Het is pyridinyl, pyrimidinyl, thiophenyl, furyl, isothiazolyl or isoxazolyl, each being substituted by groups R 4 , R 5 and R 6 ; R 1 is hydrogen or halo; R 2 is hydrogen or halo; R 3 is optionally substituted C 2-12 alkyl, optionally substituted C 2-12 alkenyl, optionally substituted C 2-12 alkynyl, optionally substituted C 3-12 cycloalkyl, optionally substituted phenyl or optionally substituted heterocyclyl; and R 4 , R 5 and R 6 are, independently, selected from hydrogen, halo, cyano, nitro, C 1-4 alkyl, C 1-4 haloalkyl, C 1-4 alkoxy(C 1-4 )alkyl and C 1-4 haloalkoxy(C 1-4 )alkyl, provided that at least one of R 4 , R 5 and R 6 is not hydrogen. The compounds of formula (I) have plant-protective properties and are suitable for protecting plants against infestations by phytopathogenic microorganisms.
Het is pyridinyl, pyrimidinyl, thiophenyl, furyl, isothiazolyl or isoxazolyl, each being substituted by groups R 4 , R 5 and R 6 ; R 1 is hydrogen or halo; R 2 is hydrogen or halo; R 3 is optionally substituted C 2-12 alkyl, optionally substituted C 2-12 alkenyl, optionally substituted C 2-12 alkynyl, optionally substituted C 3-12 cycloalkyl, optionally substituted phenyl or optionally substituted heterocyclyl; and R 4 , R 5 and R 6 are, independently, selected from hydrogen, halo, cyano, nitro, C 1-4 alkyl, C 1-4 haloalkyl, C 1-4 alkoxy(C 1-4 )alkyl and C 1-4 haloalkoxy(C 1-4 )alkyl, provided that at least one of R 4 , R 5 and R 6 is not hydrogen. The compounds of formula (I) have plant-protective properties and are suitable for protecting plants against infestations by phytopathogenic microorganisms.
摘要翻译:式(I)的化合物:Het是吡啶基,嘧啶基,噻吩基,呋喃基,异噻唑基或异恶唑基,各自被基团R 4,R 5和R 6取代; R 1是氢或卤素; R 2是氢或卤素; R 3是任选取代的C 2-12烷基,任选取代的C 2-12烯基,任选取代的C 2-12炔基,任选取代的C 3-12环烷基,任选取代的苯基或任选取代的杂环基; 和R 4,R 5和R 6独立地选自氢,卤素,氰基,硝基,C 1-4烷基,C 1-4卤代烷基,C 1-4烷氧基(C 1-4)烷基和C 1 -4-卤代烷氧基(C 1-4)烷基,条件是R 4,R 5和R 6中的至少一个不是氢。 式(I)化合物具有植物保护性质,并且适用于通过植物病原微生物保护植物免受侵袭。
摘要:
The invention relates to novel 2-alkyl-cycloalk(en)yl-carboxamides of formula (I), in which X, s, R1, L, R2 and A are defined as cited in the description, to several methods for producing said substances and to the use of the latter for controlling undesired micro-organisms. The invention also relates to novel intermediate products and to the production of said products.
