2-ALKYL-CYCLOALK(EN)YL-CARBOXAMIDE
    63.
    发明公开
    2-ALKYL-CYCLOALK(EN)YL-CARBOXAMIDE 审中-公开
    2-烷基环烷(烯)基甲酰胺

    公开(公告)号:EP1824836A2

    公开(公告)日:2007-08-29

    申请号:EP05819324.4

    申请日:2005-12-08

    摘要: The invention relates to novel 2-alkyl-cycloalk(en)yl-carboxamides of formula (I), in which X, s, R1, L, R2 and A are defined as cited in the description, to several methods for producing said substances and to the use of the latter for controlling undesired micro-organisms. The invention also relates to novel intermediate products and to the production of said products.

    摘要翻译: 2-烷基 - 环烷基(烯)基 - 甲酰胺化合物(I)是新的。 式(A-CO-N(R 1))-L-CH 2(R 2) - (CH 2)s-X的2-烷基 - 环烷基(烯) - 甲酰胺化合物(I)是新的。 X:-CR 3> R 4> R 5>或-SiR 49> R 50> R 51>; s:1-2; R 1 H,1-8C烷基,1-6C烷基亚磺酰基,1-6C烷基磺酰基,1-4C烷氧基1-4C-烷基,3-8C环烷基,1-6C卤代烷基,1-4C卤代烷硫基,1-4C卤代烷基亚磺酰基 ,1-4C卤代烷基磺酰基,卤代1-4C-烷氧基 - 1-4C-烷基,3-8C卤代环烷基(具有1-9的F,Cl和/或Br),甲酰基,甲酰基1-3C-烷基,( (1-3C-烷氧基)羰基,1-3C-烷基,卤代(1-3C-烷基)羰基,1-3C-烷基,卤代(1 (1-8C-烷基)羰基,(1-8C-烷氧基)羰基,(1-4C-烷氧基)羰基, 烷氧基-1C 1-4烷基)羰基,(3-8C-环烷基)羰基,(1-6C-卤代烷基)羰基,(1-6C-卤代烷氧基)羰基,(卤代1-4C-烷氧基1-4C- 烷基)羰基,(3-8C-卤代环烷基)羰基(具有F,Cl和/或Br的1-9),-C(= O)C(= O)R 6,-CONR 7 R 8或 -CH 2 NR 9 R 10; L:L 1>或L 2>; (3-7C-环烷基-1,2-二基)(任选被F,Cl,1-4C烷基或1-4C卤代烷基的1-4取代); (环己二烯基)(任选被F,Cl,1-4C烷基或1-4C卤代烷基的1-4取代); R 2> H,卤素,1-4C烷基或具有1-9个F,Cl和/或Br的1-4C卤代烷基; R 3>卤素,1-8C烷基或1-6C卤代烷基,其中1-13个F,Cl和/或Br; 和R 4>卤素,1-8C烷基或1-6C卤代烷基,其中1-13个F,Cl和/或Br; 或任选被不饱和的碳环或杂环(任选被卤素,1-4C烷基,1-4C烷氧基,1-4C卤代烷基或1-4C卤代烷氧基取代)取代;或者R 3' R 5> H,卤素,1-8C烷基或1-6C卤代烷基,其中1-13个F,Cl和/或Br; R 49>,R 50> H,1-8C烷基,1-8C烷氧基,1-4C烷氧基1-4C-烷基,1-4C烷硫基1-4C-烷基或1-6C卤代烷基; R 51>苯基,苯基烷基(均为任意取代的),H,1-8C烷基,1-8C烷氧基,1-4C烷氧基-14C-烷基,1-4C-烷硫基1-4C-烷基,2-8C 烯基,2-8C-炔基,1-6C卤代烷基,2-6C卤代烯基,2-6C卤代炔基或3-6C环烷基; R 6> H,1-8C烷基,1-8C烷氧基,1-4C烷氧基1-4C-烷基,3-8C环烷基,1-6C卤代烷基,1-6C卤代烷氧基,卤代1-4C-烷氧基-1 -4C-烷基或具有1-9个F,Cl和/或Br的3-8C-卤代环烷基; R 7> R 8> H,1-8C烷基,1-4C烷氧基1-4C-烷基,3-8C环烷基,1-8C卤代烷基,卤代1-4C-烷氧基-1-4C-烷基或 具有1-9个F,Cl和/或Br的3-8C-卤代环烷基; 或任选地被一个或多个卤素或1-4C烷基取代的NR 7> R 8> 5-8元饱和杂环(任选地含有1-2个另外不相邻的O,S或NR 11的杂原子) R 9> R 10> H,1-8C烷基,3-8C环烷基,1-8C卤代烷基或具有1-9个F,Cl和/或Br的3-8C-卤代环烷基; 或NR 9> R 10> 5-8元饱和杂环(任选地含有1-2个其它非相邻的O,S或NR 11的杂原子),任选被卤素或1-4C烷基取代; H或1-6C烷基; A:19(杂)环基,例如 式(1)的苯基化合物,式(2)的吡啶化合物和式(3)的硫代化合物; R 21> H,卤素,OH,CN,1-6C烷基; 或1-4C卤代烷基,1-4C卤代烷氧基或1-4C卤代烷硫基,每个具有1-5个卤素原子; R 22> H,卤素,OH,CN,1-4C烷基,1-4C烷氧基,1-4C烷硫基; 或1-4C卤代烷基,1-4C卤代烷硫基或1-4C卤代烷氧基,每个具有1-5个卤素原子; R 23> H,卤素,OH,CN,1-4C烷基,1-4C烷氧基,1-4C烷硫基; 或1-4C卤代烷基,1-4C卤代烷氧基,每个具有1-5个卤素原子,1-4C-烷基亚磺酰基或1-4C烷基磺酰基; 和R 26> 1-4C烷基或具有1-5个卤素原子的1-4C卤代烷基。 还包括:(1)(I)的准备; (2)用于防治不想要的微生物的试剂,至少包含(I)稀释剂和/或表面活性剂; (3)防治不需要的微生物的方法,包括在微生物和/或其栖息地上施用(I)稀释剂和/或表面活性剂。 活性:抗菌; 抗真菌。 行动机制:无给予。

