Invention Grant
- Patent Title: Process for preparing 1-phenylpyrazoles
- Patent Title (中): 1-苯基吡唑的制备方法
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Application No.: US13738230Application Date: 2013-01-10
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Publication No.: US08933246B2Publication Date: 2015-01-13
- Inventor: Maximilian Dochnahl , Gunter Lipowsky
- Applicant: BASF SE
- Applicant Address: DE Ludwigshafen
- Assignee: BASF SE
- Current Assignee: BASF SE
- Current Assignee Address: DE Ludwigshafen
- Agency: Brinks Gilson & Lione
- Priority: EP09169528 20090904
- Main IPC: C07D231/10
- IPC: C07D231/10 ; C07D231/20 ; C07D231/14

Abstract:
The present invention to a process for preparing 1-phenylpyrazoles of the formula I in which each R1 is independently selected from chlorine, fluorine, alkyl, haloalkyl, alkoxy and haloalkoxy; n is 1, 2 or 3; each R2 is independently selected from cyano, nitro, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio and alkoxycarbonyl; m is 0, 1 or 2; A is alkyl, aryl or aryl-C1-C4-alkyl, where A optionally bears 1, 2, 3 or 4 substituents comprising reacting a phenyl halide of the formula (II) with a pyrazole derivative of the formula (III) in which X is chlorine, iodine or bromine; and R1, n, R2, m and A are each as defined above, in the presence of a base and a catalytic system comprising a ligand and a metal compound selected from palladium compounds, iron compounds and copper compounds.
Public/Granted literature
- US20130131352A1 Process for Preparing 1-phenylpyrazoles Public/Granted day:2013-05-23
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