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公开(公告)号:US20120309800A1
公开(公告)日:2012-12-06
申请号:US13519801
申请日:2010-12-29
IPC分类号: A61K31/41 , A61P35/00 , A61P9/00 , A61P29/00 , A61P25/00 , A61P13/00 , A61P1/00 , A61P5/00 , A61P5/28 , A61P17/00 , A61P17/14 , A61P5/32 , A61P15/00 , A61P17/10 , A61P17/06 , A61P31/10 , C07D257/04
CPC分类号: C07D257/04 , A61K31/165 , A61K31/41 , A61K31/415 , A61K31/4196 , A61K45/06 , A61K2300/00
摘要: The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US20120149729A1
公开(公告)日:2012-06-14
申请号:US13324707
申请日:2011-12-13
IPC分类号: A61K31/4192 , C07D401/06 , A61K31/4709 , A61P35/00 , A61P9/00 , A61P29/00 , A61P31/00 , A61P3/00 , A61P27/02 , A61P25/00 , A61P13/00 , A61P1/00 , A61P5/00 , A61P13/08 , A61P15/00 , A61P17/00 , A61P17/14 , A61P15/08 , A61P17/10 , A61P5/26 , A61P17/06 , A61P31/10 , C07D249/04
CPC分类号: C07D249/04 , A61K31/4192 , A61K31/4709 , A61K45/06 , C07D401/06 , C07D401/14 , C07D471/10 , A61K2300/00
摘要: The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
摘要翻译: 本发明描述了具有金属酶调节活性的化合物,以及治疗由这些金属酶介导的疾病,病症或症状的方法。
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公开(公告)号:US20080318248A1
公开(公告)日:2008-12-25
申请号:US12090753
申请日:2006-10-20
IPC分类号: G01N33/53 , G01N33/566 , C40B30/04 , C12N5/02
CPC分类号: G01N33/6803 , C12Q1/00 , G01N2500/04
摘要: The present invention is directed to compositions and methods of screening apoproteins for the elucidation of modulators of metalation of apoproteins.
摘要翻译: 本发明涉及筛选载脂蛋白的组合物和方法,以阐明脱辅基蛋白的金属化调节剂。
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公开(公告)号:US09414596B2
公开(公告)日:2016-08-16
申请号:US14373304
申请日:2013-01-18
IPC分类号: A01N43/713 , A01N43/56 , A01N43/653 , A01N43/647 , A01N57/16
CPC分类号: A01N43/713 , A01N43/56 , A01N43/647 , A01N43/653 , A01N57/16
摘要: The present disclosure describes compounds having agricultural fungicidal activity.
摘要翻译: 本公开内容描述了具有农业杀真菌活性的化合物。
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公开(公告)号:US20160130263A1
公开(公告)日:2016-05-12
申请号:US14897331
申请日:2014-06-11
IPC分类号: C07D413/14 , A61K31/4439 , A61K45/06 , C07D401/14 , A61K31/496 , C07D401/06 , C07D409/14
CPC分类号: C07D413/14 , A01N43/713 , A01N43/84 , A01N43/86 , A61K31/4439 , A61K31/496 , A61K45/06 , C07D401/06 , C07D401/14 , C07D409/14 , Y02A50/409 , Y02A50/411 , Y02A50/414
摘要: The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US09221791B2
公开(公告)日:2015-12-29
申请号:US14457620
申请日:2014-08-12
发明人: William J. Hoekstra , Stephen W. Rafferty , Christopher M. Yates , Robert J. Schotzinger , Michael R. Loso , Michael T. Sullenberger , Gary D. Gustafson
IPC分类号: A01N43/54 , C07D401/06 , C07D401/14 , A01N43/56 , A01N43/647 , A01N43/713 , A01N43/76 , A01N43/78 , C07D405/06 , C07D409/14 , C07D413/06 , C07D417/06 , A01N43/653 , A01N43/84
CPC分类号: C07D401/06 , A01N43/54 , A01N43/56 , A01N43/647 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/78 , A01N43/84 , C07D401/14 , C07D405/06 , C07D409/14 , C07D413/06 , C07D417/06
摘要: The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US08754227B2
公开(公告)日:2014-06-17
申请号:US13561586
申请日:2012-07-30
IPC分类号: A61K31/44 , C07D401/00
CPC分类号: C07D401/06
摘要: The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US08748461B2
公开(公告)日:2014-06-10
申请号:US13527426
申请日:2012-06-19
申请人: William J. Hoekstra , Christopher M. Yates , Robert J. Schotzinger , Michael R. Loso , Zachary A. Buchan , Michael T. Sullenberger , Gary D. Gustafson
发明人: William J. Hoekstra , Christopher M. Yates , Robert J. Schotzinger , Michael R. Loso , Zachary A. Buchan , Michael T. Sullenberger , Gary D. Gustafson
CPC分类号: A01N43/713 , A01N25/00 , A01N43/647 , A01N43/653 , A01N43/78 , C07D401/06 , C07D401/14 , C07D409/14 , C07D417/14
摘要: The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US20130261135A1
公开(公告)日:2013-10-03
申请号:US13882443
申请日:2011-10-28
IPC分类号: C07D401/06 , A61K45/06 , A61K31/506 , C07D409/14 , C07D239/26 , A61K31/505
CPC分类号: C07D401/06 , A61K31/505 , A61K31/506 , A61K45/06 , C07D239/26 , C07D409/14
摘要: The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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公开(公告)号:US20130184309A1
公开(公告)日:2013-07-18
申请号:US13784466
申请日:2013-03-04
IPC分类号: C07D413/10 , C07D401/06 , C07D249/04
CPC分类号: A61K31/4725 , A01N43/647 , A61K31/4192 , A61K31/422 , A61K31/4709 , A61K45/06 , C07D249/04 , C07D401/06 , C07D405/12 , C07D409/14 , C07D413/10 , C07D413/12 , A61K2300/00
摘要: The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
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