摘要翻译:2-烷基 - 环烷基(烯)基 - 甲酰胺化合物(I)是新的。 式(A-CO-N(R 1))-L-CH 2(R 2) - (CH 2)s-X的2-烷基 - 环烷基(烯) - 甲酰胺化合物(I)是新的。 X:-CR 3> R 4> R 5>或-SiR 49> R 50> R 51>; s:1-2; R 1 H,1-8C烷基,1-6C烷基亚磺酰基,1-6C烷基磺酰基,1-4C烷氧基1-4C-烷基,3-8C环烷基,1-6C卤代烷基,1-4C卤代烷硫基,1-4C卤代烷基亚磺酰基 ,1-4C卤代烷基磺酰基,卤代1-4C-烷氧基 - 1-4C-烷基,3-8C卤代环烷基(具有1-9的F,Cl和/或Br),甲酰基,甲酰基1-3C-烷基,( (1-3C-烷氧基)羰基,1-3C-烷基,卤代(1-3C-烷基)羰基,1-3C-烷基,卤代(1 (1-8C-烷基)羰基,(1-8C-烷氧基)羰基,(1-4C-烷氧基)羰基, 烷氧基-1C 1-4烷基)羰基,(3-8C-环烷基)羰基,(1-6C-卤代烷基)羰基,(1-6C-卤代烷氧基)羰基,(卤代1-4C-烷氧基1-4C- 烷基)羰基,(3-8C-卤代环烷基)羰基(具有F,Cl和/或Br的1-9),-C(= O)C(= O)R 6,-CONR 7 R 8或 -CH 2 NR 9 R 10; L:L 1>或L 2>; (3-7C-环烷基-1,2-二基)(任选被F,Cl,1-4C烷基或1-4C卤代烷基的1-4取代); (环己二烯基)(任选被F,Cl,1-4C烷基或1-4C卤代烷基的1-4取代); R 2> H,卤素,1-4C烷基或具有1-9个F,Cl和/或Br的1-4C卤代烷基; R 3>卤素,1-8C烷基或1-6C卤代烷基,其中1-13个F,Cl和/或Br; 和R 4>卤素,1-8C烷基或1-6C卤代烷基,其中1-13个F,Cl和/或Br; 或任选被不饱和的碳环或杂环(任选被卤素,1-4C烷基,1-4C烷氧基,1-4C卤代烷基或1-4C卤代烷氧基取代)取代;或者R 3' R 5> H,卤素,1-8C烷基或1-6C卤代烷基,其中1-13个F,Cl和/或Br; R 49>,R 50> H,1-8C烷基,1-8C烷氧基,1-4C烷氧基1-4C-烷基,1-4C烷硫基1-4C-烷基或1-6C卤代烷基; R 51>苯基,苯基烷基(均为任意取代的),H,1-8C烷基,1-8C烷氧基,1-4C烷氧基-14C-烷基,1-4C-烷硫基1-4C-烷基,2-8C 烯基,2-8C-炔基,1-6C卤代烷基,2-6C卤代烯基,2-6C卤代炔基或3-6C环烷基; R 6> H,1-8C烷基,1-8C烷氧基,1-4C烷氧基1-4C-烷基,3-8C环烷基,1-6C卤代烷基,1-6C卤代烷氧基,卤代1-4C-烷氧基-1 -4C-烷基或具有1-9个F,Cl和/或Br的3-8C-卤代环烷基; R 7> R 8> H,1-8C烷基,1-4C烷氧基1-4C-烷基,3-8C环烷基,1-8C卤代烷基,卤代1-4C-烷氧基-1-4C-烷基或 具有1-9个F,Cl和/或Br的3-8C-卤代环烷基; 或任选地被一个或多个卤素或1-4C烷基取代的NR 7> R 8> 5-8元饱和杂环(任选地含有1-2个另外不相邻的O,S或NR 11的杂原子) R 9> R 10> H,1-8C烷基,3-8C环烷基,1-8C卤代烷基或具有1-9个F,Cl和/或Br的3-8C-卤代环烷基; 或NR 9> R 10> 5-8元饱和杂环(任选地含有1-2个其它非相邻的O,S或NR 11的杂原子),任选被卤素或1-4C烷基取代; H或1-6C烷基; A:19(杂)环基,例如 式(1)的苯基化合物,式(2)的吡啶化合物和式(3)的硫代化合物; R 21> H,卤素,OH,CN,1-6C烷基; 或1-4C卤代烷基,1-4C卤代烷氧基或1-4C卤代烷硫基,每个具有1-5个卤素原子; R 22> H,卤素,OH,CN,1-4C烷基,1-4C烷氧基,1-4C烷硫基; 或1-4C卤代烷基,1-4C卤代烷硫基或1-4C卤代烷氧基,每个具有1-5个卤素原子; R 23> H,卤素,OH,CN,1-4C烷基,1-4C烷氧基,1-4C烷硫基; 或1-4C卤代烷基,1-4C卤代烷氧基,每个具有1-5个卤素原子,1-4C-烷基亚磺酰基或1-4C烷基磺酰基; 和R 26> 1-4C烷基或具有1-5个卤素原子的1-4C卤代烷基。 还包括:(1)(I)的准备; (2)用于防治不想要的微生物的试剂,至少包含(I)稀释剂和/或表面活性剂; (3)防治不需要的微生物的方法,包括在微生物和/或其栖息地上施用(I)稀释剂和/或表面活性剂。 活性:抗菌; 抗真菌。 行动机制:无给予。
摘要:
A composition comprising at least a pyridylmethylbenzamide derivative of general formula (I) and 5,10-dihydro-5,10-dioxonaphtho[2,3-b]-1,4-dithiine-2,3-dicarbonitrile; in an (a) / (b) weight ratio of from 0.01 to 10. A composition further comprising an additional fungicidal compound. A method for preventively or curatively combating the phytopathogenic fungi of crops by using this composition.
