Invention Grant
- Patent Title: Tricyclic azaindoles
- Patent Title (中): 三环azaindoles
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Application No.: US13140357Application Date: 2009-12-03
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Publication No.: US08853391B2Publication Date: 2014-10-07
- Inventor: Bayard R. Huck , Amanda E. Sutton , Benny C. Askew, Jr. , Christopher Charles Victor Jones , Garry R. Smith , Nadia Brugger
- Applicant: Bayard R. Huck , Amanda E. Sutton , Benny C. Askew, Jr. , Christopher Charles Victor Jones , Garry R. Smith , Nadia Brugger
- Applicant Address: DE Darmstadt
- Assignee: Merck Patent GmbH
- Current Assignee: Merck Patent GmbH
- Current Assignee Address: DE Darmstadt
- Agency: EMD Serono Research Institute
- Agent Thomas W. Brown
- International Application: PCT/US2009/066534 WO 20091203
- International Announcement: WO2010/080253 WO 20100715
- Main IPC: C07D401/14
- IPC: C07D401/14 ; C07D413/14 ; C07D471/14 ; C07D471/04

Abstract:
Disclosed are dipyridyl-pyrrole derivative compounds and analogs thereof, pharmaceutical compositions comprising such compounds and processes for preparing the same. The compounds are useful in the treatment of diseases amenable to protein kinase signal transduction inhibition, regulation and/or modulation.
Public/Granted literature
- US20120022060A1 Tricyclic Azaindoles Public/Granted day:2012-01-26
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