发明授权
US08691855B2 Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist and pharmaceutical compositions containing the same
有权
化合物，其异构体或其药学上可接受的盐作为香草素受体拮抗剂和含有它们的药物组合物
- 专利标题： Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist and pharmaceutical compositions containing the same
- 专利标题（中）： 化合物，其异构体或其药学上可接受的盐作为香草素受体拮抗剂和含有它们的药物组合物
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申请号： US13002289申请日： 2009-07-02
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公开(公告)号： US08691855B2公开(公告)日： 2014-04-08
- 发明人: Byoung Young Woo , Sun-Young Kim , Yeonjoon Kim , Song Seok Shin , Jin Kwan Kim , Ki-Wha Lee , Dong Hyun Kim , Kyung Min Lim , Joo-Hyun Moh , Yeon Su Jeong , Jin Kyu Choi , Hyun Ju Koh , Jeongho Lee , Hyuk Kim , Jeong Hoon Yoon , Funan Li , Jee-Suk Kim , Young-Ger Suh
- 申请人： Byoung Young Woo , Sun-Young Kim , Yeonjoon Kim , Song Seok Shin , Jin Kwan Kim , Ki-Wha Lee , Dong Hyun Kim , Kyung Min Lim , Joo-Hyun Moh , Yeon Su Jeong , Jin Kyu Choi , Hyun Ju Koh , Jeongho Lee , Hyuk Kim , Jeong Hoon Yoon , Funan Li , Jee-Suk Kim , Young-Ger Suh
- 申请人地址： KR Seoul
- 专利权人： Amorepacific Corporation
- 当前专利权人： Amorepacific Corporation
- 当前专利权人地址： KR Seoul
- 代理机构： Merchant & Gould P.C.
- 国际申请： PCT/KR2009/003627 WO 20090702
- 国际公布： WO2010/002209 WO 20100107
- 主分类号： C07D263/42
- IPC分类号： C07D263/42 ; C07D263/38 ; C07D307/52 ; C07D277/42
摘要：
This present invention relates to novel compounds, isomer thereof or pharmaceutically acceptable salts thereof as vanilloid receptor (Vanilloid Receptor 1; VR1; TRPV1) antagonist; and a pharmaceutical composition containing the same. The present invention provides a pharmaceutical composition for preventing or treating a disease such as pain, migraine, arthralgia, neuralgia, neuropathies, nerve injury, skin disorder, urinary bladder hypersensitiveness, irritable bowel syndrome, fecal urgency, a respiratory disorder, irritation of skin, eye or mucous membrane, stomach-duodenal ulcer, inflammatory diseases, ear disease, heart disease and so on.
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