Invention Grant
US08163937B2 Process for preparing (1R,2S,5S)-N-[(1S)-3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3-[(2S)-2-[[[(1,1-dimethylethyl)amino]-carbonyl]amino]-3,3-dimethyl-1-oxobutyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide
有权
制备（1R，2S，5S）-N - [（1S）-3-氨基-1-（环丁基甲基）-2,3-二氧代丙基] -3 - [（2S）-2 - [[ 1-二甲基乙基）氨基] - 羰基]氨基] -3,3-二甲基-1-氧代丁基] -6,6-二甲基-3-氮杂双环[3.1.0]己烷-2-甲酰胺
![Process for preparing (1R,2S,5S)-N-[(1S)-3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3-[(2S)-2-[[[(1,1-dimethylethyl)amino]-carbonyl]amino]-3,3-dimethyl-1-oxobutyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide](/docs/US/2012-04-24/US08163937B2/abs.jpg.600x600.jpg)
- Patent Title: Process for preparing (1R,2S,5S)-N-[(1S)-3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3-[(2S)-2-[[[(1,1-dimethylethyl)amino]-carbonyl]amino]-3,3-dimethyl-1-oxobutyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide
- Patent Title (中): 制备（1R，2S，5S）-N - [（1S）-3-氨基-1-（环丁基甲基）-2,3-二氧代丙基] -3 - [（2S）-2 - [[ 1-二甲基乙基）氨基] - 羰基]氨基] -3,3-二甲基-1-氧代丁基] -6,6-二甲基-3-氮杂双环[3.1.0]己烷-2-甲酰胺
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Application No.: US12519485Application Date: 2007-12-18
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Publication No.: US08163937B2Publication Date: 2012-04-24
- Inventor: George S. K. Wong , Hong-Chang Lee , Jennifer A. Vance , Weidong Tong , Tetsuo Iwama
- Applicant: George S. K. Wong , Hong-Chang Lee , Jennifer A. Vance , Weidong Tong , Tetsuo Iwama
- Applicant Address: US NJ Kenilworth
- Assignee: Schering Corporation
- Current Assignee: Schering Corporation
- Current Assignee Address: US NJ Kenilworth
- Agent Julie M. Lake; Sheldon O. Heber
- International Application: PCT/US2007/025804 WO 20071218
- International Announcement: WO2008/079216 WO 20080703
- Main IPC: C07D209/52
- IPC: C07D209/52
![Process for preparing (1R,2S,5S)-N-[(1S)-3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3-[(2S)-2-[[[(1,1-dimethylethyl)amino]-carbonyl]amino]-3,3-dimethyl-1-oxobutyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide](/abs-image/US/2012/04/24/US08163937B2/abs.jpg.150x150.jpg)
Abstract:
The present invention relates also to a process for the preparation of intermediate compounds useful in preparing the compounds of Formula (I) using the process of Scheme (II).
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