发明授权
US08101629B2 Salt of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile
有权
4 - [[4 - [[4-(2-氰基乙烯基)-2,6-二甲基苯基]氨基] -2-嘧啶基]氨基]苄腈
- 专利标题: Salt of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino]benzonitrile
- 专利标题(中): 4 - [[4 - [[4-(2-氰基乙烯基)-2,6-二甲基苯基]氨基] -2-嘧啶基]氨基]苄腈
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申请号: US12845463申请日: 2010-07-28
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公开(公告)号: US08101629B2公开(公告)日: 2012-01-24
- 发明人: Jérôme Emile Georges Guillemont , Paul Theodoor Agnes Stevens , Alex Herman Copmans , Jozef Peeters , Alfred Elisabeth Stappers , Roger Petrus Gerebern Vandecruys , Paul Stoffels
- 申请人: Jérôme Emile Georges Guillemont , Paul Theodoor Agnes Stevens , Alex Herman Copmans , Jozef Peeters , Alfred Elisabeth Stappers , Roger Petrus Gerebern Vandecruys , Paul Stoffels
- 申请人地址: BE Beerse
- 专利权人: Janssen Pharmaceutica N.V.
- 当前专利权人: Janssen Pharmaceutica N.V.
- 当前专利权人地址: BE Beerse
- 代理商 Rajiv S. Shah
- 优先权: EPEP01203090 20010813; EPEP02077748 20020610; MYPI20043578 20040902; EPPCT/EP2004/052028 20040903; EP05101467 20050225
- 主分类号: A61K31/505
- IPC分类号: A61K31/505 ; C07D239/48 ; A61P31/18
摘要:
The present invention relates to a pharmaceutical composition comprising as active ingredient the hydrochloric acid salt of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethyl-phenyl]amino]-2-pyrimidinyl]amino]benzonitrile and to processes for their preparation.