摘要:
The present invention provides an at least binary composition for controlling nematodes and insects or representatives of the order Acarina, which composition comprises: (A) a nernaticidally effective amount of at least one macrolide, and (B) an insecticidally effective amount of at least one insecticide selected from the neonicotinoids.
摘要:
The invention relates to novel hexyl carboxanilides of formula (I), in which L, R1, R3 and A are defined as cited in the description, to several methods for producing said substances, to their use for controlling undesirable micro-organisms and to novel intermediate products and the production thereof.
摘要:
A method for treating plants in need of growth promotion, comprising applying to said plants, to the seeds from which they grow or to the locus in which they grow, a non-phytotoxic, effective plant growth promoting amount of an amide compound having the formula A-CO-NR1R2 in which A is an aryl group or an aromatic or non-aromatic, 5- or 6-membered heterocycle which has from 1 to 3 hetero atoms which are selected from O, N and S; where the aryl group or the heterocycle may or may not have 1, 2 or 3 substituents which are selected, independently of one another, from alkyl, halogen, CHF2, CF3, alkoxy, haloalkoxy, alkylthio, alkylsulfinyl and alkylsulfonyl; R1 is a hydrogen atom; R2 is a phenyl or cycloalkyl group which may or may not have 1, 2 or 3 substituents which are selected, independently of one another, from alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkyl, cycloalkenyl, cycloalkyloxy, cycloal- kenyloxy, phenyl and halogen, where the aliphatic and cycloaliphatic radicals may be partially or fully halogenated and/or the cycloaliphatic radicals may be substituted by from 1 to 3 alkyl groups and where the phenyl group may have from 1 to 5 halogen atoms and/or from 1 to 3 substituents which are selected, in dependently of one another, from alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio and haloalkylthio, and where the amidic phenyl group may or may not be condensed with a saturated 5-membered ring which may or may not be substituted by one or more alkyl groups and/or may have a hetero atom selected from O and S.
摘要:
Certain novel phenyl substituted cyclic derivatives have unexpected insecticidal activity. These compounds are represented by formula (I): where B is a cyclic bridging group containing at least one N or N oxide link and a, A, b, B, c, d, D, L, M, R1 through R9, inclusively, and R13, R14 and R15 are fully described herein. In addition, novel intermediates useful in preparing compounds of Formula (I), compositions comprising an insecticidally effective amount of at least one compound of formula (I), and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要:
A composition comprising an organic carbonate such as propylene carbonate and O,O-diethyl-O-(2-isopropyl-4-methyl-6-pyrimidinyl)phosphorothioate, S-[1,2-bis(ethoxycarbonyl)ethyl]O,O-dimethylphosphorodithioate, or 6,7,8,9,10,10-hexachloro-1,5,5a,6,9,9a-hexahydro-6,9-methano-2,4,3-benzodioxathiepin-3-oxide, and methods thereof.