公开(公告)号：EP2262794A1

公开(公告)日：2010-12-22

申请号：EP09713047.0

申请日：2009-02-12

Applicant: BASF SE

Inventor： GRAMMENOS, Wassilios ,  LOHMANN, Jan Klaas ,  GROTE, Thomas ,  DIETZ, Jochen ,  MÜLLER, Bernd ,  PUHL, Michael ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  VRETTOU, Marianna ,  RHEINHEIMER, Joachim

IPC: C07D401/14 ,  C07D417/14 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78

CPC classification number: C07D417/14 ,  A01N43/10 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/60 ,  A01N43/653 ,  A01N43/76 ,  A01N43/78 ,  C07D401/14

Abstract: The present invention relates to pyridin-4-ylmethyl-sulfonamides of formula (I), wherein R
a , n, R, A,Y and Het are as defined in the claims, and to the N-oxides, and salts thereof and their use for combating harmful fungi, and also to compositions and seed comprising at least one such compound. The invention also relates to a process and intermediates for preparing these compounds.

公开(公告)号：EP2224812A2

公开(公告)日：2010-09-08

申请号：EP08861013.4

申请日：2008-12-15

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GROTE, Thomas ,  MÜLLER, Bernd ,  LOHMANN, Jan Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  GLÄTTLI, Alice ,  VRETTOU, Marianna

IPC: A01N43/653 ,  C07D407/06 ,  C07D407/14 ,  C07F9/40 ,  A61K31/4025 ,  A61P31/00 ,  C07D303/12 ,  C07D303/36 ,  C07D303/08

CPC classification number: A01N43/653 ,  C07D303/36 ,  C07D405/06 ,  C07F9/65586

Abstract: The invention relates to the triazolylmethyloxiranes of formula (I), wherein variables D and B have the meanings as defined in the description and the claims.

公开(公告)号：EP2035414B1

公开(公告)日：2009-12-16

申请号：EP07730149.7

申请日：2007-06-14

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GROTE, Thomas ,  MÜLLER, Bernd ,  LOHMANN, Jan Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  GLÄTTLI, Alice

IPC: C07D405/06 ,  A01N43/653

CPC classification number: C07D405/06

Abstract: The present invention relates to azolylmethyloxiranes of the general formula I, in which A is phenyl substituted by three F, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl, or is phenyl substituted by from one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to their acid addition or metal salts compatible with plants, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising them.

公开(公告)号：EP2041122B1

公开(公告)日：2009-11-25

申请号：EP07765658.5

申请日：2007-06-27

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GROTE, Thomas ,  MÜLLER, Bernd ,  LOHMANN, Jan Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  GLÄTTLI, Alice

IPC: C07D405/14 ,  A01N43/653

CPC classification number: C07D405/14 ,  A01N43/653

Abstract: The invention relates to azolylmethyloxiranes of general formula (I), wherein A or B represent a 6-membered heteroaryl, selected from pyridinyl, pyrimidinyl, pyrazinyl, pyridazinyl and triazinyl, which is substituted by one to three of the following substituents: halogen, NO2, amine, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy, C1-C4 alkylamino, C1-C4 dialkylamino, thio or C1-C4 alkylthio, and the respective other substituent A or B represents phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amine, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy, C1-C4 alkylamino, C1-C4 dialkylamino, thio or C1-C4 alkylthio, and to the acid addition or metal salts thereof that are tolerated by plants. The invention also relates to the use of the compounds of formula (I) for controlling phytopathogenic fungi and to agents containing said compounds.

