-
公开(公告)号:US08613914B2
公开(公告)日:2013-12-24
申请号:US13614902
申请日:2012-09-13
IPC分类号: A61K45/00
CPC分类号: C07K7/06 , A61K31/403 , A61K31/4439 , A61K38/06 , A61K38/07 , A61K38/08 , A61K45/06 , C07D209/96 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D417/14 , C07K5/06165 , C07K5/08 , C07K5/0808 , C07K5/0812 , C07K5/10 , C07K5/101 , C07K5/1016
摘要: The present application describes organic compounds that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的有机化合物。
-
12.Derivatised proline containing peptide compounds as protease inhibitors 有权
标题翻译: 含有肽化合物的衍生脯氨酸作为蛋白酶抑制剂公开(公告)号:US08512690B2
公开(公告)日:2013-08-20
申请号:US12755852
申请日:2010-04-07
IPC分类号: A61K45/00
CPC分类号: C07K7/06 , A61K31/403 , A61K31/4439 , A61K38/06 , A61K38/07 , A61K38/08 , A61K45/06 , C07D209/96 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D417/14 , C07K5/06165 , C07K5/08 , C07K5/0808 , C07K5/0812 , C07K5/10 , C07K5/101 , C07K5/1016
摘要: The present application describes organic compounds that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的有机化合物。
-
公开(公告)号:US20140357551A1
公开(公告)日:2014-12-04
申请号:US14462406
申请日:2014-08-18
CPC分类号: C07K7/06 , A61K31/403 , A61K31/4439 , A61K38/06 , A61K38/07 , A61K38/08 , A61K45/06 , C07D209/96 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D417/14 , C07K5/06165 , C07K5/08 , C07K5/0808 , C07K5/0812 , C07K5/10 , C07K5/101 , C07K5/1016
摘要: The present application describes organic compounds of Formula (II) that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的式(II)的有机化合物。
-
公开(公告)号:US08840878B2
公开(公告)日:2014-09-23
申请号:US13614813
申请日:2012-09-13
IPC分类号: A61K45/00 , C07D417/14 , C07D401/12 , C07D209/96 , C07D401/14 , C07K5/087 , C07K5/078 , C07K5/107 , C07D403/12 , C07D403/14 , C07D405/14 , C07K5/103 , C07K5/083
CPC分类号: C07K7/06 , A61K31/403 , A61K31/4439 , A61K38/06 , A61K38/07 , A61K38/08 , A61K45/06 , C07D209/96 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D417/14 , C07K5/06165 , C07K5/08 , C07K5/0808 , C07K5/0812 , C07K5/10 , C07K5/101 , C07K5/1016
摘要: The present application describes organic compounds that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的有机化合物。
-
公开(公告)号:US08222425B2
公开(公告)日:2012-07-17
申请号:US13185683
申请日:2011-07-19
申请人: Shawn D. Britt , Lech Andrzej Ciszewski , Jiping Fu , Subramanian Karur , Yugang Liu , Peichao Lu , David Thomas Parker , Mahavir Prashad , Prakash Raman , Pascal Rigollier , Mohindra Seepersaud , Aregahegn Yifru , Rui Zheng
发明人: Shawn D. Britt , Lech Andrzej Ciszewski , Jiping Fu , Subramanian Karur , Yugang Liu , Peichao Lu , David Thomas Parker , Mahavir Prashad , Prakash Raman , Pascal Rigollier , Mohindra Seepersaud , Aregahegn Yifru , Rui Zheng
IPC分类号: C07D207/00
CPC分类号: C07D401/12 , C07D403/12 , C07K5/0812 , C07K5/1016
摘要: The present application describes organic compounds that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的有机化合物。
-
公开(公告)号:US20090137495A1
公开(公告)日:2009-05-28
申请号:US12249186
申请日:2008-10-10
申请人: Shawn D. Britt , Lech Andrzej Ciszewski , Jiping Fu , Subramanian Karur , Yugang Liu , Peichao Lu , David Thomas Parker , Mahavir Prashad , Prakash Raman , Pascal Rigollier , Mohindra Seepersaud , Aregahegn Yifru , Rui Zheng
发明人: Shawn D. Britt , Lech Andrzej Ciszewski , Jiping Fu , Subramanian Karur , Yugang Liu , Peichao Lu , David Thomas Parker , Mahavir Prashad , Prakash Raman , Pascal Rigollier , Mohindra Seepersaud , Aregahegn Yifru , Rui Zheng
