Fungicidal and plant growth-regulating hydroxyethyl-azolyl derivatives
    52.
    发明授权
    Fungicidal and plant growth-regulating hydroxyethyl-azolyl derivatives 失效
    杀真菌剂和植物生长调节羟乙基 - 唑基衍生物

    公开(公告)号:US4938791A

    公开(公告)日:1990-07-03

    申请号:US211799

    申请日:1988-06-24

    摘要: Fungicidal and plant growth regulating hydroxyethylazolyl derivatives of the formula ##STR1## in which R represents hydrogen, alkyl or acyl,R.sup.1 represents halogen, optionaly substituted phenyl or the grouping --Z--R.sup.3, whereinZ represents oxygen, sulphur, SO or SO.sub.2 andR.sup.3 represents optionally substituted phenyl,R.sup.2 represents halogen, alkyl having 1 to 4 carbon atoms, alkoxy having 1 to 4 carbon atoms, alkylthio having 1 to 4 carbon atoms, halogenoalkyl having 1 or 2 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 or 2 carbon atoms and 1 to 5 halogen atoms, halogenoalkylthio having 1 or 2 carbon atoms and 1 to 5 halogen atoms, alkoximinomethyl with 1 to 4 carbon atoms in the alkoxy group, phenyl which is optionally substituted by alkyl having 1 or 2 carbon atoms and/or halogen, or phenoxy, which is optionally substituted by alkyl having 1 or 2 carbon atoms and/or halogen,m represents the number 0, 1, 2 or 3,X represents nitrogen or a CH group andY represents oxygen, sulphur, SO or SO.sub.2,and addition products thereof with acids and metal salts. Intermediates of the formulas ##STR2## are also new.

    摘要翻译: 杀真菌剂和植物生长调节下式(I)的羟乙基唑基衍生物,其中R表示氢,烷基或酰基,R 1表示卤素,任选取代的苯基或基团-Z-R 3,其中Z表示氧,硫,SO或 SO 2和R 3表示任选取代的苯基,R 2表示卤素,具有1至4个碳原子的烷基,具有1至4个碳原子的烷氧基,具有1至4个碳原子的烷硫基,具有1或2个碳原子的卤代烷基和1至5个卤素原子, 具有1或2个碳原子和1至5个卤素原子的卤代烷氧基,具有1或2个碳原子和1至5个卤素原子的卤代烷硫基,烷氧基中具有1至4个碳原子的烷基亚氨基甲基,任选被具有1或 2个碳原子和/或卤素,或苯氧基,其任选被具有1或2个碳原子的烷基和/或卤素取代,m表示数0,1,2或3,X表示氮或CH基,Y表示 氧, 硫,SO或SO 2,以及其与酸和金属盐的加成产物。 (VII)(IV)(XII)的中间体也是新的。

    N-arylcarbamic acid esters
    53.
    再颁专利
    N-arylcarbamic acid esters 失效
    N-芳基氨基甲酸酯

    公开(公告)号:USRE30578E

    公开(公告)日:1981-04-14

    申请号:US853971

    申请日:1977-11-22

    摘要: New N-arylcarbamic acid esters of the formula ##STR1## in which R is lower aliphatic hydrocarbyl, optionally substituted,R.sup.1, R.sup.2 and R.sup.3, which may be identical or different, are each hydrogen, alkyl, cycloalkyl, alkoxy, haloalkyl or halogen,R.sup.4 is alkyl, alkenyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxyalkyl or alkylthioalkyl, acylalkyl (i.e., alkanoyloxyalkyl), alkoxycarbonylalkyl, carbalkoxyalkyl, carbalkoxyalkenyl, or an optionally substituted cycloalkyl, aryl, aralkyl, aryloxyalkyl or arylthioalkyl radical, or the grouping ##STR2## wherein R.sup.4' is hydrogen or is defined as R.sup.4 is defined above, andY and Y' are oxygen or sulfur,are outstandingly effective in regulating the growth of plants, i.e., to inhibit, stimulate or alter the growth of plants.

    N-Arylcarbamic acid esters and plant growth regulant compositions and
methods
    54.
    发明授权
    N-Arylcarbamic acid esters and plant growth regulant compositions and methods 失效
    N-芳基氨基甲酸酯和植物生长调节剂组合物和方法

    公开(公告)号:US4093447A

    公开(公告)日:1978-06-06

    申请号:US632742

    申请日:1975-11-17

    摘要: New N-arylcarbamic acid esters of the formula ##STR1## in which R is lower aliphatic hydrocarbyl, optionally substituted,R.sup.1, r.sup.2 and R.sup.3, which may be identical or different, are each hydrogen, alkyl, cycloalkyl, alkoxy, haloalkyl or halogen,R.sup.4 is alkyl, alkenyl, alkynyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxyalkyl or alkylthioalkyl, acylalkyl (i.e., alkanoyloxyalkyl), alkoxycarbonylalkyl, carbalkoxyalkyl, carbalkoxyalkenyl, or an optionally substituted cycloalkyl, aryl, aralkyl, aryloxyalkyl or arylthioalkyl radical, or the grouping ##STR2## wherein R.sup.4' is hydrogen or is defined as R.sup.4 is defined above, andY and Y' are oxygen or sulfur.Are outstanding effective in regulating the growth of plants, i.e., to inhibit, stimulate or alter the growth of plants.