    METHOD OF PLANT GROWTH PROMOTION USING AMIDE COMPOUNDS
    67.
    发明公开
    METHOD OF PLANT GROWTH PROMOTION USING AMIDE COMPOUNDS 有权
    程序对促进植物生长USING酰胺化合物

    公开(公告)号:EP1659864A2

    公开(公告)日:2006-05-31

    申请号:EP04763247.6

    申请日:2004-07-15

    摘要: A method for treating plants in need of growth promotion, comprising applying to said plants, to the seeds from which they grow or to the locus in which they grow, a non-phytotoxic, effective plant growth promoting amount of an amide compound having the formula A-CO-NR1R2 in which A is an aryl group or an aromatic or non-aromatic, 5- or 6-membered heterocycle which has from 1 to 3 hetero atoms which are selected from O, N and S; where the aryl group or the heterocycle may or may not have 1, 2 or 3 substituents which are selected, independently of one another, from alkyl, halogen, CHF2, CF3, alkoxy, haloalkoxy, alkylthio, alkylsulfinyl and alkylsulfonyl; R1 is a hydrogen atom; R2 is a phenyl or cycloalkyl group which may or may not have 1, 2 or 3 substituents which are selected, independently of one another, from alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkyl, cycloalkenyl, cycloalkyloxy, cycloal- kenyloxy, phenyl and halogen, where the aliphatic and cycloaliphatic radicals may be partially or fully halogenated and/or the cycloaliphatic radicals may be substituted by from 1 to 3 alkyl groups and where the phenyl group may have from 1 to 5 halogen atoms and/or from 1 to 3 substituents which are selected, in dependently of one another, from alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio and haloalkylthio, and where the amidic phenyl group may or may not be condensed with a saturated 5-membered ring which may or may not be substituted by one or more alkyl groups and/or may have a hetero atom selected from O and S.