公开(公告)号：US4758570A

公开(公告)日：1988-07-19

申请号：US49953

申请日：1987-05-15

申请人： Martin Harris ,  Michael Pearson

发明人： Martin Harris ,  Michael Pearson

IPC分类号： A01N43/54 ,  C07D239/06 ,  A61K31/505

CPC分类号： C07D239/06 ,  A01N43/54

摘要： The invention provides 2-nitromethylene hexahydropyrimidines of the general formula: ##STR1## in which R represents a hydrogen atom; a cycloalkyl group optionally substituted by alkyl and/or halogen; or a group of formula --(CO).sub.n (Y).sub.m R.sup.2 in which n is 0 or 1, Y is oxygen or sulphur, m is 0 or 1 and R.sup.2 represents an alkyl, alkenyl or alkynyl group optionally substituted by one or more substituents selected from halogen; alkoxy; haloalkoxy; alkoxyalkoxy; hydroxy; acyloxy; thiol; cycloalkyl optionally substituted by alkyl and/or halogen; and optionally substituted phenyl; and R.sup.1 represents an optionally substituted phenyl group; their preparation and their use as pesticides.

摘要翻译： 本发明提供了通式如下的2-硝基亚甲基六氢嘧啶：其中R表示氢原子; 任选被烷基和/或卤素取代的环烷基; 或其中n为0或1的式 - （CO）n（Y）m R 2的基团，Y为氧或硫，m为0或1，R 2为任选被一个或多个取代基取代的烷基，链烯基或炔基 选自卤素 烷氧基 卤代烷氧基 烷氧基烷氧基 羟基; 酰氧基 硫醇 任选被烷基和/或卤素取代的环烷基; 和任选取代的苯基; 并且R 1表示任选取代的苯基; 他们的准备和用作农药。