-
公开(公告)号:US20080108808A1
公开(公告)日:2008-05-08
申请号:US11929673
申请日:2007-10-30
申请人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Zhiyuan Zhang , Bruce Elder , Paul Isbester , Grant Palmer , Jonathon Salsbury , Luckner Ulysse
发明人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Zhiyuan Zhang , Bruce Elder , Paul Isbester , Grant Palmer , Jonathon Salsbury , Luckner Ulysse
IPC分类号: C07D401/04 , C07D401/14 , C07D403/04
CPC分类号: C07D403/04 , C07D239/545 , C07D401/04 , C07D401/14 , C07D403/12 , C07D409/14
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound comprising: wherein M is N or CR4; Q1 and Q2 are each independently selected from the group consisting of CO, SO, SO2, and C═NR9; and each L, X, R1, R2, and R3 are as defined herein.
摘要翻译: 提供化合物,药物,试剂盒和方法用于DPP-IV和其它S9蛋白酶,其包含包含以下的化合物:其中M为N或CR 4; Q 1和Q 2各自独立地选自CO,SO,SO 2和C-NR 9 SUB> 并且每个L,X,R 1,R 2和R 3 3如本文所定义。
-
公开(公告)号:US20080108807A1
公开(公告)日:2008-05-08
申请号:US11929482
申请日:2007-10-30
申请人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Zhiyuan Zhang , Bruce Elder , Paul Isbester , Grant Palmer , Jonathon Salsbury , Luckner Ulysse
发明人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Zhiyuan Zhang , Bruce Elder , Paul Isbester , Grant Palmer , Jonathon Salsbury , Luckner Ulysse
IPC分类号: C07D401/04 , C07D401/14 , C07D403/04
CPC分类号: C07D403/04 , C07D239/545 , C07D401/04 , C07D401/14 , C07D403/12 , C07D409/14
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound comprising: wherein M is N or CR4; Q1 and Q2 are each independently selected from the group consisting of CO, SO, SO2, and C═NR9; and each L, X, R1, R2, and R3 are as defined herein.
-
公开(公告)号:US20050261271A1
公开(公告)日:2005-11-24
申请号:US11080992
申请日:2005-03-15
申请人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Zhiyuan Zhang , Bruce Elder , Paul Isbester , Grant Palmer , Jonathon Salsbury , Luckner Ulysse
发明人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Zhiyuan Zhang , Bruce Elder , Paul Isbester , Grant Palmer , Jonathon Salsbury , Luckner Ulysse
IPC分类号: C07D239/54 , A61K9/08 , A61K9/20 , A61K31/506 , A61K31/513 , A61K31/53 , A61K31/55 , A61P3/10 , A61P13/12 , A61P17/06 , A61P19/02 , A61P25/00 , A61P29/00 , A61P31/18 , A61P35/00 , A61P37/02 , A61P37/06 , A61P39/02 , A61P43/00 , C07D239/545 , C07D239/553 , C07D401/04 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/12 , C07D403/14 , C07D409/14 , C07D43/02
CPC分类号: C07D403/04 , C07D239/545 , C07D401/04 , C07D401/14 , C07D403/12 , C07D409/14
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a compound comprising: wherein M is N or CR4; Q1 and Q2 are each independently selected from the group consisting of CO, SO, SO2, and C═NR9; and each L, X, R1, R2, and R3 are as defined herein.
摘要翻译: 提供化合物,药物,试剂盒和方法用于DPP-IV和其它S9蛋白酶,其包含包含以下的化合物:其中M为N或CR 4; Q 1和Q 2各自独立地选自CO,SO,SO 2和C-NR 9 SUB> 并且每个L,X,R 1,R 2和R 3 3如本文所定义。
-
公开(公告)号:US20080003283A1
公开(公告)日:2008-01-03
申请号:US11835295
申请日:2007-08-07
申请人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Zhiyuan Zhang , Bruce Elder , Paul Isbester , Grant Palmer , Jonathan Salsbury , Luckner Ulysse
发明人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Zhiyuan Zhang , Bruce Elder , Paul Isbester , Grant Palmer , Jonathan Salsbury , Luckner Ulysse
IPC分类号: A61K31/506 , A61K9/20 , A61P13/12 , A61P19/00 , A61P3/10 , A61P35/00 , A61P37/00 , C07D239/08 , C12N9/99
CPC分类号: C07D403/04 , C07D239/545 , C07D401/04 , C07D401/14 , C07D403/12 , C07D409/14
摘要: Compounds are provided for use with DPP-IV of the formula: Also provided are pharmaceutical compositions, kits and articles of manufacture comprising such compounds; methods and intermediates useful for making the compounds; and methods of using said compounds.
摘要翻译: 化合物被提供用于下式的DPP-IV:还提供包含这些化合物的药物组合物,试剂盒和制品; 用于制备化合物的方法和中间体; 以及使用所述化合物的方法。
-
公开(公告)号:US20060135767A1
公开(公告)日:2006-06-22
申请号:US11305818
申请日:2005-12-16
申请人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
发明人: Jun Feng , Stephen Gwaltney , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
IPC分类号: C07D487/04
CPC分类号: C07D471/04 , C07D487/04 , C07D513/04
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV and other S9 proteases that comprise a member selected from the group consisting of: wherein E is CH or N, Q is selected from the group consisting of CO, CS, SO, SO2, or C═NR4, and L, X, Z, R2 and R3 are as defined herein.
