Invention Application
- Patent Title: COMPOUNDS AND THEIR USE IN A METHOD FOR MODULATING AR (ANDROGEN RECEPTOR) TRANSCRIPTIONAL ACTIVITY
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Application No.: PCT/EP2021/076120Application Date: 2021-09-22
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Publication No.: WO2023046283A1Publication Date: 2023-03-30
- Inventor: SALVATELLA GIRALT, Xavier , RIERA ESCALÉ, Antoni , FRIGOLÉ VIVAS, Marta , SÁNCHEZ ZARZALEJO, Carolina , RUFFONI, Alessandro , VERDAGUER ESPAULELLA, Francesc Xavier , SADAR, Marianne Dorothy , BANUELOS, Carmen Adriana , MAWJI, Nasrin
- Applicant: FUNDACIÓ INSTITUT DE RECERCA BIOMÈDICA (IRB BARCELONA) , UNIVERSITAT DE BARCELONA , INSTITUCIÓ CATALANA DE RECERCA I ESTUDIS AVANÇATS , PROVINCIAL HEALTH SERVICES AUTHORITY
- Applicant Address: Baldiri Reixac 10; Centro de Patentes de la UB; Passeig Lluís Companys, 23; 675 West 10th Avenue
- Assignee: FUNDACIÓ INSTITUT DE RECERCA BIOMÈDICA (IRB BARCELONA),UNIVERSITAT DE BARCELONA,INSTITUCIÓ CATALANA DE RECERCA I ESTUDIS AVANÇATS,PROVINCIAL HEALTH SERVICES AUTHORITY
- Current Assignee: FUNDACIÓ INSTITUT DE RECERCA BIOMÈDICA (IRB BARCELONA),UNIVERSITAT DE BARCELONA,INSTITUCIÓ CATALANA DE RECERCA I ESTUDIS AVANÇATS,PROVINCIAL HEALTH SERVICES AUTHORITY
- Current Assignee Address: Baldiri Reixac 10; Centro de Patentes de la UB; Passeig Lluís Companys, 23; 675 West 10th Avenue
- Agency: HOFFMANN EITLE S.L.U.
- Main IPC: A61K31/09
- IPC: A61K31/09 ; A61K31/519 ; A61P5/26 ; A61P5/28 ; A61P35/00
Abstract:
The present invention relates to compounds of formula (I) and their use for modulating the transcriptional activity of the androgen receptor and its splice variants for treating various indications including prostate cancer
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