Invention Grant
US08350086B2 Process for preparing cinacalcet hydrochloride 有权
盐酸西那卡塞的制备方法

  • Patent Title: Process for preparing cinacalcet hydrochloride
  • Patent Title (中): 盐酸西那卡塞的制备方法
  • Application No.: US12678971
    Application Date: 2008-09-18
  • Publication No.: US08350086B2
    Publication Date: 2013-01-08
  • Inventor: Mangion Bernardino
  • Applicant: Mangion Bernardino
  • Applicant Address: ES Barcelona
  • Assignee: Medichem, S.A.
  • Current Assignee: Medichem, S.A.
  • Current Assignee Address: ES Barcelona
  • Agency: Cozen O'Connor
  • International Application: PCT/US2008/076793 WO 20080918
  • International Announcement: WO2009/039241 WO 20090326
  • Main IPC: C07C211/00
  • IPC: C07C211/00
Process for preparing cinacalcet hydrochloride
Abstract:
The invention relates to an improved process for preparing cinacalcet hydrochloride. The invention provides an efficient and economic process for preparing cinacalcet hydrochloride which is suitable for industrial implementation i.e., affords cinacalcet hydrochloride with high purity, and uses small volumes of acidifying agent and solvents. The invention also related to a process for preparing a cinacalcet carboxylate salt, including cinacalcet accetate
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