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15 条记录 (耗时 0.019 秒)

    Co-crystal
    2.
    发明授权
    Co-crystal 失效
    共晶

    公开(公告)号：US07625910B2

    公开(公告)日：2009-12-01

    申请号：US11748651

    申请日：2007-05-15

    申请人： George Joseph Sependa ,  Richard Storey

    发明人： George Joseph Sependa ,  Richard Storey

    IPC分类号： A61K31/517

    CPC分类号： C07D403/12 ,  C07F9/65583

    摘要： The present invention relates to a novel co-crystal of 2-{ethyl[3-({4-[(5-{2-[(3-fluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]quinazolin-7-yl}oxy)propyl]amino}ethyl dihydrogen phosphate (AZD1152) which is an aurora kinase inhibitor that is useful in the treatment of hyperproliferative diseases such as cancer.

    摘要翻译： 本发明涉及2- {乙基[3 - （{4 - [（5- {2 - [（3-氟苯基）氨基] -2-氧代乙基} -1H-吡唑-3-基 ）氨基]喹唑啉-7-基}氧基）丙基]氨基}乙基磷酸二氢酯（AZD1152），其是可用于治疗过度增殖性疾病如癌症的极光激酶抑制剂。

    NOVEL CO-CRYSTAL
    6.
    发明申请
    NOVEL CO-CRYSTAL 失效

    公开(公告)号：US20080045481A1

    公开(公告)日：2008-02-21

    申请号：US11748651

    申请日：2007-05-15

    申请人： George Sependa ,  Richard Storey

    发明人： George Sependa ,  Richard Storey

    IPC分类号： A61K31/66 ,  A61P35/00 ,  C07F9/02

    CPC分类号： C07D403/12 ,  C07F9/65583

    摘要： The present invention relates to a novel co-crystal of 2-{ethyl[3-({4-[(5-{2-[(3-fluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]quinazolin-7-yl}oxy)propyl]amino}ethyl dihydrogen phosphate (AZD1152) which is an aurora kinase inhibitor that is useful in the treatment of hyperproliferative diseases such as cancer.

    摘要翻译： 本发明涉及2- {乙基[3 - （{4 - [（5- {2 - [（3-氟苯基）氨基] -2-氧代乙基} -1H-吡唑-3-基 ）氨基]喹唑啉-7-基}氧基）丙基]氨基}乙基磷酸二氢酯（AZD1152），其是可用于治疗过度增殖性疾病如癌症的极光激酶抑制剂。

    Movement detector for television signals
    7.
    发明授权
    Movement detector for television signals 失效
    运动检测器用于电视信号

    公开(公告)号：US4364087A

    公开(公告)日：1982-12-14

    申请号：US174426

    申请日：1980-08-01

    申请人： Richard Storey ,  Alan Roberts

    发明人： Richard Storey ,  Alan Roberts

    IPC分类号： H04N5/14 ,  H04N7/18

    CPC分类号： H04N5/144 ,  H04N5/147

    摘要： A movement detector for television signals measures the difference between maximum and minimum values of the movement components of a picture difference signal over a chosen interval. A television signal at an input (12) is delayed in a picture delay (2), and the delayed and undelayed signals subtracted in a subtractor (1) to form a picture difference signal. This is rectified in rectifier (3) and smoothed in a filter (4). A maximum detector (6) and a minimum detector (7) are coupled to the filter output and are re-set at prescribed intervals. A subtractor (8) determines the difference between the output of detectors (6) and (7) and this is compared with a reference value in a comparator (9), the output of which is sampled and stored in a store (10).

    摘要翻译： 用于电视信号的移动检测器测量在所选择的间隔上的图像差分信号的运动分量的最大值和最小值之间的差异。 在输入端（12）处的电视信号在图像延迟（2）中延迟，并且延迟和未延迟的信号在减法器（1）中减去以形成图像差分信号。 这在整流器（3）中整流并在滤波器（4）中平滑化。 最大检测器（6）和最小检测器（7）耦合到滤波器输出，并以规定的间隔重新设定。 减法器（8）确定检测器（6）和（7）的输出之间的差异，并且将其与比较器（9）中的参考值进行比较，比较器（9）的输出被采样并存储在存储器（10）中。

    Bandwidth compression for television signals
    8.
    发明授权
    Bandwidth compression for television signals 失效
    电视信号的带宽压缩

    公开(公告)号：US4942466A

    公开(公告)日：1990-07-17

    申请号：US90584

    申请日：1987-10-05

    申请人： Charles P. Sandbank ,  Ian Childs ,  Richard Storey

    发明人： Charles P. Sandbank ,  Ian Childs ,  Richard Storey

    IPC分类号： G06T7/20 ,  H04N5/14 ,  H04N7/015 ,  H04N7/12 ,  H04N7/26 ,  H04N7/36 ,  H04N7/46 ,  H04N9/64 ,  H04N11/00 ,  H04N11/02 ,  H04N11/16 ,  H04N11/24

    CPC分类号： H04N11/167 ,  G06T7/206 ,  H04N11/006 ,  H04N11/02 ,  H04N19/43 ,  H04N19/51 ,  H04N19/523 ,  H04N19/527 ,  H04N19/547 ,  H04N19/59 ,  H04N19/80 ,  H04N5/145 ,  H04N7/0155 ,  H04N7/0157 ,  H04N7/125 ,  H04N9/646

    摘要： A video signal received from a source (10) is bandwidth-compressed by filters (12, 14, 16), filter (14) being a temporal filter and filter (16) being a spatial filter. Selection of the filter to be used is dependent upon picture content. The transmitter reconstitutes in interpolators (44, 46) the signal which would be regenerated at the receiver, determines which filter gives the best results, and transmits an indication of which filter has been used in a digital signal associated with the analogue video signal. Preferably a determination of motion vectors associated with the signal is made and the digital signal indicates which of the determined motion vectors is applicable to different areas of the picture. By transmitting the control signal digitally with the analogue video signal the receiver circuitry is greatly simplified while its reliability is improved.

