发明授权
- 专利标题： Octapeptide compounds and therapeutic use thereof
- 专利标题（中）： 八肽化合物及其治疗用途
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申请号： US13806510申请日： 2011-06-21
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公开(公告)号： US09040482B2公开(公告)日： 2015-05-26
- 发明人: Jean-Christophe Cintrat , Melinda Ligeti , Bernard Rousseau , Franck Artzner , Christophe Tarabout , Marie-Thérèse Paternostre , Nicolas Fay , Roland Cherif-Cheikh , Céline Valery
- 申请人： Jean-Christophe Cintrat , Melinda Ligeti , Bernard Rousseau , Franck Artzner , Christophe Tarabout , Marie-Thérèse Paternostre , Nicolas Fay , Roland Cherif-Cheikh , Céline Valery
- 申请人地址： FR Boulogne-Billancourt FR Paris FR Paris
- 专利权人： IPSEN PHARMA S.A.S.,COMMISSARIAT A L'ENERGIE ATOMIQUE (C.E.A.),CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.)
- 当前专利权人： IPSEN PHARMA S.A.S.,COMMISSARIAT A L'ENERGIE ATOMIQUE (C.E.A.),CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.)
- 当前专利权人地址： FR Boulogne-Billancourt FR Paris FR Paris
- 代理机构： Hunton & Williams LLP
- 优先权： EP10290336 20100622
- 国际申请： PCT/FR2011/000352 WO 20110621
- 国际公布： WO2011/161332 WO 20111229
- 主分类号： C07K14/655
- IPC分类号： C07K14/655 ; A61K38/31 ; A61P5/02 ; C07K7/54 ; A61K38/00
摘要：
The present invention relates to novel octapeptide compounds of general formula (I), R-AA1-cyclo(AA2-Tyr3-D-Trp4-AA5-Val6-Cys7)-Thr8-NH2 (I) As these products have a good affinity for certain sub-types of somatostatin receptors, they are particularly useful for treating the pathological states or diseases in which one (or more) of the somatostatin receptors is (are) involved. The invention also relates to pharmaceutical compositions containing said products and their use for the preparation of a medicament.
公开/授权文献
- US20130252892A1 NOVEL OCTAPEPTIDE COMPOUNDS AND THERAPEUTIC USE THEREOF 公开/授权日：2013-09-26
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