Invention Grant
- Patent Title: Azetidinyl diamides as monoacylglycerol lipase inhibitors
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Application No.: US12765076Application Date: 2010-04-22
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Publication No.: US08367653B2Publication Date: 2013-02-05
- Inventor: Haiyan Bian , Kristen Chevalier , Jose Clemente , Pete Connolly , Chris Flores , Shu-Chen Lin , Li Liu , John Mabus , Mark MacIelag , Mark McDonnell , Philip Pitis , Yue-Mei Zhang , Sui-Po Zhang , Bin Zhu
- Applicant: Haiyan Bian , Kristen Chevalier , Jose Clemente , Pete Connolly , Chris Flores , Shu-Chen Lin , Li Liu , John Mabus , Mark MacIelag , Mark McDonnell , Philip Pitis , Yue-Mei Zhang , Sui-Po Zhang , Bin Zhu
- Applicant Address: BE Beerse
- Assignee: Janssen Pharmaceutica NV
- Current Assignee: Janssen Pharmaceutica NV
- Current Assignee Address: BE Beerse
- Main IPC: A61K31/496
- IPC: A61K31/496 ; C07D401/12 ; C07D403/14 ; C07D417/12 ; C07D417/14 ; C07D487/04 ; C07D495/04

Abstract:
Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula (I) as follows: wherein Y, Z, R1, and s are defined herein.
Public/Granted literature
- US20100324013A1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS Public/Granted day:2010-12-23
Information query
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