摘要翻译: 提供化合物,药物,试剂盒和方法用于DPP-IV和其它S9蛋白酶,其包含选自以下的成员:其中E是CH或N,Q选自CO,CS,SO ,SO 2 2或C-NR 4,以及L,X,Z,R 2和R 3, 如本文所定义。
-
公开(公告)号:US20050070535A1
公开(公告)日:2005-03-31
申请号:US10918317
申请日:2004-08-12
申请人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
发明人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
IPC分类号: A61K9/08 , A61K9/20 , A61K31/506 , A61P3/10 , A61P7/00 , A61P13/12 , A61P17/06 , A61P19/00 , A61P19/02 , A61P25/00 , A61P31/04 , A61P31/18 , A61P35/00 , A61P37/00 , A61P37/06 , A61P43/00 , C07D239/02 , C07D239/36 , C07D239/46 , C07D239/52 , C07D285/16 , C07D401/04 , C07D401/14 , C07D405/04 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04 , A61K31/538 , C07D273/04
CPC分类号: C07D239/36 , C07D239/47 , C07D239/52 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formula I: wherein the substituents are as described herein.
-
公开(公告)号:US20050070530A1
公开(公告)日:2005-03-31
申请号:US10917955
申请日:2004-08-12
申请人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
发明人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
IPC分类号: A61K9/08 , A61K9/20 , A61K31/506 , A61P3/10 , A61P7/00 , A61P13/12 , A61P17/06 , A61P19/00 , A61P19/02 , A61P25/00 , A61P31/04 , A61P31/18 , A61P35/00 , A61P37/00 , A61P37/06 , A61P43/00 , C07D239/02 , C07D239/36 , C07D239/46 , C07D239/52 , C07D285/16 , C07D401/04 , C07D401/14 , C07D405/04 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04 , A61K31/54 , A61K31/505 , A61K31/513
CPC分类号: C07D239/36 , C07D239/47 , C07D239/52 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formula I: wherein the substituents are as described herein.
-
公开(公告)号:US20050070706A1
公开(公告)日:2005-03-31
申请号:US10918326
申请日:2004-08-12
申请人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
发明人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
IPC分类号: A61K9/08 , A61K9/20 , A61K31/506 , A61P3/10 , A61P7/00 , A61P13/12 , A61P17/06 , A61P19/00 , A61P19/02 , A61P25/00 , A61P31/04 , A61P31/18 , A61P35/00 , A61P37/00 , A61P37/06 , A61P43/00 , C07D239/02 , C07D239/36 , C07D239/46 , C07D239/52 , C07D285/16 , C07D401/04 , C07D401/14 , C07D405/04 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04
CPC分类号: C07D239/36 , C07D239/47 , C07D239/52 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formula I: wherein the substituents are as described herein.
-
公开(公告)号:US20050070531A1
公开(公告)日:2005-03-31
申请号:US10918186
申请日:2004-08-12
申请人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
发明人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
IPC分类号: A61K9/08 , A61K9/20 , A61K31/506 , A61P3/10 , A61P7/00 , A61P13/12 , A61P17/06 , A61P19/00 , A61P19/02 , A61P25/00 , A61P31/04 , A61P31/18 , A61P35/00 , A61P37/00 , A61P37/06 , A61P43/00 , C07D239/02 , C07D239/36 , C07D239/46 , C07D239/52 , C07D285/16 , C07D401/04 , C07D401/14 , C07D405/04 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04 , A61K31/549 , A61K31/513
CPC分类号: C07D239/36 , C07D239/47 , C07D239/52 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formula I: wherein the substituents are as described herein.
-
公开(公告)号:US20050065148A1
公开(公告)日:2005-03-24
申请号:US10918318
申请日:2004-08-12
申请人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
发明人: Jun Feng , Stephen Gwaltney , Stephen Kaldor , Jeffrey Stafford , Michael Wallace , Zhiyuan Zhang
IPC分类号: A61K9/08 , A61K9/20 , A61K31/506 , A61P3/10 , A61P7/00 , A61P13/12 , A61P17/06 , A61P19/00 , A61P19/02 , A61P25/00 , A61P31/04 , A61P31/18 , A61P35/00 , A61P37/00 , A61P37/06 , A61P43/00 , C07D239/02 , C07D239/36 , C07D239/46 , C07D239/52 , C07D285/16 , C07D401/04 , C07D401/14 , C07D405/04 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04 , C07D273/04 , A61K31/539
CPC分类号: C07D239/36 , C07D239/47 , C07D239/52 , C07D401/04 , C07D401/14 , C07D405/14 , C07D409/06 , C07D409/14 , C07D417/04
摘要: Compounds, pharmaceuticals, kits and methods are provided for use with DPP-IV inhibitors comprising Formula I: wherein the substituents are as described herein.
-
-
-
-
-
-
-
-
-