Abstract translation: 本发明涉及通式（I）的唑基甲基环氧乙烷，其中A或B代表选自吡啶基，嘧啶基，吡嗪基，哒嗪基和三嗪基的6元杂芳基，其被以下取代基中的1-3个取代：卤素，NO 2 ，胺，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4二烷基氨基，硫代或C 1 -C 4烷硫基，并且各别的取代基A或B代表苯基 其任选被1-3个以下取代基取代：卤素，NO 2，胺，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4二烷基氨基， 或C 1 -C 4烷硫基，并且涉及植物耐受的酸加成或其金属盐。 本发明还涉及式（I）化合物用于防治植物病原性真菌的用途和含有所述化合物的药剂的用途。

公开(公告)号：EP2096921A1

公开(公告)日：2009-09-09

申请号：EP07847722.1

申请日：2007-12-04

Applicant: BASF SE

Inventor： RENNER, Jens ,  GROTE, Thomas ,  MÜLLER, Bernd ,  LOHMANN, Jan, Klaas ,  ULMSCHNEIDER, Sarah ,  GLÄTTLI, Alice ,  DIETZ, Jochen

IPC: A01N43/653 ,  C07D405/06

CPC classification number: C07D405/06 ,  A01N43/653

Abstract: The present invention relates to azolylmethyloxiranes of the general formula (I) in which A stands for phenyl which is optionally substituted by one to three of the following substituents: halogen,NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, with the proviso that A does not stand for 2-methylphenyl, and also their plant-compatible acid addition salts or metal salts, and also to the use of the compounds of the formula I for controlling phytopathogenic fungi, and to compositions comprising them.

Abstract translation: 本发明涉及通式（I）的唑基甲基环氧乙烷，其中A代表任选被1-3个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4烷氧基， C1-C4-卤代烷基，C1-C4-卤代烷氧基，C1-C4-烷基氨基，C1-C4-二烷基氨基，硫代或C1-C4-烷硫基，条件是A不代表2-甲基苯基， 相容的酸加成盐或金属盐，并且还涉及式I化合物用于防治植物病原性真菌的用途，以及包含它们的组合物。

公开(公告)号：EP2046794A1

公开(公告)日：2009-04-15

申请号：EP07787081.4

申请日：2007-07-05

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GRAMMENOS, Wassilios ,  MÜLLER, Bernd ,  LOHMANN, Jan Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  VRETTOU,Marianna

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to azolopyrimidines of formula (I), wherein the substituents are defined as indicated in the description, methods and intermediate products for producing said compounds, substances containing the same, and the use thereof for controlling plant-pathogenic fungi.

公开(公告)号：EP2046784A2

公开(公告)日：2009-04-15

申请号：EP07787619.1

申请日：2007-07-17

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GROTE, Thomas ,  MÜLLER, Bernd ,  LOHMANN, Jan Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  GLÄTTLI, Alice

IPC: C07D405/14 ,  C07D409/14 ,  A01N43/707

CPC classification number: C07D405/14 ,  A01N43/653 ,  C07D409/14

Abstract: The invention relates to azolylmethyloxiranes of general formula (I), wherein A or B is benzodioxolyl which is optionally substituted by between one and five of the following substituents, halogen, CN, NO2, amino, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy, C1-C4 alkylamino, C1-C4 dialkylamino, thio or C1-C4 alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, said substituents being optionally substituted by between one and three of the following substituents, halogen, CN, NO2, amino, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy, C1-C4 alkylamino, C1-C4 dialkylamino, thio or C1-C4 alkylthio. The invention also relates to the plant-tolerant acid addition salts or metal salts of said compounds, to the use of the compounds of formula (I) for controlling plant-pathogenic fungi, and to agents containing the same.

公开(公告)号：EP2046780A1

公开(公告)日：2009-04-15

申请号：EP07787668.8

申请日：2007-07-18

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GROTE, Thomas ,  MÜLLER, Bernd ,  LOHMANN, Jan Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  GLÄTTLI, Alice

IPC: C07D405/06 ,  A01N43/653

CPC classification number: C07D405/06

Abstract: The invention relates to azolylmethyloxiranes of general formula (I) wherein A or B is phenyl which is substituted with a CN and optionally by between one and three of the following substituents, halogen, NO2, amino, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy, C1-C4 alkylamino, C1-C4 dialkylamino, thio or C1-C4 alkylthio, and the respective other substituent A or B is phenyl or a 5-membered or 6-membered heteroaryl, said substituents being optionally substituted by between one and three of the following substituents, halogen, CN, NO2, amino, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy, C1-C4 alkylamino, C1-C4 dialkylamino, thio or C1-C4 alkylthio. The invention also relates to the plant-tolerant acid addition salts or metal salts of said compounds, to the use of compounds of formula (I) for controlling plant pathogenic fungi, and to agents containing the same.