    摘要翻译: 其中R是低级脂族烃基,任选被取代的,可以相同或不同的R 1,R 2和R 3的新的N-芳基氨基甲酸酯,其中R 1是氢,烷基,环烷基,烷氧基,卤代烷基 或卤素,R4是烷基,烯基,炔基,环烯基,卤代烷基,卤代烯基,卤代炔基,烷氧基烷基或烷硫基烷基,酰基烷基(即烷酰氧基烷基),烷氧基羰基烷基,碳烷氧基烷基,碳烷氧基烯基或任选取代的环烷基,芳基,芳烷基,芳氧基烷基或芳硫基烷基 或者其中R4'为氢或被定义为R4的分组“IMAGE”定义如上,Y和Y'为氧或硫。

    Substituted triazolinone herbicides and plant growth regulators
    56.
    发明授权
    Substituted triazolinone herbicides and plant growth regulators 失效
    取代的三唑啉酮除草剂和植物生长调节剂

    公开(公告)号:US5523409A

    公开(公告)日:1996-06-04

    申请号:US125975

    申请日:1993-09-23

    摘要: Novel herbicides and plant growth regulants of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, alkoxy, cycloalkylalkyl or cycloalkyl, or represents in each case optionally substituted aralkyl or aryl,R.sup.2 represents a radical ##STR2## or represents a radical --S(O).sub.n --R.sup.7, R.sup.3 and R.sup.4 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylaminoalkyl, alkoxycarbonylalkyl or alkoxycarbonylalkenyl, or represent in each case optionally substituted cycloalkyl, cycloalkylalkyl, cycloalkenyl or cycloalkenylalkyl, or represent optionally substituted heterocyclylalkyl, or represent in each case optionally substituted aralkyl, aroyl or aryl, or represent alkoxy, alkenyloxy, alkinyloxy, aralkyloxy or aryloxy, or, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical,X represents oxygen or sulphur andY represents oxygen or sulphur,whereinR.sup.5 and R.sup.6 independently of one another each represent alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, alkoxy, cycloalkyl or cycloalkylalkyl, or represent in each case optionally substituted aryl, aralkyl or heteroaryl, or, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical,R.sup.7 represents alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkylalkyl, or represents in each case optionally substituted aralkyl or aryl andn represents the number 0, 1 or 2,but wherein R.sup.2 only represents a radical --S(O).sub.n --R.sup.7 if R.sup.3 and R.sup.4 do not simultaneously represent methyl.Intermediates therefor where NR.sup.3 R.sup.4 is replaced by Cl are also new.

    摘要翻译: 式(I)的新型除草剂和植物生长调节剂,其中R 1表示氢,烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,烷氧基烷基,烷氧基,环烷基烷基或环烷基,或在每种情况下表示任选取代的芳烷基或 芳基,R 2表示基团,或表示基团-S(O)n -R 7,R 3和R 4彼此独立地表示氢,烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,氰基烷基,羟基烷基,烷氧基烷基 或烷基氨基烷基,烷氧基羰基烷基或烷氧基羰基烯基,或在每种情况下表示任选取代的环烷基,环烷基烷基,环烯基或环烯基烷基,或代表任选取代的杂环基烷基,或在每种情况下表示任选取代的芳烷基,芳酰基或芳基,或代表烷氧基,烯氧基,烷氧基,芳烷氧基 或芳氧基,或者与它们所键合的氮原子一起代表任选的 取代的杂环基,X表示氧或硫,Y表示氧或硫,其中R5和R6彼此独立地表示烷基,烯基,炔基,卤代烷基,卤代烯基,卤代烷基,烷氧基烷基,烷氧基,环烷基或环烷基烷基,或各自表示 任选取代的芳基,芳烷基或杂芳基,或与它们所键合的氮原子一起表示任选取代的杂环基,R 7表示烷基,烯基,炔基,环烷基或环烷基烷基,或在每种情况下表示任选取代的芳烷基或 芳基,n表示数字0,1或2,但如果R3和R4不同时表示甲基,则其中R2仅表示基团-S(O)n-R7。 NR3R4被Cl取代的中间体也是新的。

    Isoxazolecarboxylic acid derivatives
    58.
    发明授权
    Isoxazolecarboxylic acid derivatives 失效
    异恶唑羧酸衍生物

    公开(公告)号:US5374605A

    公开(公告)日:1994-12-20

    申请号:US2307

    申请日:1993-01-08

    摘要: The invention relates to isoxazolecarboxylic acid derivatives of the general formula (I) ##STR1## in which A represents alkanediyl,Q represents oxygen, sulphur, imino (NH) or alkylimino (N-alkyl),R.sup.1 represents an in each case optionally substituted radical from the series comprising alkyl, cycloalkyl or phenyl,R.sup.2 represents hydrogen, halogen or optionally substituted alkyl, andR.sup.3 represents in each case optionally substituted cyclohexyl or phenyl,with the exception of the compounds: N-benzyl-5-cyclopropyl-isoxazole-3-carboxamide N-(2-phenyl-ethyl)-5-methyl-isoxazole-3-carboxamide and N-benzyl-5-methyl-isoxazole-3-carboxamide, a process for their preparation, and their use as herbicides.

    摘要翻译: 本发明涉及通式(I)的化合物(I)的异恶唑羧酸衍生物,其中A代表烷二基,Q代表氧,硫,亚氨基(NH)或烷基亚氨基(N-烷基),R1代表每种情况 任选取代的烷基,环烷基或苯基系列的取代基,R 2表示氢,卤素或任选取代的烷基,R 3表示在任何情况下均为任选取代的环己基或苯基,但化合物除外:N-苄基-5-环丙基 - 异恶唑-3-甲酰胺N-(2-苯基 - 乙基)-5-甲基 - 异恶唑-3-甲酰胺和N-苄基-5-甲基 - 异恶唑-3-甲酰胺,其制备方法及其作为除草剂的用途 。