公开(公告)号：US06767923B2

公开(公告)日：2004-07-27

申请号：US10282023

申请日：2002-10-29

申请人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann ,  Paul Carter ,  Jürgen Curtze

发明人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann ,  Paul Carter ,  Jürgen Curtze

IPC分类号： A61K31215

CPC分类号： C07C323/25 ,  A01N31/16 ,  C07C43/23 ,  C07C69/017

摘要： Benzhydryl derivatives of the formula I, where the index and the variables are as defined below: X is oxygen or sulfur; R1, R3 are halogen, cyano, nitro, hydroxyl, mercapto, amino, alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, alkylcarbonyloxy, formyloxy, alkylthio, alkenylthio, alkynylthio, alkylamino, dialkylamino, alkylcarbonyl or formyl, where the carbon atoms in the radicals mentioned may be partially or fully halogenated; R2 is halogen, cyano, nitro, hydroxyl, mercapto, amino, alkyl, alkoxy, haloalkyl or haloalkoxy, where the groups R2 may be different if n=2; R4 is alkyl, alkenyl or alkynyl, where the carbon atoms in these radicals may be unsubstituted or partially or fully halogenated; R5, R6 are hydroxyl, alkyl, alkenyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, cycloalkyl, cycloalkylalkyl, cycloalkoxy or cycloalkylalkoxy; n is 0, 1 or 2; processes for preparing the compounds I, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的二苯甲基衍生物，其中指数和变量如下定义：X是氧或硫; R 1，R 3是卤素，氰基，硝基，羟基，巯基，氨基，烷基，烯基， 炔基，烷氧基，烯氧基，炔氧基，烷基羰基氧基，甲酰氧基，烷硫基，烯硫基，炔硫基，烷基氨基，二烷基氨基，烷基羰基或甲酰基，其中所述基团中的碳原子可以被部分或完全卤化; R 2是卤素，氰基， 硝基，羟基，巯基，氨基，烷基，烷氧基，卤代烷基或卤代烷氧基，其中如果n = 2，基团R 2可以不同; R 4是烷基，烯基或炔基，其中这些基团中的碳原子 R 5为羟基，烷基，烯基，卤代烷基，卤代烯基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，环烷基，环烷基烷基，环烷氧基或环烷基烷氧基; n为0,1或 2;制备化合物I的方法，包含它们的组合物及其用途 描述了植物病原性有害真菌。