu Mochizuki
- 申请人地址: JP Osaka
- 专利权人: Takeda Pharmaceutical Company Limited
- 当前专利权人: Takeda Pharmaceutical Company Limited
- 当前专利权人地址: JP Osaka
- 代理机构: Sughrue Mion, PLLC
- 优先权: JP2002-202204 20020711
- 国际申请: PCT/JP03/08791 WO 20030710
- 国际公布: WO2004/007495 WO 20040122
- 主分类号: A61K31/44
- IPC分类号: A61K31/44 ; C07D513/02
摘要:
A novel pyrrolopyridine derivative which is a compound represented by the formula wherein Ring A represents an optionally substituted pyridine ring; X represents an electron-attracting group; Y represents an optionally substituted divalent C1-6 chain hydrocarbon group; R1 represents an optionally substituted hydrocarbon group; and R2 and R3 each independently represents hydrogen, an optionally substituted hydrocarbon group or an optionally-substituted heterocyclic group, or R2 and R3 may form an optionally substituted ring in cooperation with the adjacent nitrogen atom, or a salt of the compound. The pyrrolopyridine derivative has vanilloid receptor agonist activity and is useful as medicines such as a preventive/therapeutic agent and analgesic for overactive bladder.
公开/授权文献
- US20060167038A1 Pyrrolopyridine derivative and use thereof 公开/授权日:2006-07-27
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