公开(公告)号：US20070275981A1

公开(公告)日：2007-11-29

申请号：US11661922

申请日：2005-09-05

申请人： Markus Gewehr ,  Thomas Grote ,  Bernd Muller ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Jan Rether ,  Siefgried Strathmann ,  Reinhard Stierl ,  Maria Scherer

发明人： Markus Gewehr ,  Thomas Grote ,  Bernd Muller ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Jan Rether ,  Siefgried Strathmann ,  Reinhard Stierl ,  Maria Scherer

IPC分类号： A01N43/40 ,  A01N43/54 ,  A01P3/00 ,  C07D239/28 ,  C07D401/04

CPC分类号： A01N43/78 ,  A01N43/56 ,  C07D213/82 ,  C07D231/40 ,  C07D277/56 ,  C07D333/38 ,  C07D401/12 ,  C07D403/12 ,  C07D409/12 ,  C07D417/12

摘要： The invention relates to the use of (hetero)cyclylcarboxamides of general formula (I) and to the agriculturally useful salts thereof for controlling plant pathogenic fungi, the variables in formula (I) having the following designations: A represents phenyl or an at least monosaturated five-membered or six-membered heterocycle with 1, 2 or 3 heteroatoms as ring members selected from N, O, S, S(═O) and S(═O)2, where phenyl and the at least monosaturated five-membered or six-membered heterocycle can be unsubstituted or substituted according to the description; Y represents oxygen or sulphur; R1 represents H, OH, alkyl, cycloalkyl, alkoxy, halogenalkyl, halogencycloalkyl or halogenalkoxy; R2 and R3 represent H, halogen, nitro, CN, alkyl, cycloalkyl, alkenyl, alkinyl, alkoxy, halogenalkyl, halogencycloalkyl, halogenalkenyl, halogenalkinyl or halogenalkoxy; R4 represents halogen, nitro, CN, alkyl, cycloalkyl, alkenyl, alkinyl, alkoxy, halogenalkyl, halogencycloalkyl, halogenalkenyl, halogenalkinyl or halogenalkoxy; R5 represents hydrogen, halogen, nitro, CN, OH, alkyl, cycloalkyl, alkenyl, alkinyl, alkoxy, alkenyloxy, alkinyloxy, alkoxyalkoxy, halogenalkyl, halogencycloalkyl, halogenalkenyl, halogenalkinyl or halogenalkoxy; alklthio, halogenalkylthio, alkylsulfinyl, halogenalkylsulfinyl, alkylsulfonyl, halogenalkylsulfonyl, —(CR6)═NOR7, —C(O)R8, NR9R10, —C(O)NR9R10, —C(S)NR9R10, phenyl or phenylalkyl, the phenyl ring in the last two radicals optionally comprising between 1 and 4 of the radicals cited for R4; R6, R7, R8, R9 and R10 have the designations cited in the description; the two radicals R4 and R5 bound to adjacent carbon atoms can also represent an alkylene chain with 3 to 5 members, wherein 1 or 2 non-adjacent CH2 groups can also be replaced by O or S, and part or all of the hydrogens can be replaced by halogen; Ar represents phenyl, naphtyl or a five-membered or six-membered heteroaromatic radical with 1, 2 or 3 heteroatoms as ring members selected from N, O, and S, that can optionally also carry a fused benzene ring; and n represents 0, 1, 2, 3, or 4. The invention also relates to crop protection agents containing said compounds.

公开(公告)号：US20080108686A1

公开(公告)日：2008-05-08

申请号：US11628325

申请日：2005-06-16

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

IPC分类号： A01N43/56 ,  A01P3/00 ,  C07D231/12

CPC分类号： A01N43/56 ,  C07D231/14

摘要： The present invention relates to N-(ortho-phenyl)-1-methyl-3-difluoromethylpyrazole-4-carboxanilides of the formula I in which the substituents are as defined below:R1 and R2 independently of one another are halogen, C1-C6-alkyl, C1-C6-haloalkyl, cyano, nitro, methoxy, trifluoromethoxy or difluoromethoxy.