Abstract translation: 本发明涉及通式（I）的唑基甲基环氧乙烷，其中A或B是被CN取代的苯基和任选地一至三个下列取代基：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4烷氧基 C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4二烷基氨基，硫代或C 1 -C 4烷硫基，并且相应的其它取代基A或B为苯基或5-元或6-元杂芳基， 卤素，CN，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4取代基 二烷基氨基，硫代或C 1 -C 4烷硫基。 本发明还涉及所述化合物的耐植物酸加成盐或金属盐，涉及式（I）化合物用于防治植物致病真菌的用途，并涉及含有它们的试剂。

公开(公告)号：EP2035415A1

公开(公告)日：2009-03-18

申请号：EP07765511.6

申请日：2007-06-20

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GROTE, Thomas ,  MÜLLER, Bernd ,  LOHMANN, Jan Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  GLÄTTLI, Alice

IPC: C07D405/06 ,  C07D405/14 ,  C07D409/14 ,  A01N43/653

CPC classification number: C07D405/06

Abstract: The present invention relates to azolylmethyloxiranes of the general formula I, in which A is phenyl substituted by one F and a further substituent selected from Cl, C1-C4-alkyl, C1-C4-haloalkyl and C1-C4-alkoxy, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl, or is phenyl substituted by from one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, with the proviso that B is not o-methylphenyl when A is 2-chloro-4-fluorophenyl, and to their acid addition or metal salts compatible with plants, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising them.

Abstract translation: 本发明涉及通式I的唑基甲基环氧乙烷，其中A是被一个F和另外的选自Cl，C 1 -C 4烷基，C 1 -C 4卤代烷基和C 1 -C 4烷氧基的取代基取代的苯基，B是未取代的 吡啶基，噻吩基，噻唑基，恶唑基或呋喃基，或是被1-3个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷基， C4-卤代烷氧基，C1-C4-烷基氨基，C1-C4-二烷基氨基，硫代或C1-C4-烷硫基，条件是当A是2-氯-4-氟苯基时B不是邻甲基苯基，并且它们的酸加成 或与植物相容的金属盐，用于控制植物病原性真菌的式I化合物的用途和包含它们的组合物。

公开(公告)号：EP2035414A1

公开(公告)日：2009-03-18

申请号：EP07730149.7

申请日：2007-06-14

Applicant: BASF SE

Inventor： DIETZ, Jochen ,  GROTE, Thomas ,  MÜLLER, Bernd ,  LOHMANN, Jan Klaas ,  RENNER, Jens ,  ULMSCHNEIDER, Sarah ,  GLÄTTLI, Alice

IPC: C07D405/06 ,  A01N43/653

CPC classification number: C07D405/06

Abstract: The present invention relates to azolylmethyloxiranes of the general formula I, in which A is phenyl substituted by three F, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl, or is phenyl substituted by from one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to their acid addition or metal salts compatible with plants, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising them.

Abstract translation: 本发明涉及通式I的唑基甲基环氧乙烷，其中A是被三个F取代的苯基，B是未取代的吡啶基，噻吩基，噻唑基，恶唑基或呋喃基，或者是被1-3个以下取代基取代的苯基：卤素 C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4二烷基氨基，硫代或C 1 -C 4烷硫基， 它们的酸加成或与植物相容的金属盐，用于控制植物病原性真菌的式I化合物的用途以及包含它们的组合物。