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US07915422B2 Processes for the preparation of substituted sulfoxides 有权
制备取代亚砜的方法

Processes for the preparation of substituted sulfoxides
Abstract:
The present invention relates to a process for enantioselective synthesis of substituted pyridinylmethyl sulfinyl-benzimidazole of compound of Formula (I). The process includes enantioselective catalytic oxidation of a substituted pyridinylmethyl prochiral sulfide derivative of compound of Formula (II) with an oxidizing agent in the presence of a chiral transition metal complex and a base in the absence of an organic solvent.
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