摘要:
5-Alkyl-7-aminotriazolopyrimidines of the formula I, where: R1, R2 are hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cycloalkyl, phenyl, naphthyl; 5- or 6-membered saturated, unsaturated or aromatic heterocyclyl which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or R1 and R2 together with the bridging nitrogen atom can form a 5- or 6-membered ring which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 is cycloalkyl or bicycloalkyl; where R1, R2 and R3 may be substituted as outlined in the description; X is alkyl or haloalkyl; and their salts; processes and intermediates for their preparation, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.
摘要:
6-(2-Halo-4-alkoxyphenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, phenylalkyl, mono- or dialkoxyalkyl; R1, R2 and/or R3 may be substituted as mentioned in the description; L is hydrogen, fluorine or chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要翻译:其中取代基如下定义的式I的6-(2-卤代-4-烷氧基苯基)三唑并嘧啶:R 1是烷基,卤代烷基,环烷基,卤代环烷基,烯基,卤代烯基,环烯基,卤代环烯基 ,炔基,卤代炔基或苯基,萘基或五元或六元饱和的部分不饱和或芳族杂环,其含有一至四个由O,N和S组成的组的杂原子,R 2, 是氢或R 1,R 1和R 2所提及的基团之一与它们所连接的氮原子一起也可以 形成通过N连接的五元或六元杂环基或杂芳基,并且可以含有一个至三个由O,N和S组成的组的另外的杂原子作为环成员; R 3是烷基,卤代烷基,烯基,卤代烯基,炔基,卤代炔基,苯基烷基,单或二烷氧基烷基; R 1,R 2和/或R 3可以如说明书中所述被取代; L是氢,氟或氯; X是氰基,烷基,烷氧基,烯氧基,卤代烷氧基或卤代烯氧基; 制备这些化合物的方法,包含它们的组合物及其用于控制植物病原性有害真菌的用途。
摘要:
The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R2 represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R1 and/or R2 being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.
摘要翻译:本发明涉及式(I)的5,6-二烷基-7-氨基 - 三唑并嘧啶,其中取代基定义如下:R 1表示烷基,烷氧基烷基,烯基或炔基; R 2表示根据描述被取代的烷基,烷氧基烷基,烯基或炔基,R 1和/或R 2 2。 本发明还涉及一种生产所述化合物的方法,含有后者的药剂及其用于控制植物致病真菌的用途。
摘要:
The invention relates to 6-(2,3,6-trifluorophenyl)-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R2 represents hydrogen or one of the groups cited for R1; R1 and R2, together with the nitrogen atom, to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded via N and can contain one to three additional heteroatoms from the groups O, N and S as a ring member; R1 and/or R2 can be substituted in accordance with the description; X represents cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy. The invention also relates to methods for producing said compounds, to agents containing the latter and to their use for combating plant-pathogenic fungi.
摘要翻译:本发明涉及式(I)的6-(2,3,6-三氟苯基) - 三唑并嘧啶,其中取代基定义如下:R 1表示烷基,卤代烷基,环烷基,卤代环烷基, 烯基,卤代烯基,环烯基,卤代环烯基,炔基,卤代炔基或苯基,萘基或含有一至四个O,N或S基的杂原子的五元或六元饱和的部分不饱和或芳族杂环; R 2表示氢或R 1所引用的基团之一; R 1和R 2与它们所键合的氮原子一起也可以形成五或六元杂环基或杂芳基,其通过 并且可以含有一个至三个作为环成员的来自基团O,N和S的另外的杂原子; R 1和/或R 2可以根据描述代替; X表示氰基,烷基,烷氧基,烯氧基,卤代烷氧基或卤代烯氧基。 本发明还涉及生产所述化合物的方法,含有后者的试剂和用于对抗植物致病性真菌的用途。
摘要:
6-(2,4,6-Trifluorophenyl)triazolopyrimidines of the formula I in which the substituents have the following meanings: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl, cycloalkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned in R1, R1 and R2 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered ring which is interrupted by an atom from the group consisting of O, N and S, and/or R1 and/or R2 can be substituted according to the description; X is cyano, C1-C4-alkoxy, C3-C4-alkenyloxy, C1-C2-haloalkoxy or C3-C4-halo-alkenyloxy; process for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.
摘要:
The invention relates to 5,6-cycloalkyl-7-aminotriazolopyrimidines of formula (I), where X=alkylene or alkenylene, whereby the carbon chain can be interrupted by one or two heteroatoms selected from S, O or NR1, R1═H, alkyl or C(═O)alkyl, L=halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyl, alkinyl or NR2R3; R2,R3=each one of the groups given for R1 and m=a whole number from 0 to 5, whereby the aliphatic groups can be substituted by one to three of the following groups: halogen, cyano, nitro, hydroxy, alkoxy, alkylthio, or NRaRb, where Ra, Rb═H or alkyl in which the carbon chains can be halogenated. The invention further relates to methods for production of said compounds, agents comprising the same and use thereof for the prevention of fungal pests harmful to plants.
