Invention Grant
- Patent Title: Substituted pyrido[3,4-b]pyrazines as GPR6 modulators
- Patent Title (中): 取代的吡啶并[3,4-b]吡嗪作为GPR6调节剂
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Application No.: US14577480Application Date: 2014-12-19
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Publication No.: US09181249B2Publication Date: 2015-11-10
- Inventor: Jason Brown , Steve Hitchcock , Maria Hopkins , Shota Kikuchi , Holger Monenschein , Holly Reichard , Kristin Schleicher , Huikai Sun , Todd Macklin
- Applicant: Takeda Pharmaceutical Company Limited
- Applicant Address: JP Osaka
- Assignee: Takeda Pharmaceutical Company Limited
- Current Assignee: Takeda Pharmaceutical Company Limited
- Current Assignee Address: JP Osaka
- Agent David M. Stemerick; Matthew J. Russo
- Main IPC: A61K31/4965
- IPC: A61K31/4965 ; C07D471/04
![Substituted pyrido[3,4-b]pyrazines as GPR6 modulators](/abs-image/US/2015/11/10/US09181249B2/abs.jpg.150x150.jpg)
Abstract:
The present invention provides compounds of formula I: which are useful as modulators of GPR6, pharmaceutical compositions thereof, methods for treatment of conditions associated with GPR6, processes for making the compounds and intermediates thereof.
Public/Granted literature
- US20150175602A1 TETRAHYDROPYRIDOPYRAZINES MODULATORS OF GPR6 Public/Granted day:2015-06-25
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