2-(2-pyridyl)-5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi
    12.
    发明授权
    2-(2-pyridyl)-5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi 失效
    2-(2-吡啶基)-5-苯基-6-氨基嘧啶,用于生产和用于对抗有害真菌的方法和中间产物

    公开(公告)号:US07320975B2

    公开(公告)日:2008-01-22

    申请号:US10505146

    申请日:2003-02-06

    IPC分类号: C07D401/04 A01N43/54

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(2-pyridyl)-5-phenyl-6-aminopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants

    摘要翻译: 本发明涉及式I的2-(2-吡啶基)-5-苯基-6-氨基嘧啶,其中取代基和指数具有以下含义:R 1表示卤素,羟基,杂环基, 烷氧基,烷氧基羰基,氨基甲酰基,烷基氨基羰基,二烷基氨基羰基,吗啉代羰基,吡咯烷基羰基,烷基羰基氨基,烷基氨基。 二烷基氨基,烷硫基,烷基亚磺酰基,烷基磺酰基,羟基磺酰基,氨基磺酰基,烷基氨基磺酰基,二烷基氨基磺酰基; m = 0或1-4; R 2表示氢,卤素,氰基,烷基,卤代烷基或烷氧基; R 3,R 4表示氢,烷基,卤代烷基,环烷基,卤代烷基,烯基,卤代烯基,环烯基,炔基,卤代炔基或环炔基,R 3 O 和R 4与它们连接的氮原子一起形成5或6元环,其被来自基团O,N或S的原子和/或可被取代 根据说明; R 5表示卤素,烷基或卤代烷基; R 6表示氢或R 5中的已知基团之一; R 7,R 8表示氢,卤素,烷基或卤代烷基; R 9表示氢,卤素,羟基,氰基,烷基,烷氧基,环烷氧基,卤代烷氧基,烷氧基羰基或烷基氨基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物,除了其用于对抗不期望的植物之外

    2-(Pyridin-2-yl)-pyrimidines and Their Use for Controlling Harmful Fungi
    14.
    发明申请
    2-(Pyridin-2-yl)-pyrimidines and Their Use for Controlling Harmful Fungi 审中-公开
    2-(吡啶-2-基) - 嘧啶及其用于控制​​有害真菌的用途

    公开(公告)号:US20100286175A1

    公开(公告)日:2010-11-11

    申请号:US12840392

    申请日:2010-07-21

    IPC分类号: A01N43/54 C07D401/04 A01P3/00

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

    摘要翻译: 本发明涉及通式(I)的2-(吡啶-2-基) - 嘧啶化合物及其用于控制​​致病真菌的用途,作为作为活性成分的植物保护产品含有这种化合物:通式 (I)中,k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素,OH,CN,NO 2,C 1 -C 4烷基,C 1 -C 4烷基卤,C 1 -C 4烷氧基,C 1 -C 4烷氧基卤化物,C 2 -C 4烯基,C 2 -C 4炔基, C8环烷基,C1-C4烷氧基-C1-C4烷基,氨基,苯氧基,其任选被卤素或C 1 -C 4烷基取代,NHR,NR 2,C(R a)= N-OR b,S(= O)p A1或C (ΟO)A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-,其中Alk表示直链或支链C 1 -C 4亚烷基,和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤,C1-C4烷氧基,C1-C4烷氧基卤化物,羟基,卤素,CN或NO2; 其中当满足以下三个条件中的至少一个时,R2还可以表示氢或C1-C4烷基:n表示3,4或5; k表示1,2或3; 如果m不等于0,则基团R1中的至少一个表示与卤素,C 1 -C 4烷基,C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团, R3表示C1-C4烷基。

    2-(pyridin-2-yl)-pyrimidines and their use for controlling harmful fungi
    15.
    发明授权
    2-(pyridin-2-yl)-pyrimidines and their use for controlling harmful fungi 失效
    2-(吡啶-2-基) - 嘧啶及其用于控制​​有害真菌的用途

    公开(公告)号:US07786043B2

    公开(公告)日:2010-08-31

    申请号:US11632342

    申请日:2005-07-22

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

    摘要翻译: 本发明涉及通式(I)的2-(吡啶-2-基) - 嘧啶化合物及其用于控制​​致病真菌的用途,作为作为活性成分的植物保护产品含有这种化合物:通式 (I)中,k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素,OH,CN,NO 2,C 1 -C 4烷基,C 1 -C 4烷基卤,C 1 -C 4烷氧基,C 1 -C 4烷氧基卤化物,C 2 -C 4烯基,C 2 -C 4炔基, C8环烷基,C1-C4烷氧基-C1-C4烷基,氨基,苯氧基,其任选被卤素或C 1 -C 4烷基取代,NHR,NR 2,C(R a)= N-OR b,S(= O)p A1或C (ΟO)A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-,其中Alk表示直链或支链C 1 -C 4亚烷基,和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤,C1-C4烷氧基,C1-C4烷氧基卤化物,羟基,卤素,CN或NO2; 其中当满足以下三个条件中的至少一个时,R2还可以表示氢或C1-C4烷基:n表示3,4或5; k表示1,2或3; 如果m不等于0,则基团R1中的至少一个表示与卤素,C 1 -C 4烷基,C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团, R3表示C1-C4烷基。