IPC分类号: A61K38/07 , C07K5/113 , C07D498/04 , C07D207/08 , A61P31/12
CPC分类号: C07D401/12 , C07D403/12 , C07K5/0812 , C07K5/1016
摘要: The present application describes organic compounds that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的有机化合物。
-
公开(公告)号:US20110182850A1
公开(公告)日:2011-07-28
申请号:US12755856
申请日:2010-04-07
IPC分类号: A61K38/20 , C07D209/96 , C07D401/14 , C07D401/12 , C07D471/04 , C07D403/14 , C07D403/12 , C07D413/12 , A61K38/21 , A61K31/713 , A61K31/7036 , A61K31/437 , A61K31/7056 , A61K31/496 , A61K31/427 , A61K38/13 , A61K31/7048 , A61K31/403 , A61K31/454 , A61K31/4375 , A61K31/4184 , A61K31/497 , A61K31/5377 , A61P31/14
CPC分类号: C07D401/12 , A61K38/13 , A61K38/2013 , A61K38/204 , A61K38/208 , A61K38/21 , A61K38/212 , C07D403/12 , C07D413/12 , C07K5/101 , C07K7/06 , A61K2300/00
摘要: The present application describes organic compounds that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的有机化合物。
-
公开(公告)号:US20100260709A1
公开(公告)日:2010-10-14
申请号:US12755852
申请日:2010-04-07
IPC分类号: A61K38/20 , C07D209/54 , C07D211/18 , C07D273/01 , A61K31/4025 , A61K31/4439 , A61K31/497 , A61K31/5377 , A61K38/21 , A61K31/713 , A61K31/437 , A61K31/7056 , A61K31/7036 , A61K31/7076 , A61K31/496 , A61K38/13 , A61K31/7105 , A61P31/20
CPC分类号: C07K7/06 , A61K31/403 , A61K31/4439 , A61K38/06 , A61K38/07 , A61K38/08 , A61K45/06 , C07D209/96 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D417/14 , C07K5/06165 , C07K5/08 , C07K5/0808 , C07K5/0812 , C07K5/10 , C07K5/101 , C07K5/1016
摘要: The present application describes organic compounds that are useful for the treatment, prevention and/or amelioration of human diseases.
-
公开(公告)号:US09206232B2
公开(公告)日:2015-12-08
申请号:US14462406
申请日:2014-08-18
IPC分类号: C07D401/12 , C07D403/12 , A61K31/403 , A61K31/4439 , C07K7/06 , C07D209/96 , C07D401/14 , C07D403/14 , C07D405/14 , C07D417/14 , C07K5/078 , C07K5/083 , C07K5/087 , C07K5/103 , C07K5/107 , A61K38/06 , A61K38/07 , A61K38/08 , A61K45/06 , C07K5/08 , C07K5/10
CPC分类号: C07K7/06 , A61K31/403 , A61K31/4439 , A61K38/06 , A61K38/07 , A61K38/08 , A61K45/06 , C07D209/96 , C07D401/12 , C07D401/14 , C07D403/12 , C07D403/14 , C07D405/14 , C07D417/14 , C07K5/06165 , C07K5/08 , C07K5/0808 , C07K5/0812 , C07K5/10 , C07K5/101 , C07K5/1016
摘要: The present application describes organic compounds of Formula (II) that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的式(II)的有机化合物。
-
公开(公告)号:US08008263B2
公开(公告)日:2011-08-30
申请号:US12249186
申请日:2008-10-10
申请人: Shawn D. Britt , Lech Andrzej Ciszewski , Jiping Fu , Subramanian Karur , Yugang Liu , Peichao Lu , David Thomas Parker , Mahavir Prashad , Prakash Raman , Pascal Rigollier , Mohindra Seepersaud , Aregahegn Yifru , Rui Zheng
发明人: Shawn D. Britt , Lech Andrzej Ciszewski , Jiping Fu , Subramanian Karur , Yugang Liu , Peichao Lu , David Thomas Parker , Mahavir Prashad , Prakash Raman , Pascal Rigollier , Mohindra Seepersaud , Aregahegn Yifru , Rui Zheng
CPC分类号: C07D401/12 , C07D403/12 , C07K5/0812 , C07K5/1016
摘要: The present application describes organic compounds that are useful for the treatment, prevention and/or amelioration of human diseases.
摘要翻译: 本申请描述了可用于治疗,预防和/或改善人类疾病的有机化合物。
-
-
-
-
-
-
-
-
-