Invention Grant
US08362012B2 Benzoxazine benzimidazole derivative, a pharmaceutical composition comprising the same, and a use thereof
有权
苯并恶嗪苯并咪唑衍生物，含有它们的药物组合物及其用途
- Patent Title: Benzoxazine benzimidazole derivative, a pharmaceutical composition comprising the same, and a use thereof
- Patent Title (中): 苯并恶嗪苯并咪唑衍生物，含有它们的药物组合物及其用途
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Application No.: US12934638Application Date: 2009-04-16
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Publication No.: US08362012B2Publication Date: 2013-01-29
- Inventor: Ji Duck Kim , Hong-Chul Yoon , Seong Hee Cho , Inwoo Kim , Min Jae Cho , In Young Lee , Hyae Jung Hyun , Eunkyung Park
- Applicant: Ji Duck Kim , Hong-Chul Yoon , Seong Hee Cho , Inwoo Kim , Min Jae Cho , In Young Lee , Hyae Jung Hyun , Eunkyung Park
- Applicant Address: KR Sungnam-si
- Assignee: Daewoong Pharmaceutical Co., Ltd.
- Current Assignee: Daewoong Pharmaceutical Co., Ltd.
- Current Assignee Address: KR Sungnam-si
- Agency: Seed IP Law Group PLLC
- Priority: KR10-2008-0036301 20080418
- International Application: PCT/KR2009/001977 WO 20090416
- International Announcement: WO2009/128661 WO 20091022
- Main IPC: C07D413/14
- IPC: C07D413/14 ; A61K31/538
Abstract:
The present invention relates to a novel benzoxazine benzimidazole derivative of formula (1) as an antagonist against a vanilloid receptor-1, a pharmaceutical composition comprising the same as an active ingredient, and a use thereof. The benzoxazine benzimidazole derivative of the present invention may be useful for preventing or treating a disease associated with antagonistic activity of vanilloid receptor-1: wherein, R1, R2, R3, R3′, Q1, Q2, Q3 and Q4 have same meanings as defined in the specification.
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