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公开(公告)号:EP2252582A4
公开(公告)日:2012-03-07
申请号:EP09718154
申请日:2009-02-25
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: JIAANG WEIR-TORN , CHAO YU-SHENG , TSAI TING-YUEH , HSU TSU
IPC: C07D207/09 , A61P3/10 , C07D207/02 , C07D207/06
CPC classification number: C07D417/12 , C07D207/16 , C07D401/12 , C07D403/12 , C07D413/12 , C07D487/08
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公开(公告)号:EP1689389A4
公开(公告)日:2009-06-17
申请号:EP04812524
申请日:2004-11-30
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: HSIEH HSING-PANG , MAHINDROO NEERAJ , HSU TSU-AN , HUANG CHIEN-FU , CHEN XIN , CHAO YU-SHENG
IPC: A61K31/404 , A61K31/405 , A61K31/41 , A61K31/42 , C07D20060101 , C07D209/04 , C07D261/20 , C07D413/12
CPC classification number: A61K31/404 , A61K31/405 , A61K31/41 , A61K31/42 , C07D209/08 , C07D401/12 , C07D403/06 , C07D403/12 , C07D403/14 , C07D405/12 , C07D413/12 , C07D413/14 , C07D417/06 , C07D487/04
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公开(公告)号:EP1729774A4
公开(公告)日:2009-05-06
申请号:EP05725171
申请日:2005-03-09
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: JIAANG WEIR-TOM , CHEN XIN , WU SU-YING , HSIEH HSING-PANG , CHAO YU-SHENG
IPC: A61K31/4725 , A61K31/401 , A61K31/421 , A61K31/426 , A61P3/10 , C07D207/34 , C07D217/00 , C07D233/64 , C07D263/02 , C07D277/18 , C07D401/06 , C07D401/12 , C07D403/06 , C07D417/12
CPC classification number: C07D207/16 , C07D207/34 , C07D401/06 , C07D401/12 , C07D403/06 , C07D403/12 , C07D417/12
Abstract: A compound of the following formula (I) wherein R1, R2, R3, R4, R5, R6, W, X, Y, Z, m, n, and p are as defined herein. This invention also covers methods for inhibiting dipeptidyl peptidase IV or VIII, or treating Type II diabetes with such a compound.
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公开(公告)号:EP2310363A4
公开(公告)日:2012-03-28
申请号:EP09795224
申请日:2009-07-10
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: YEH TENGKUANG , CHEN CHIUNG-TONG , CHAO YU-SHENG
CPC classification number: A61K31/427 , A61K9/0019 , A61K9/0095 , A61K9/08 , A61K9/4858 , A61K47/10 , A61K47/22 , A61K47/60
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5.FUSED BICYCLIC PYRIMIDINE COMPOUNDS AS AURORA KINASE INHIBITORS 有权
Title translation: 稠环双嘧啶类化合物作为AURORIN BOINASE抑制剂公开(公告)号:EP2276346A4
公开(公告)日:2011-08-24
申请号:EP09739460
申请日:2009-04-22
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: HSIEH HSING-PANG , COUMAR MOHANE SELVARAJ , HSU TSU-AN , WU SU-YING , CHAO YU-SHENG
IPC: A01N43/54 , A61K31/505 , C07D239/42
CPC classification number: C07F7/0812 , C07D239/70 , C07D413/14 , C07D487/02
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公开(公告)号:EP2084135A4
公开(公告)日:2010-07-28
申请号:EP07868353
申请日:2007-10-02
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: SHIA KAK-SHAN , TAI CHIA-LIANG , TSAO JING-PO , HSIEH WAN-PING , TSENG SHI-LIANG , CHAO YU-SHENG , HUNG MING-SHIU
IPC: C07D231/00 , A61P29/00
CPC classification number: C07D421/04 , C07D231/14 , C07D409/04
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公开(公告)号:EP2507232A4
公开(公告)日:2013-12-18
申请号:EP10835108
申请日:2010-12-02
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: CHERN JYH-HAUR , CHAO YU-SHENG
IPC: C07D417/14 , A61K31/427 , A61P31/14 , C07D403/14 , C07D413/14
CPC classification number: C07D417/14 , C07D403/14 , C07D413/14
Abstract: Compounds useful for treating hepatitis C virus infection. The compounds are of formula (I): wherein A, B, C, D, R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, m, n, p, q, r, t, u, and v are defined herein. Also disclosed is a method for treating hepatitis C virus infection with these compounds.
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8.
公开(公告)号:EP2331530A4
公开(公告)日:2012-02-22
申请号:EP09816751
申请日:2009-09-22
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: HSIEH HSING-PANG , COUMAR SELVARAJ MOHANE , CHAO YU-SHENG
IPC: C07D403/12 , A61K31/4365 , A61P35/00 , C07D401/12
CPC classification number: A61K31/4365 , A61K31/517 , A61K31/519 , C07D239/94 , C07D401/12 , C07D403/12 , C07D417/12 , C07D417/14 , C07D471/04 , C07D487/04 , C07D491/04 , C07D495/04 , C07D495/14 , C07D498/04 , C07D513/04 , C12N9/99
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公开(公告)号:EP2068870A4
公开(公告)日:2010-08-25
申请号:EP07868354
申请日:2007-10-02
Applicant: NAT HEALTH RESEARCH INSTITUTES
Inventor: SHIA KAK-SHAN , TAI CHIA-LIANG , LIAO JYH-HSIUNG , HUNG MING-SHIU , CHAO YU-SHENG
IPC: A61K31/4155 , A61K31/4439 , A61K31/454 , A61P3/00 , A61P25/00 , A61P29/00 , A61P35/00 , C07D409/04 , C07D409/14
CPC classification number: C07D409/04 , C07D409/14