摘要翻译： 本发明涉及式I的N-（邻苯基）-1-甲基-3-二氟甲基吡唑-4-甲酰苯胺，其中取代基如下：R 1和R 2 > 2个彼此独立地是卤素，C 1 -C 6 - 烷基，C 1 -C 6 氰基，硝基，甲氧基，三氟甲氧基或二氟甲氧基。

公开(公告)号：US20070299115A1

公开(公告)日：2007-12-27

申请号：US11661679

申请日：2005-09-05

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Shwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Shwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

IPC分类号： A01N37/48 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01P3/00 ,  C07C233/00 ,  C07D213/82 ,  C07D231/14 ,  C07D277/56

CPC分类号： C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  C07D231/14 ,  C07D277/56

摘要： The invention relates to (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I) and to salts of said anilides that can be used for agricultural purposes for controlling pathogenic fungi. In said formula, the variables are defined as follows: A represents a phenyl or at least a monounsaturated 5- or 6-membered heterocycle comprising 1, 2 or 3 heteroatoms, selected from N, O, S, S(═O) and S(═O)2 as ring members, whereby phenyl and the monounsaturated 5- or 6-membered heterocycle can be unsubstituted or can be substituted according to the description; B represents a group of general formula (II), in which the variables R3, R4, R5 and the index m are defined as cited in the claims and the description; Y represents oxygen or sulphur, R1 represents H, OH, alkyl, cycloalkyl, alkoxy, haloalkyl, halocycloalkyl or haloalkoxy; R2 represents halogen, nitro, CN, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, haloalkyl, halocycloalkyl, haloalkenyl, haloalkynyl or haloalkoxy; and n represents 0, 1, 2, 3 or 4; and salts that can be used for agricultural purposes. The invention also relates to the use of the (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I), to a method for controlling pathogenic fungi and to a crop protection agent containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound.

摘要翻译： 本发明涉及通式（I）的（杂）环（硫代）羧酸酰苯胺和可用于农业目的的用于控制致病真菌的所述酰苯胺的盐。 在所述式中，变量定义如下：A表示苯基或至少一个单不饱和的5-或6-元杂环，其包含1,2或3个选自N，O，S，S（-O）和S （-O）2，作为环成员，由此苯基和单不饱和的5-或6-元杂环可以是未取代的或可以根据描述被取代; B表示通式（II）的基团，其中定义了变量R 3，R 4，R 5和指数m， 如权利要求和说明书所引用的; Y表示氧或硫，R 1表示H，OH，烷基，环烷基，烷氧基，卤代烷基，卤代环烷基或卤代烷氧基; R 2表示卤素，硝基，CN，烷基，环烷基，烯基，炔基，烷氧基，卤代烷基，卤代环烷基，卤代烯基，卤代炔基或卤代烷氧基。 并且n表示0,1,2,3或4; 和可用于农业目的的盐。 本发明还涉及通式（I）的（杂）环（硫代）羧酸二酰苯胺用于控制致病真菌的方法和含有至少一种通式（I）的化合物的作物保护剂， 和/或所述化合物的农业上相容的盐。

公开(公告)号：US20070249634A1

公开(公告)日：2007-10-25

申请号：US11597409

申请日：2005-06-08

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bern Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Petere Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Liliana Rapado ,  Michael Rack ,  Barbara Nave ,  Maria Schere ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bern Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Petere Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Liliana Rapado ,  Michael Rack ,  Barbara Nave ,  Maria Schere ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A01P3/00

CPC分类号： A01N43/90

摘要： The invention relates to the use of triazolopyrimidines of the formula I In which: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl, C3-C6-cycloalkynyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one, two, three or four heteroatoms from the group consisting of O, N and S, where R1, R2 may be substituted as defined in the description or R1 and R2 together with the nitrogen atom to which they are attached may form five- to eight-membered heterocyclyl or heteroaryl which is attached via nitrogen and may contain one, two or three further heteroatoms from the group consisting of O, N and S as ring members and/or may be substituted as defined in the description; L independently of one another are halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyloxy, cyano, C(═O)A1, S(═O)mA2, NRcRd or NRc—(C═O)—Rd, where A1, A2, Rc, Rd and m are as defined in the description; L1 is halogen, alkyl or haloalkyl; L2 is nitro, a group —C(S)NR3R4, a group —C(═N—OR5)(NR6R7) or a group —C(═N—NR8R9)(NR10OR11); X is halogen, cyano, alkyl, alkoxy, haloalkyl or haloalkoxy; R3, R4, R5, R6, R7, R8, R9, R10 and R11 are independently of one another selected from the group consisting of hydrogen, alkyl, cycloalkyl, alkenyl and alkynyl, where the 4 last-mentioned radicals may be substituted as defined in the description; or R3 and R4, or R6 and R7, or R8 and R9 or R10 and R11 together with the nitrogen atom to which they are attached form a four, five, or six-membered saturated or partially unsaturated ring which may be substituted as defined in the description; n is 0, 1, 2 or 3; and the agriculturally acceptable salts thereof, novel triazolopyrimidines, crop protection compositions comprising at least one compound of the formula I and at least one solid or liquid carrier, and a method for controlling phytopathogenic harmful fungi.