摘要翻译:本发明涉及式(I)的5,6-环烷基-7-氨基三唑并嘧啶,其中X =亚烷基或亚烯基,其中碳链可被一个或两个选自S,O或NR 1的杂原子中断, 卤素,氰基,硝基,烷基,卤代烷基,烷氧基,卤代烷氧基,烯基,炔基或NR 2(O) 3 SUP> 3 SUP> R 2,R 3 =每个给定R 1的基团,m = 0至5的整数,由此脂族基 基团可以被一至三个以下基团取代:卤素,氰基,硝基,羟基,烷氧基,烷硫基或NR a R b,其中R 0, 或其中碳链可以被卤化的烷基。 本发明还涉及生产所述化合物的方法,包含该化合物的试剂及其用于预防对植物有害的真菌害虫的用途。
摘要:
Bicyclic compounds of the formula I in which A1 or A5 is C and the other of the two variables A1, A5 is N, C or C—R3; A2, A3, A4 independently of one another are N or C—R3a, where one of the variables A2, A3 or A4 may also be S or a group N—R4 if A1 and A5 are both C, and where A4 is not N or C—R3a if A1 is N, A3 is C—R3a and A5 is C, and where A1 is attached to A2 and A3 to A4 or A2 is attached to A3 and A4 to A5 or A1 is attached to A5 and A2 to A3 or A1 is attached to A5 and A3 to A4 or A1 is attached to A2 and A4 to A5 by double bonds; n is 0, 1, 2, 3, 4 or 5; Ra is halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R5; R1 is halogen, cyano, C1-C10-alkyl, where a carbon atom of the C1-C10-alkyl radical may be replaced by a silicium atom, C1-C6-haloalkyl, C2-C10-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, where the cycloalkyl moiety of the two last-mentioned groups may be unsubstituted or contain 1, 2, 3, 4, 5, or 6 radicals selected from the group consisting of C1-C4-alkylidene, C1-C4-alkyl, halogen, C1-C4-haloalkyl and hydroxy and the alkyl moiety of C3-C8-cycloalkyl-C1-C4-alkyl may be unsubstituted or contain 1, 2, 3, or 4 radicals selected from the group consisting of halogen, C1-C4-haloalkyl and hydroxy, C5-C8-cycloalkenyl which may be unsubstituted or contain 1, 2, 3 or 4 radicals selected from the group consisting of C1-C4-alkyl, halogen, C1-C4-haloalkyl and hydroxy, OR6, SR6, NR7R8, a radical of the formula —C(R11)(R12)C(═NOR13)(R14) or a radical of the formula —C(═NOR15)C(═NOR16)(R17); R2 is halogen, cyano, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C5-C8-cycloalkenyl, OR6, SR6 or NR7R8; and the agriculturally acceptable salts of the compounds I, crop protection compositions comprising at least one compound of the formula I and/or an agriculturally acceptable salt of I and at least one solid or liquid carrier and a method for controlling phytopathogenic harmful fungi are described.
摘要:
The invention relates to 7-aminomethyl-1,2,4-triazolo[1,5-a]pyrimidine compounds of general formula (I) and the agriculturally compatible salts of said compounds. In said formula: R1 and R2 represent hydrogen, alkyl, haloalkyl, alkoxy, cycloalkyl, bicycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1 to 4 heteroatoms from the group containing O, N or S, or R1 and R2, together with the nitrogen atom to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded by means of N and can contain 1 to 3 additional heteroatoms from the group containing O, N and S as the ring member and can be substituted according to the description; R3 and R4 represent hydrogen, alkyl, haloalkyl, haloalkoxy, alkoxy, or alkoxyalkyl; X represents halogen, cyano, a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1, 2 or 3 heteroatoms from the group containing O, N or S as the ring member, alkyl, alkoxy, alkenyl or alkynyl, whereby the latter 4 groups can be substituted according to the description; L is defined as cited in the claims and the description; and m represents 0, 1, 2, 3, 4 or 5. The invention also relates to the use of the triazolopyrimidine compounds of general formula (I) and their agriculturally compatible salts for controlling plant-pathogenic fungi, to a method for controlling plant-pathogenic fungi, containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound and at least one liquid or solid carrier.
摘要:
6-Pentafluorophenyltriazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy, processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
摘要翻译:式I的6-五氟苯基三唑并嘧啶,其中取代基如下:R 1是烷基,卤代烷基,环烷基,卤代环烷基,烯基,卤代烯基,环烯基,卤代环烯基,炔基,卤代炔基或苯基,萘基, 或五元或六元饱和,部分不饱和或芳族杂环,其含有一至四个由O,N和S组成的组的杂原子,R 2是氢或下述基团之一 R 1,R 1和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基 或杂芳基,其通过N连接并且可以含有一个至三个由O,N和S组成的组的另外的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; X是氰基,烷基,烷氧基,烯氧基,卤代烷氧基或卤代烯氧基,制备这些化合物的方法,包含它们的组合物及其用于控制植物病原性有害真菌的用途。
摘要:
Triazolopyrimidines of the formula I in which the substituents are as defined below: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and may be substituted as defined in the description; L1, L2 are hydrogen, cyano, haloalkyl, alkoxy, alkenyloxy or C(═O)A, where at least one group L1 or L2 is not hydrogen; A is hydrogen, hydroxyl, alkyl, alkoxy, haloalkoxy, C1-C8-alkylamino or dialkylamino; L3 is hydrogen, halogen, cyano, nitro, haloalkyl, alkoxy or alkoxycarbonyl; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.