Invention Grant
US09273067B2 Pyrazolopyrimidine macrocycles as inhibitors of human immunodeficiency virus replication
有权
吡唑并嘧啶大环化合物作为人类免疫缺陷病毒复制的抑制剂
- Patent Title: Pyrazolopyrimidine macrocycles as inhibitors of human immunodeficiency virus replication
- Patent Title (中): 吡唑并嘧啶大环化合物作为人类免疫缺陷病毒复制的抑制剂
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Application No.: US14619728Application Date: 2015-02-11
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Publication No.: US09273067B2Publication Date: 2016-03-01
- Inventor: B. Narasimhulu Naidu , Michael A. Walker , Margaret E. Sorenson , Manoj Patel , Zhizhen Barbara Zheng , John F. Kadow , Bin Zheng , Martin D. Eastgate , Ke Chen , Francisco Gonzalez-Bobes
- Applicant: BRISTOL-MYERS SQUIBB COMPANY
- Applicant Address: US NJ Princeton
- Assignee: Bristol-Myers Squibb Company
- Current Assignee: Bristol-Myers Squibb Company
- Current Assignee Address: US NJ Princeton
- Agent James Epperson
- Main IPC: C07D498/22
- IPC: C07D498/22 ; C07D211/48

Abstract:
The disclosure generally relates to compounds of formula I, including compositions and methods for treating human immunodeficiency virus (HIV) infection. The disclosure provides novel inhibitors of HIV, pharmaceutical compositions containing such compounds, and methods for making and using these compounds in the treatment of HIV infection.
Public/Granted literature
- US20150232481A1 Pyrazolopyrimidine Macrocycles as Inhibitors of Human Immunodeficiency Virus Replication Public/Granted day:2015-08-20
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