发明授权
- 专利标题: Amino acid surrogates for peptidic constructs
- 专利标题(中): 氨基酸替代肽结构
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申请号: US11694181申请日: 2007-03-30
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公开(公告)号: US07964181B2公开(公告)日: 2011-06-21
- 发明人: Shubh D. Sharma , Margarita Bastos , Wei Yang , Hui-Zhi Cai
- 申请人: Shubh D. Sharma , Margarita Bastos , Wei Yang , Hui-Zhi Cai
- 申请人地址: US NJ Cranbury
- 专利权人: Palatin Technologies, Inc.
- 当前专利权人: Palatin Technologies, Inc.
- 当前专利权人地址: US NJ Cranbury
- 代理商 Stephen A. Slusher
- 主分类号: A61K31/785
- IPC分类号: A61K31/785 ; A61K47/16 ; A61K38/02 ; A01N43/34
摘要:
Ring-constrained amino acid surrogates of formula I: where R1, R2, R3, R4, R5, R6a, R6b, R7, and y are as defined in the specification, methods for synthesizing ring-constrained amino acid surrogates of formula I, methods of use of ring-constrained amino acid surrogates of formula I, including use in linear or cyclic compounds which include a plurality of amino acid residues and one or more ring-constrained amino acid surrogates of formula I and linear or cyclic compounds which include a plurality of amino acid residues and one or more ring-constrained amino acid surrogates of formula I.
公开/授权文献
- US20070260040A1 Amino Acid Surrogates for Peptidic Constructs 公开/授权日:2007-11-08