公开(公告)号：US07820647B2

公开(公告)日：2010-10-26

申请号：US11596891

申请日：2005-05-17

申请人： Anja Schwögler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Carsten Blettner ,  Peter Schäfer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwögler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Carsten Blettner ,  Peter Schäfer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： C07D239/48 ,  C07D403/04 ,  A01N43/54 ,  A01N43/58 ,  A01N43/34 ,  A01P3/00

CPC分类号： C07D401/04 ,  C07D403/04

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents L and R1 to R3 are as defined in the description and X is a group —CH—Ra, —N—Rb—, —O— or —S—; Ra may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, cyano or C1-C6-alkoxycarbonyl; Rb is hydrogen, C1-C6-alkyl or C3-C6-cycloalkyl; T is a group —CH—Ra—; p is an integer from 1 to 4; Y is a group —CH—Ra— or —N—Rb—, o is 0 or 1; Z is O, S or a group N(Rc) Rc is hydrogen, C1-C6-alkyl or C1-C6-alkoxy, and to processes for their preparation, to pesticidal compositions comprising them and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基L和R1至R3如说明书中所定义，X为基团-CH-Ra，-N-Rb-，-O- 或-S-; R a可以是氢，卤素，C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，氰基或C 1 -C 6 - 烷氧基羰基; R b是氢，C 1 -C 6 - 烷基或C 3 -C 6 - 环烷基; T是基团-CH-R a; p是1至4的整数; Y是基团-CH-R a或-N-R b - ，o是0或1; Z是O，S或基团N（R c）R c是氢，C 1 -C 6烷基或C 1 -C 6 - 烷氧基，并且其制备方法，包含它们的杀虫组合物和它们作为农药的用途。

公开(公告)号：US20060293314A1

公开(公告)日：2006-12-28

申请号：US10570893

申请日：2004-09-10

申请人： Wassilos Grammenos ,  Carsten Blettner ,  Bernd Müller ,  Marker Gewehr ,  Jordi Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Maria Scherer ,  Reinhard Stierl

发明人： Wassilos Grammenos ,  Carsten Blettner ,  Bernd Müller ,  Marker Gewehr ,  Jordi Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/541 ,  A61K31/5377 ,  A61K31/496 ,  A61K31/4439 ,  A61K31/44 ,  C07D417/02 ,  C07D403/02 ,  C07D413/02

CPC分类号： C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

摘要： Sulfonamides of the formula I where the substituents are as follows: R1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R2, R3, R4, R5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R2, and R3,, R2,, R3, are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R2, R3, R4 and R5 are hydrogen: X is phenyl substituted by a group —C(R6)═NOR7, where R6 is alkyl and R7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R2, R3, R4 and R5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的磺酰胺，其中取代基如下：R 1是氢，烷基，烷氧基，烯基或炔基; R 2，R 3，R 4，R 5是氢，卤素，烷基，烷氧基或卤代甲基 ; R 2和R 3一起也可以形成苯基，环戊基或环己基环，这些环可以携带两个基团R 2， R 3，R 3，R 3，R 3，R 3，R 3和R 3分别为氢，卤素，烷基，烷氧基或卤代甲基; 在a）情况下，如果R 2，R 3，R 4和R 5是氢：X是 由基团-C（R 6） - NOR 7取代的苯基，其中R 6为烷基，R 7为H 烷基，苄基，烯基，卤代烷基，卤代烯基，炔基或卤代炔基; 并且在情况b）中，如果R 2，R 3，R 4和R 5中的至少一个， SUP>不是氢：X是苯基，萘基或五或六元饱和或部分不饱和或芳族杂环，其通过碳原子连接并含有一至四个由O，N和S组成的组的杂原子 ，其中X可以根据描述被替代; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080227796A1

公开(公告)日：2008-09-18

申请号：US11793286

申请日：2005-12-16

申请人： Oliver Wagner ,  Thomas Grote ,  Joachim Rheinheimer ,  Barbara Nave ,  Reinhard Stierl

发明人： Oliver Wagner ,  Thomas Grote ,  Joachim Rheinheimer ,  Barbara Nave ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC分类号： A01N43/90 ,  C07D213/55 ,  C07D237/14 ,  C07D487/04