    摘要翻译： PCT No.PCT / GB86 / 00799 Sec。 371日期：1987年10月5日 102（e）日期1987年10月5日PCT申请日1986年12月23日PCT公布。 公开号WO87 / 04034 日期1987年7月2日。从源（10）接收的视频信号被滤波器（12,14,16）带宽压缩，作为时间滤波器的滤波器（14）和作为空间滤波器的滤波器（16）。 要使用的滤波器的选择取决于图像内容。 发射机在内插器（44,46）中重建将在接收机处重新生成的信号，确定哪个滤波器给出最佳结果，并且发送与在模拟视频信号相关联的数字信号中使用哪个滤波器的指示。 优选地，确定与信号相关联的运动矢量，并且数字信号指示哪个确定的运动矢量适用于图像的不同区域。 通过用模拟视频信号数字地发送控制信号，大大简化了接收机电路，同时提高了其可靠性。

    Video transmission systems
    9.
    发明授权
    Video transmission systems 失效
    视频传输系统

    公开(公告)号：US4884138A

    公开(公告)日：1989-11-28

    申请号：US174792

    申请日：1988-04-04

    申请人： Richard Storey

    发明人： Richard Storey

    IPC分类号： H04N11/00 ,  H04N7/00 ,  H04N7/015 ,  H04N11/24

    CPC分类号： H04N11/006

    摘要： An HDTV video signal with 1249 lines per picture is transmitted over a transmission channel designed for 625 lines per picture by transmitting alternate samples of two lines of the 1249 line signal on a single line of the 625 line signal. An HDTV receiver can interpolate to give a 1249 line picture but a 625 line receiver will still receive a signal that is adequately compatible to give a display.

    摘要翻译： PCT No.PCT / GB86 / 00797 Sec。 371日期：1988年4月4日 102（e）日期1988年4月4日PCT Filted 1986年12月23日PCT公布。 出版物WO88 / 01462 日期：1988年2月25日。每个图像具有1249行的HDTV视频信号通过专为每个图像625行设计的传输通道传输，通过在625行信号的单行上发送1249行信号的两行的替代采样。 HDTV接收机可以插值以提供1249线路图像，但是625线路接收机仍将接收到足够兼容的信号以给出显示。

    Method of and apparatus for deriving a PAL color television signal corresponding to any desired field in an 8-field PAL sequence from one stored field or picture of a PAL signal
    10.
    发明授权
    Method of and apparatus for deriving a PAL color television signal corresponding to any desired field in an 8-field PAL sequence from one stored field or picture of a PAL signal 失效
    用于从PAL信号的一个存储的场或图像中导出与8场PAL序列中的任何所需场对应的PAL彩色电视信号的方法和装置

    公开(公告)号：US4288810A

    公开(公告)日：1981-09-08

    申请号：US43540

    申请日：1979-05-29

    申请人： John O. Drewery ,  Richard Storey

    发明人： John O. Drewery ,  Richard Storey

    IPC分类号： G06T7/20 ,  H04N5/14 ,  H04N5/262 ,  H04N9/64 ,  H04N9/877 ,  H04N9/39 ,  H04N9/535

    CPC分类号： H04N9/877 ,  G06T7/2053 ,  H04N5/144 ,  H04N5/2625 ,  H04N9/64

    摘要： A single field of a PAL color television signal is stored in a store (50) and provides a signal at an input (52). The signal is delayed by one-line delays (56,58) in series to provide one and two-line delayed signals. Separate switching units (60,62) select desired ones or combinations of the input and delayed signals to constitute respectively the low-frequency and chrominance part of the signal at the output (82). The switch positions are changed between fields, and for at least some fields of the PAL sequence each component of the output signal is formed by combining signals from more than one line, i.e. a halving adder (64;66) averages successive lines for the low frequency part of the signal and a halving subtractor (68) forms the difference between lines two lines apart for the chrominance part. The selector unit outputs are combined in an adder (78) which receives the output of the first selector (60), and also the difference between the output of the two selectors after band pass filtering (76). The store (50) can be replaced by a random access store capable of outputting three successive lines simultaneously. The apparatus has special utility in equipment for movement portrayal.

    摘要翻译： PAL彩色电视信号的单个场被存储在存储器（50）中，并在输入端（52）提供信号。 信号被串行延迟一行延迟（56,58），以提供一行和两行延迟信号。 分离的开关单元（60,62）选择所需的输入和延迟信号的组合，分别构成输出端（82）处的信号的低频和色度部分。 开关位置在场之间改变，并且对于PAL序列的至少一些场，输出信号的每个分量通过组合来自多于一个线的信号形成，即，一半加法器（64; 66）将连续的线平均为低 信号的频率部分和减法减法器（68）形成色度部分两行分开的行之间的差异。 选择器单元输出在接收第一选择器（60）的输出的加法器（78）中以及带通滤波后的两个选择器的输出之间的差（76）组合。 存储器（50）可以由能够同时输出三个连续行的随机存取存储器代替。 该装置在运动描绘设备中具有特殊效用。