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公开(公告)号:US5028698A
公开(公告)日:1991-07-02
申请号:US464695
申请日:1990-01-18
申请人: Yukiko Tone , Toshiro Iwahashi , Etsuko Ohkouchi , Hiroshi Kitagawa , Isamu Sugawara , Hiroshi Okazaki , Akio Fukuda , Hans G. Berscheid , Hitoko Numata , Junko Usui , Shunji Senda , Akihiko Matsuo , Hiroshi Watanabe , Itsuo Kurobane
发明人: Yukiko Tone , Toshiro Iwahashi , Etsuko Ohkouchi , Hiroshi Kitagawa , Isamu Sugawara , Hiroshi Okazaki , Akio Fukuda , Hans G. Berscheid , Hitoko Numata , Junko Usui , Shunji Senda , Akihiko Matsuo , Hiroshi Watanabe , Itsuo Kurobane
IPC分类号: A61K31/35 , A61K31/70 , A61K31/7028 , A61K31/7034 , A61K31/704 , A61K39/395 , A61P35/00 , C07D493/14 , C07H15/252 , C07K16/30
CPC分类号: C07H15/252
摘要: Cytorhodin S derivatives, especially cytorhodin S-immunoglobulin complexes are disclosed. Cytorhodin S possesses very high anticancer activity, but the complexes act more selectively on cancer cells and are more useful as an anticancer agent. New intermediate derivatives are also useful as an anticancer agent.
摘要翻译: 公开了细胞因子S衍生物,特别是细胞因子S-免疫球蛋白复合物。 细胞因子S具有非常高的抗癌活性,但复合物对癌细胞的选择性更高,更可用作抗癌剂。 新的中间体衍生物也可用作抗癌剂。