摘要： The present invention relates to novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds and to their agriculturally acceptable salts, and also to their use for controlling harmful fungi, and also to crop protection compositions comprising at least one such compound as active component.The novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds can be described by the formula I where the substituents R1, R2, Het, X and Y in formula I are as defined below: Het is a 6-membered heteroaromatic radical selected from the group consisting of pyridinyl, pyridazinyl, pyrazinyl, 1,2,4-triazinyl and 1,3,5-triazinyl, where the 6-membered heteroaromatic radical may have 1, 2 or 3 identical or different substituents L, R1, R2 independently of one another are hydrogen, C1-C8-alkyl, C1-C8-haloalkyl, C1-C8-alkoxy, C3-C8-cycloalkyl, C3-C8-cycloalkoxy, C5-C10-bicycloalkyl, C3-C8-halocycloalkyl, C2-C8-alkenyl, C2-C8-alkenyloxy, C4-C10-alkadienyl, C2-C8-haloalkenyl, C3-C8-cycloalkenyl, C3-C8-halocycloalkenyl, C2-C8-alkynyl, C2-C8-alkynyloxy, C2-C8-haloalkynyl, NH2, C1-C8-alkylamino, di-C1-C8-alkylamino, phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, X is hydrogen, halogen, OH, cyano, C1-C4-alkyl and the like, Y is hydrogen, halogen, cyano, C1-C4-alkyl and the like.

公开(公告)号：US06613931B1

公开(公告)日：2003-09-02

申请号：US09913978

申请日：2001-08-21

申请人： Oliver Wagner ,  Thomas Grote ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Klaus Grossmann

发明人： Oliver Wagner ,  Thomas Grote ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Klaus Grossmann

IPC分类号： C07C25503

CPC分类号： C07C255/41 ,  A01N37/34

摘要： The resent invention relates to the use of phenylacetamides as crop protection agents, to novel crop protection compositions comprising, as active compounds, phenylacetamides, and to novel phenylacetamides. The present invention provides the use of phenylacetamides of the formula I as crop protection agents having herbicidal and/or fungicidal action, where the radicals have the following meanings: A is an unsubstituted or substituted aryl radical; R1 is an unsubstituted or substituted aryl radical; R2, R3 are hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C3-C7-cycloalkyl, C1-C6-alkylaryl, which may be unsubstituted or partially or fully halogenated or may carry one to three substituents selected from the group consisting of C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkylthio, C3-C7-cycloalkyl, C5-C7-cycloalkenyl; R4 is hydrogen or C1-C6-alkyl; R5 is hydroxyl, C1-C4-alkoxy, aryl-C1-C4-alkoxy, aryloxy, and their agriculturally useful salts.

摘要翻译： 本发明涉及苯基乙酰胺作为作物保护剂的用途，作为新的作物保护组合物，其包含作为活性化合物的苯乙酰胺和新的苯乙酰胺。本发明提供了下式的苯基乙酰胺的用途：具有除草和 /或杀真菌作用，其中基团具有以下含义：A是未取代或取代的芳基; R 1是未取代或取代的芳基; R 2，R 3是氢，C 1 -C 6 - 烷基，C 2 -C 6 - 烯基，C 3 C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷基芳基， C 3 -C 7 - 环烷基，C 5 -C 7 - 环烯基; R 4是氢或C 1 -C 6烷基; R 5是羟基，C 1 -C 4 - 烷氧基，芳基-C 1 -C 4 - 烷氧基，芳氧基和它们的农业上有用的盐。

公开(公告)号：US5831093A

公开(公告)日：1998-11-03

申请号：US860671

申请日：1997-07-07

申请人： Norbert Gotz ,  Bernd Muller ,  Hubert Sauter ,  Joachim Gebhardt ,  Oliver Wagner

发明人： Norbert Gotz ,  Bernd Muller ,  Hubert Sauter ,  Joachim Gebhardt ,  Oliver Wagner

IPC分类号： B01J23/42 ,  B01J23/44 ,  C07B61/00 ,  C07C239/10 ,  C07C239/12 ,  C07C251/48 ,  C07C253/30 ,  C07C255/64 ,  C07D213/76 ,  C07D215/38 ,  C07D215/40 ,  C07D231/22 ,  C07D239/54 ,  C07D249/12 ,  C07D471/04 ,  C07D239/10 ,  C07D211/72 ,  C07D239/00 ,  C07D249/04

CPC分类号： C07D213/76 ,  C07C239/10 ,  C07C239/12 ,  C07C251/48 ,  C07C253/30 ,  C07D215/38 ,  C07D215/40 ,  C07D231/22 ,  C07D239/54 ,  C07D249/12 ,  C07D471/04

