METHOD FOR PRODUCING N-SULFONYL-SUBSTITUTED OXINDOLES
    41.
    发明申请
    METHOD FOR PRODUCING N-SULFONYL-SUBSTITUTED OXINDOLES 有权
    生产N-磺基取代的氧化物的方法

    公开(公告)号:US20140005388A1

    公开(公告)日:2014-01-02

    申请号:US13995898

    申请日:2011-12-19

    IPC分类号: C07D403/04

    摘要: Process for the selective N-sulfonylation of oxindoles, in particular process for the N-sulfonylation of 3-triazinyloxindoles, and also N-sulfonyl-substituted 3-triazinyloxindoles and the use of N-sulfonyl-substituted oxindoles and of N-sulfonyl-substituted 3-triazinyloxindoles as intermediates for the synthesis of fine chemicals and of active ingredients in the field of pharmacy and agriculture, and also the use of these compounds as active ingredients in the field of agriculture.

    摘要翻译: 用于N-羟基吲哚的选择性N-磺酰化的方法,特别是3-三嗪基氧基吲哚的N-磺酰化方法,以及N-磺酰基取代的3-三嗪并氧基吲哚和使用N-磺酰基取代的羟基吲哚和N-磺酰基取代的 3-三嗪基氧吲哚作为合成精细化学品和药物和农业领域的活性成分的中间体,以及这些化合物作为农业领域的活性成分的用途。

    Pyridyl phosphates, compositions containing them and their use as
pesticides
    46.
    发明授权
    Pyridyl phosphates, compositions containing them and their use as pesticides 失效
    吡啶磷酸酯,它们的组合物及其作为杀虫剂的用途

    公开(公告)号:US5075294A

    公开(公告)日:1991-12-24

    申请号:US256780

    申请日:1988-10-12

    CPC分类号: C07F9/585 A01N57/08

    摘要: Pyridylphosphates, a process for their preparation, agents containing them, and their use as pesticides compounds of the formula I ##STR1## where A is N or N-->O,R.sup.1, R.sup.2 independently of one another are halogen,X=O or S,R.sup.3 and R.sup.4 independently of one another are H, halogen, phenyl, phenylthio, phenoxy, phenylsulfenyl, phenylsulfinyl, phenylsulfonyl, phenylsulfonylamino, phenylamino, phenylcarbonylamino, all of which can be substituted in the phenyl moiety by halogen, alkyl, alkoxy, alkylcarbonyl, alkoxycarbonyl, haloalkoxy, haloalkyl, nitro, dialkylamino, alkylthio, cyano or carboxyl, or are alkyl, alkoxy, alkylthio, alkylcarbonyl, alkoxycarbonyl, haloalkoxy, haloalkyl, alkylsulfenyl, alkylsulfinyl, alkylsulfonyl, cyano, nitro, carboxyl, sulfo, heteroaryl, heteroaryloxy, alkenyl, alkinyl, both of which can optionally be mono- substituted or polysubstituted by halogen, or are amino, monoalkylamino, dialkylamino, it being possible for the two alkyl groups, together with the N atom, to form a 5- to 7-membered ring, or are alkylsulfonylamino, thiocyanato or cyanato andR.sup.5 and R.sup.6 independently of one another are alkyl, alkoxy, monoalkylamino, dialkylamino, it being possible for the two alkyl groups together with the N atom to form a 5- to 7-membered ring, or are phenyl, phenoxy, phenylthio, all of which can be substituted by halogen, alkyl, alkoxy, alkylcarbonyl, alkoxycarbonyl, haloalkoxy, haloalkyl, nitro, dialkylamino, alkylthio, cyano or carboxyl, or denote alkylthio, have advantageous insecticidal, acaricidal or nematocidal properties.

