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公开(公告)号:US06376710B2
公开(公告)日:2002-04-23
申请号:US09818789
申请日:2001-03-28
申请人: Osamu Matsumoto , Toru Uekawa
发明人: Osamu Matsumoto , Toru Uekawa
IPC分类号: C07C25710
CPC分类号: A01N37/52 , A01N47/12 , C07C257/14 , C07C257/20 , C07C271/64 , C07C323/60
摘要: The present invention provides novel amidine compounds and novel pesticides containing these amidine compounds as active ingredients. The amidine compounds are expressed by formula I: wherein X and Y are the same or different and are independently halogen, nitro, cyano, or C1-C6 alkyl; Z is C1-C6 haloalkyl or C1-C6 haloalkoxy; R1 is hydrogen, halogen, C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxy, C1-C6 haloalkoxy, or a group of formula: S(O)n—R5 (wherein R5 is C1-C6 alkyl or C1-C6 haloalkyl; and n is 0, 1, or 2); R2 and R3 are the same or different and are independently halogen or C1-C6 haloalkyl; and R4 is a group of formula: NR6R7 or N═CR8R9 (wherein R6 is hydrogen, C1-C6 alkyl, (C1-C6 alkoxy)-carbonyl, (C1-C6 alkoxy) C1-C6 alkyl, or C2-C6 acyl; R7 is hydrogen, C1-C6 alkyl, (C1-C6 alkoxy)carbonyl, or C2-C6 acyl; R8 is C1-C6 alkyl or hydrogen; and R9 is C1-C6 alkoxy, C1-C6 alkyl, or di(C1-C6 alkyl)amino).
摘要翻译: 本发明提供新的脒化合物和含有这些脒化合物作为活性成分的新型农药。 脒化合物由式I表示:其中X和Y相同或不同,独立地为卤素,硝基,氰基或C 1 -C 6烷基; Z是C 1 -C 6卤代烷基或C 1 -C 6卤代烷氧基; R 1是氢,卤素,C 1 -C 6烷基,C 1 -C 6卤代烷基,C 1 -C 6烷氧基,C 1 -C 6卤代烷氧基或下式基团:S(O)n -R 5(其中R 5是C 1 -C 6烷基或C1- C6卤代烷基; n为0,1或2); R2和R3相同或不同,独立地为卤素或C1-C6卤代烷基; 并且R 4是下式的基团:NR 6 R 7或N = CR 8 R 9(其中R 6是氢,C 1 -C 6烷基,(C 1 -C 6烷氧基) - 羰基,(C 1 -C 6烷氧基)C 1 -C 6烷基或C 2 -C 6酰基; R7是氢,C1-C6烷基,(C1-C6烷氧基)羰基或C2-C6酰基; R8是C1-C6烷基或氢; R9是C1-C6烷氧基,C1-C6烷基或二(C1- C6烷基)氨基)。
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公开(公告)号:US06380430B1
公开(公告)日:2002-04-30
申请号:US09674267
申请日:2000-12-29
申请人: Dieter Dorsch , Horst Juraszyk , Werner Mederski , Joachim Gante , Hanns Wurziger , Hans-Peter Buchstaller , Sabine Bernotat-Danielowski , Guido Melzer
发明人: Dieter Dorsch , Horst Juraszyk , Werner Mederski , Joachim Gante , Hanns Wurziger , Hans-Peter Buchstaller , Sabine Bernotat-Danielowski , Guido Melzer
IPC分类号: C07C25710
CPC分类号: C07C257/18 , C07C279/22
摘要: Novel compounds of the formula I in which X, R1, R2, R3, R4 and R5 have the meaning indicated in Patent Claim 1, are inhibitors of the coagulation factor Xa and can be employed for the prophylaxis and/or therapy of thromboembolic disorders.
摘要翻译: X 1,R 1,R 2,R 3,R 4和R 5具有专利权利要求1中所示含义的式Iin的新型化合物是凝血因子Xa的抑制剂,可用于预防和/或治疗血栓栓塞性疾病。
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