摘要： A process for preparing aromatic or heteroaromatic hydroxylamines of the general formula I ##STR1## where R.sup.1 is an unsubstituted or substituted aryl radical or an unsubstituted or substituted hetaryl radical from the pyridine or quinoline groups, by hydrogenation of nitro compounds of the general formula II R.sup.1 --NO.sub.2 (II) where R.sup.1 has the meaning indicated above, in the presence of a platinum catalyst on an activated carbon support or in the presence of a palladium catalyst doped with sulfur or selenium on an activated carbon support, by carrying out the reaction in the presence of a nitrogen-substituted morpholine compound of the general formula III ##STR2## R.sup.2 being alkyl radicals having 1 to 5 carbon atoms and R.sup.3 to R.sup.10 being hydrogen atoms or alkyl radicals having 1 to 5 carbon atoms is described.

摘要翻译： PCT No.PCT / EP96 / 00170 Sec。 371日期1997年7月7日 102（e）日期1997年7月7日PCT 1996年1月17日PCT PCT。 第WO96 / 22967号公报 日本1996年8月1日制备通式Ⅰ（I）的芳族或杂芳族羟胺的方法，其中R 1为未取代或取代的芳基或未取代或取代的杂芳基，通过氢化吡啶或喹啉基 通式IIR1-NO2（II）的硝基化合物，其中R 1具有上述含义，在铂催化剂存在下，在活性炭载体上或在活性炭载体上掺杂有硫或硒的钯催化剂存在下， 通过在通式III（III）的氮取代的吗啉化合物的存在下进行反应，R2是具有1至5个碳原子的烷基，R3至R10是氢原子或具有1至 描述了5个碳原子。

公开(公告)号：US6069144A

公开(公告)日：2000-05-30

申请号：US11610

申请日：1998-02-12

申请人： Oliver Wagner ,  Frank Wetterich ,  Karl Eicken ,  Michael Rack ,  Gerhard Hamprecht ,  Gunther Lamm ,  John-Bryan Speakman ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann

发明人： Oliver Wagner ,  Frank Wetterich ,  Karl Eicken ,  Michael Rack ,  Gerhard Hamprecht ,  Gunther Lamm ,  John-Bryan Speakman ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann

IPC分类号： A01N43/40 ,  A01N43/42 ,  A01N43/54 ,  A01N43/78 ,  A01N43/90 ,  C07D213/70 ,  C07D213/71 ,  C07D213/82 ,  C07D213/85 ,  C07D215/54 ,  C07D239/38 ,  C07D277/74 ,  C07D277/76 ,  C07D513/04 ,  A01N43/58 ,  A61K31/505 ,  C07D211/36 ,  C07D215/16 ,  C07D515/02

CPC分类号： C07D213/70 ,  A01N43/40 ,  A01N43/42 ,  A01N43/54 ,  A01N43/78 ,  A01N43/90 ,  C07D213/71 ,  C07D213/82 ,  C07D213/85 ,  C07D215/54 ,  C07D239/38 ,  C07D277/74 ,  C07D277/76 ,  C07D513/04

摘要： N-heterocyclic compounds I ##STR1## or their salts or N-oxides, wherein A is an N-heterocycle selected from the group consisting of ##STR2## R.sup.1 -R.sup.6, R.sup.24 -R.sup.26 are hydrogen, cyano, nitro, halogen, aminocarbonyl, methylsulfonyl, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, alkoxyalkyl, alkoxycarbonyl, aryl or aryloxy;m is 0, 1 or 2;Alk is optionally substituted 1,2-ethylidene, 1,3-propylidene cycloalkyl or cycloalkenyl;X is oxygen or sulfur;Q is optionally substituted aryl, cycloalkyl, cycloalkenyl, or arylalkyl;their manufacture and suitable intermediates therefore, as well as compositions comprising them and their use for controlling harmful fungi.

摘要翻译： PCT No.PCT / EP96 / 03680 Sec。 371日期1998年2月12日 102（e）1998年2月12日PCT PCT 1996年8月21日PCT公布。 公开号WO97 / 08147 日期1997年3月6日N-杂环化合物I或其盐或N-氧化物，其中A为选自由R 1 -R 6，R 24-R 26组成的组的N-杂环为氢，氰基，硝基，卤素，氨基羰基，甲基磺酰基 烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，烷氧基烷基，烷氧基羰基，芳基或芳氧基; m为0,1或2; Alk是任选取代的1,2-亚乙基，1,3-亚丙基环烷基或环烯基; X是氧或硫; Q是任选取代的芳基，环烷基，环烯基或芳基烷基; 因此它们的制造和合适的中间体，以及包含它们的组合物及其用于控制​​有害真菌的用途。