发明授权
- 专利标题： Fused polycyclic compounds having a heterocyclic ring(s) and pharmaceutical use thereof
- 专利标题（中）： 具有杂环的稠合多环化合物及其药物用途
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申请号： US13040882申请日： 2011-03-04
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公开(公告)号： US08299064B2公开(公告)日： 2012-10-30
- 发明人: Ryusuke Hirama , Seiji Niwa , Hideyuki Tanaka , Toshihiro Hatanaka , Yoko Masuzawa , Akiyo Yamazaki , Takao Ikenoue , Nobuo Kondo , Wataru Miyanaga , Masaru Takayanagi
- 申请人： Ryusuke Hirama , Seiji Niwa , Hideyuki Tanaka , Toshihiro Hatanaka , Yoko Masuzawa , Akiyo Yamazaki , Takao Ikenoue , Nobuo Kondo , Wataru Miyanaga , Masaru Takayanagi
- 申请人地址： JP Tokyo
- 专利权人： Ajinomoto Co., Inc.
- 当前专利权人： Ajinomoto Co., Inc.
- 当前专利权人地址： JP Tokyo
- 代理机构： Oblon, Spivak, McClelland, Maier & Neustadt, L.L.P.
- 优先权： JP2003-373270 20031031
- 主分类号： A61P3/10
- IPC分类号： A61P3/10 ; A61P3/04 ; A61P9/00 ; A61P13/12 ; A61P25/02 ; A61P27/02 ; A61K31/5517 ; C07D487/04
摘要：
The present invention provides a fused polycyclic compound of the following formula, analogues thereof and pharmaceutically acceptable salts thereof; and agents for increasing the sugar-transporting capacity, hypoglycemic agents and pharmaceutical compositions containing the above compounds. This fused polycyclic compound has high medicinal properties and few side-effects, and a therapeutic effect on diabetes. wherein R represents an alkoxy group, R′ represents an oxazolylpropionyl group or a thiazolylpropionyl group, and R″ represent a hydrogen atom.