发明授权
US08455550B2 Derivatives of aminocyclobutane or aminocyclobutene, their method of preparation and their use as medical products
有权
氨基环丁烷或氨基环丁烯的衍生物，其制备方法及其用作医药产品
- 专利标题： Derivatives of aminocyclobutane or aminocyclobutene, their method of preparation and their use as medical products
- 专利标题（中）： 氨基环丁烷或氨基环丁烯的衍生物，其制备方法及其用作医药产品
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申请号： US13258546申请日： 2010-04-02
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公开(公告)号： US08455550B2公开(公告)日： 2013-06-04
- 发明人: Stéphane Cuisiat , Adrian Newman-Tancredi , Olivier Vitton , Bernard Vacher
- 申请人： Stéphane Cuisiat , Adrian Newman-Tancredi , Olivier Vitton , Bernard Vacher
- 申请人地址： FR Boulogne-Billancourt
- 专利权人： Pierre Fabre Medicament
- 当前专利权人： Pierre Fabre Medicament
- 当前专利权人地址： FR Boulogne-Billancourt
- 代理机构： Birch, Stewart, Kolasch & Birch, LLP
- 优先权： FR0952196 20090403
- 国际申请： PCT/EP2010/054452 WO 20100402
- 国际公布： WO2010/112597 WO 20101007
- 主分类号： A61K31/165
- IPC分类号： A61K31/165 ; A61P25/00 ; C07C237/24
摘要：
The present invention concerns compounds of general formula (1), where in:—-a- is a single or double bond, Ar is an aromatic group, substituted or unsubstituted, R1 and R2 each independently or together are: a hydrogen atom or C1-C6 alkyl group, branched or unbranched, saturated or unsaturated, substituted or unsubstituted; the groups R1 and R2 may also form a heterocycle, R3 and R3′ each independently or together are a hydrogen atom or C1-C6 alkyl group, X is an oxygen atom or a sulphur atom, and the addition salts of the compounds of general formula (1) with pharmaceutically acceptable mineral acids or organic acids.