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1.
公开(公告)号:US20130184313A1
公开(公告)日:2013-07-18
申请号:US13789085
申请日:2013-03-07
申请人: Jayaraman Chandrasekhar , Alan P. Kozikowski , Jianhua Liu , Werner Tueckmantel , Joel R. Walker , Po-wai Yuen
发明人: Jayaraman Chandrasekhar , Alan P. Kozikowski , Jianhua Liu , Werner Tueckmantel , Joel R. Walker , Po-wai Yuen
IPC分类号: A61K31/4439 , C07D401/12 , C07D401/14 , C07D401/02
CPC分类号: C07D401/12 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D471/04 , C07D487/08
摘要: The invention relates to pyridinyl nicotinic acetylcholine receptor ligands, compositions comprising an effective amount of a pyridinyl nicotinic acetylcholine receptor ligand and methods to treat or prevent a condition, such as depression and nicotine dependence, comprising administering to an animal in need thereof an effective amount of a pyridinyl nicotinic acetylcholine receptor ligand.
摘要翻译: 本发明涉及吡啶基烟碱乙酰胆碱受体配体,包含有效量的吡啶基烟碱乙酰胆碱受体配体的组合物以及治疗或预防诸如抑郁症和尼古丁依赖之类的病症的方法,包括向有需要的动物施用有效量的 吡啶基烟碱乙酰胆碱受体配体。
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2.
公开(公告)号:US20100152450A1
公开(公告)日:2010-06-17
申请号:US12578020
申请日:2009-10-13
申请人: Jayaraman Chandrasekhar , Alan P. Kozikowski , Jianhua Liu , Werner Tueckmantel , Joel R. Walker , Po-wai Yuen
发明人: Jayaraman Chandrasekhar , Alan P. Kozikowski , Jianhua Liu , Werner Tueckmantel , Joel R. Walker , Po-wai Yuen
IPC分类号: C07D401/14 , C07D401/12
CPC分类号: C07D401/12 , C07D401/14 , C07D413/14 , C07D471/18
摘要: The invention relates to pyridinyl nicotinic acetylcholine receptor ligands, compositions comprising an effective amount of a pyridinyl nicotinic acetylcholine receptor ligand and methods to treat or prevent a condition, such as depression and nicotine dependence, comprising administering to an animal in need thereof an effective amount of a pyridinyl nicotinic acetylcholine receptor ligand.
摘要翻译: 本发明涉及吡啶基烟碱乙酰胆碱受体配体,包含有效量的吡啶基烟碱乙酰胆碱受体配体的组合物以及治疗或预防诸如抑郁症和尼古丁依赖之类的病症的方法,包括向有需要的动物施用有效量的 吡啶基烟碱乙酰胆碱受体配体。
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公开(公告)号:US08445684B2
公开(公告)日:2013-05-21
申请号:US12578020
申请日:2009-10-13
申请人: Jayaraman Chandrasekhar , Alan P. Kozikowski , Jianhua Liu , Werner Tueckmantel , Joel R. Walker , Po-wai Yuen
发明人: Jayaraman Chandrasekhar , Alan P. Kozikowski , Jianhua Liu , Werner Tueckmantel , Joel R. Walker , Po-wai Yuen
IPC分类号: C07D409/00 , C07D411/00 , C07D413/00 , C07D417/00 , C07D401/00 , C07D421/00
CPC分类号: C07D401/12 , C07D401/14 , C07D413/14 , C07D471/18
摘要: The invention relates to pyridinyl nicotinic acetylcholine receptor ligands, compositions comprising an effective amount of a pyridinyl nicotinic acetylcholine receptor ligand and methods to treat or prevent a condition, such as depression and nicotine dependence, comprising administering to an animal in need thereof an effective amount of a pyridinyl nicotinic acetylcholine receptor ligand.
摘要翻译: 本发明涉及吡啶基烟碱乙酰胆碱受体配体,包含有效量的吡啶基烟碱乙酰胆碱受体配体的组合物以及治疗或预防诸如抑郁症和尼古丁依赖之类的病症的方法,包括向有需要的动物施用有效量的 吡啶基烟碱乙酰胆碱受体配体。
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