    摘要翻译: 吡啶基磷酸酯,其制备方法,含有它们的试剂,以及它们作为农药的用途,其中A是N或N-> O,R 1,R 2彼此独立地是卤素,X = O或S,R 3和R 4彼此独立地是H,卤素,苯基,苯硫基,苯氧基,苯基亚磺酰基,苯基亚磺酰基,苯基磺酰基,苯基磺酰基氨基,苯基氨基,苯基羰基氨基,它们都可以在苯基部分被卤素,烷基, ,烷基羰基,烷氧基羰基,卤代烷氧基,卤代烷基,硝基,二烷基氨基,烷硫基,氰基或羧基,或者是烷基,烷氧基,烷硫基,烷基羰基,烷氧基羰基,卤代烷氧基,卤代烷基,烷基亚磺酰基,烷基亚磺酰基,烷基磺酰基,氰基,硝基,羧基,磺基, ,杂芳基氧基,烯基,炔基,它们都可以任选被卤素单取代或多取代,或者是氨基,单烷基氨基,二烷基氨基,两个烷基可能与N原子t o形成5-至7-元环,或者为烷基磺酰基氨基,氰硫基或氰基,R 5和R 6彼此独立地为烷基,烷氧基,单烷基氨基,二烷基氨基,两个烷基与N原子一起形成 烷基,烷氧基,烷基羰基,烷氧基羰基,卤代烷氧基,卤代烷基,硝基,二烷基氨基,烷硫基,氰基或羧基,或者表示 烷硫基,具有有利的杀虫,杀螨或杀线虫性质。

    SUBSTITUTED 4-CYAN-3-(2,6-DIFLUOROPHENYL)-4-PHENYLBUTANOATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS
    49.
    发明申请
    SUBSTITUTED 4-CYAN-3-(2,6-DIFLUOROPHENYL)-4-PHENYLBUTANOATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS 审中-公开
    取代的4-氰基-3-(2,6-二氟苯基)-4-苯基丁酸酯,其生产方法及其作为除草剂和植物生长调节剂的用途

    公开(公告)号:US20140087945A1

    公开(公告)日:2014-03-27

    申请号:US14005759

    申请日:2012-03-12

    摘要: Compounds of the formula (I) or salts thereof, in which R1 is H or a hydrolyzable radical, (R2)n is n substituents R2, where R2 independently of the others is Hal, CN, NO2, (C1-C8)-alkyl, (C1-C8)-alkoxy, (C1-C8)-alkylthio, (C1-C8)-alkylsulfinyl, (C1-C8)-alkylsulfonyl, (C1-C6)-haloalkyl, (C1-C6)-haloalkoxy, (C1-C6)-haloalkylthio, (C1-C6)-haloalkylsulfinyl, (C1-C6)-haloalkylsulfonyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl, tri-[(C1-C4)-alkyl]-silyl or tri-[(C1-C4)-alkyl]-silyl-(C1-C4)-alkyl or where in each case two groups R2 located ortho at the ring together are —Z1-A*-Z2, in which A* is (C1-C4)-alkylene, which is optionally substituted by radicals from the group consisting of halogen, (C1-C4)-alkyl, (C1-C4)-haloalkyl, (C1-C4)-alkoxy and (C1-C4)-haloalkoxy, Z1, Z2 are each a direct bond, O or S and where the group —Z1-A*-Z2 together with the carbon atoms, attached to the group, of the phenyl ring form a fused-on 5- or 6-membered ring, and n is 0, 1, 2, 3, 4 or 5, excluding the compound in which R1 is methyl and (R2)n is 3-fluoro (n=1), are suitable for use as herbicides and plant growth regulators and can be prepared by the process of claim 8.

    摘要翻译: 式(I)化合物或其盐,其中R 1为H或可水解基团,(R2)n为n取代基R2,其中R2独立地为Hal,CN,NO2,(C1-C8) - 烷基 ,(C1-C8) - 烷氧基,(C1-C8) - 烷硫基,(C1-C8)烷基亚磺酰基,(C1-C8) - 烷基磺酰基,(C1-C6) - 卤代烷基,(C1-C6) - 卤代烷氧基,( (C 1 -C 6) - 卤代烷基亚磺酰基,(C 1 -C 6) - 卤代烷基磺酰基,(C 2 -C 6) - 烯基,(C 2 -C 6) - 炔基,三 - [(C 1 -C 4) - 烷基] 甲硅烷基或三 - [(C 1 -C 4) - 烷基] - 甲硅烷基 - (C 1 -C 4) - 烷基或其中在每种情况下两个位于环的环上的两个R一起为-Z1-A * -Z2,其中A (C1-C4) - 烷基,(C1-C4) - 烷氧基,(C1-C4) - 烷氧基,(C1-C4) - 烷氧基,(C1-C4) C 4) - 卤代烷氧基,Z 1,Z 2各自为直接键,O或S,并且其中与基团连接的苯基上的基团-Z1-A * -Z2与碳原子一起形成稠合的5- 或6元环,n为0,1,2,3,4或5,不包括化合物i n,其中R1是甲基,(R2)n是3-氟(n = 1),适合用作除草剂和植物生长调节剂,并且可以通过权利要求8的方法制备。