公开(公告)号：US20090036691A1

公开(公告)日：2009-02-05

申请号：US12235720

申请日：2008-09-23

申请人： DENNIS P. CURRAN ,  YOUSEUNG SHIN ,  NAKYEN CHOY ,  BILLY W. DAY ,  RAGHAVAN BALACHANDRAN ,  CHARITHA MADIRAJU ,  TIFFANY TURNER

发明人： DENNIS P. CURRAN ,  YOUSEUNG SHIN ,  NAKYEN CHOY ,  BILLY W. DAY ,  RAGHAVAN BALACHANDRAN ,  CHARITHA MADIRAJU ,  TIFFANY TURNER

IPC分类号： C07D313/00

CPC分类号： C07D407/06 ,  C07B2200/07 ,  C07C33/02 ,  C07C59/10 ,  C07C59/42 ,  C07C69/732 ,  C07C69/734 ,  C07D309/10 ,  C07D309/30 ,  C07D313/00 ,  C07D319/06 ,  C07F7/1804

摘要： A compound of the following structure: wherein R1 is H, an alkyl group, an aryl group, an alkenyl group, an alkynyl group, or a halogen atom; R2 is H, an alkyl group, an aryl group, a benzyl group, a trityl group, —SiRaRbRc, CH2ORd, or CORe; Ra, Rb and Rc are independently an alkyl group or an aryl group; Rd is an alkyl group, an aryl group, an alkoxylalkyl group, —RiSiRaRbRc or a benzyl group, wherein Ri is an alkylene group; Re is an alkyl group, an allyl group, a benzyl group, an aryl group, an alkoxy group, or —NRgRh, wherein Rg and Rh are independently H, an alkyl group or an aryl group; R3 is (CH2)n where n is and integer in the range of 0 to 5, —CH2CH(CH3)—, —CH═CH—, —CH═C(CH3)—, or —C≡C—; R4 , wherein y1 and y2 are 1 and y3, y4 and y5 are independently 0 or 1, Rk1, Rk2, Rk3, Rk4 and Rk5 are independently H, CH3, or OR2a, and Rs1, Rs2, Rs3, and Rs4 are independently H or CH3, wherein R2a is H, an alkyl group, an aryl group, a benzyl group, a trityl group, —SiRaRbRc, CH2ORd, or CORe; and R5 is H or OR2b, wherein R2b is H, an alkyl group, an aryl group, an aryl group, a benzyl group, a trityl group, —SiRaRbRc, CH2ORd, or CORe.

摘要翻译： 下列结构的化合物：其中R1是H，烷基，芳基，烯基，炔基或卤素原子; R2是H，烷基，芳基，苄基，三苯甲基，-SiRaRbRc，CH2ORd或CORe; Ra，Rb和Rc独立地为烷基或芳基; Rd是烷基，芳基，烷氧基烷基，-RiSiRaRbRc或苄基，其中R 1是亚烷基; Re为烷基，烯丙基，苄基，芳基，烷氧基或-NRgRh，其中Rg和Rh独立地为H，烷基或芳基; R3是（CH2）n，其中n是0-5的整数，-CH2CH（CH3） - ， - CH-CH-，-CH-C（CH3） - 或-C≡C-; R4，其中y1和y2是1，y3，y4和y5独立地是0或1，Rk1，Rk2，Rk3，Rk4和Rk5独立地是H，CH3或OR2a，Rs1，Rs2，Rs3和Rs4独立地是H 或CH3，其中R2a是H，烷基，芳基，苄基，三苯甲基，-SiRaRbRc，CH2ORd或CORe; R5是H或OR2b，其中R2b是H，烷基，芳基，芳基，苄基，三苯甲基，-SiRaRbRc，CH2ORd或CORe。