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公开(公告)号:US20060141448A1
公开(公告)日:2006-06-29
申请号:US11354387
申请日:2006-02-15
申请人: Frank Fan , Yinduo Ji , Howard Kallender , Tong Li , Damien McDevitt
发明人: Frank Fan , Yinduo Ji , Howard Kallender , Tong Li , Damien McDevitt
CPC分类号: G01N33/5023 , C12N9/1096 , G01N33/5008
摘要: This invention relates to newly developed methods for discovering therapeutic compounds using a cell-based assay system. This invention also relates to compositions of matter useful in carrying out the methods of the invention as well as therapeutic compounds developed using such methods.
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公开(公告)号:US06489139B1
公开(公告)日:2002-12-03
申请号:US09339614
申请日:1999-06-24
IPC分类号: C12N1500
摘要: The invention provides fabZ polypeptides and polynucleotides encoding fabZ polypeptides and methods for producing such polypeptides by recombinant techniques. Also provided are methods for utilizing fabZ polypeptides to screen for antibacterial compounds.
摘要翻译: 本发明提供编码fabZ多肽的fabZ多肽和多核苷酸以及通过重组技术产生此类多肽的方法。 还提供了利用fabZ多肽筛选抗菌化合物的方法。
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公开(公告)号:US06451556B1
公开(公告)日:2002-09-17
申请号:US09218197
申请日:1998-12-21
IPC分类号: C12P2106
摘要: The invention provides EF-Tu polypeptides and polynucleotides encoding EF-Tu polypeptides and methods for producing such polypeptides by recombinant techniques. Also provided are methods for utilizing EF-Tu polypeptides to screen for antibacterial compounds.
摘要翻译: 本发明提供了EF-Tu多肽和编码EF-Tu多肽的多核苷酸以及通过重组技术产生此类多肽的方法。 还提供了利用EF-Tu多肽筛选抗菌化合物的方法。
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公开(公告)号:US20130252956A1
公开(公告)日:2013-09-26
申请号:US13988561
申请日:2011-11-21
申请人: Howard Kallender , Lone Ottesen
发明人: Howard Kallender , Lone Ottesen
IPC分类号: A61K31/5377
CPC分类号: A61K31/5377
摘要: Methods for treating a human having heptocellular carcinoma comprising administering to the human a therapeutically effective amount of Compound A: or a pharmaceutically acceptable salt thereof, wherein the human has a complete response or partial response.
摘要翻译: 用于治疗患有肝细胞癌的人的方法包括向人施用治疗有效量的化合物A或其药学上可接受的盐,其中所述人具有完全反应或部分反应。
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公开(公告)号:US06448038B1
公开(公告)日:2002-09-10
申请号:US09237119
申请日:1999-01-26
IPC分类号: C12P2106
CPC分类号: C12N9/93 , A61K38/00 , C12Y603/04015
摘要: The invention provides birA polypeptides and polynucleotides encoding birA polypeptides and methods for producing such polypeptides by recombinant techniques. Also provided are methods for utilizing birA polypeptides to screen for antibacterial compounds.
摘要翻译: 本发明提供了birA多肽和编码birA多肽的多核苷酸以及通过重组技术产生此类多肽的方法。 还提供了利用birA多肽筛选抗菌化合物的方法。
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公开(公告)号:US06331411B1
公开(公告)日:2001-12-18
申请号:US09153277
申请日:1998-09-15
申请人: Michael Gwynn , Howard Kallender , Lisa K Katz , Daniel Sylvester , Christopher M Traini , Richard Lloyd Warren
发明人: Michael Gwynn , Howard Kallender , Lisa K Katz , Daniel Sylvester , Christopher M Traini , Richard Lloyd Warren
IPC分类号: C12N510
CPC分类号: C12N9/90 , A61K38/00 , C07K14/3156 , C12Q1/689
摘要: The invention provides topA polypeptides and polynucleotides encoding topA polypeptides and methods for producing such polypeptides by recombinant techniques. Also provided are methods for utilizing topA polypeptides to screen for antibacterial compounds.
摘要翻译: 本发明提供了topA多肽和编码topA多肽的多核苷酸以及通过重组技术产生此类多肽的方法。 还提供了利用topA多肽筛选抗菌化合物的方法。
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公开(公告)号:US06207449B1
公开(公告)日:2001-03-27
申请号:US09213081
申请日:1998-12-16
申请人: Howard Kallender
发明人: Howard Kallender
IPC分类号: C12N1500
CPC分类号: C07K14/3156 , A61K38/00 , A61K39/00 , A61K2039/51 , Y10S530/806 , Y10S530/825
摘要: The invention provides gidB polypeptides and DNA (RNA) encoding gidB polypeptides and methods for producing such polypeptides by recombinant techniques. Also provided are methods for utilizing gidB polypeptides to screen for antibacterial compounds.
摘要翻译: 本发明提供gidB多肽和编码gidB多肽的DNA(RNA),以及通过重组技术产生此类多肽的方法。 还提供了利用gidB多肽筛选抗菌化合物的方法。
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公开(公告)号:US06294357B1
公开(公告)日:2001-09-25
申请号:US09386875
申请日:1999-08-31
IPC分类号: C07K1431
CPC分类号: C12N9/1029 , A61K38/00 , A61K48/00
摘要: The invention provides fabF polypeptides and polynucleotides encoding fabF polypeptides and methods for producing such polypeptides by recombinant techniques. Also provided are methods for utilizing fabF polypeptides to screen for antibacterial compounds.
摘要翻译: 本发明提供了fabF多肽和编码fabF多肽的多核苷酸以及通过重组技术产生此类多肽的方法。 还提供了利用fabF多肽筛选抗菌化合物的方法。
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公开(公告)号:US06238882B1
公开(公告)日:2001-05-29
申请号:US09104068
申请日:1998-06-24
申请人: Jason Craig Fedon , Deborah D Jaworski , Howard Kallender , Anna Lisa Lenox , Leslie Marie Palmer , Min Wang
发明人: Jason Craig Fedon , Deborah D Jaworski , Howard Kallender , Anna Lisa Lenox , Leslie Marie Palmer , Min Wang
IPC分类号: C12P2106
CPC分类号: C07K14/3156 , A61K38/00 , A61K48/00 , C07K2319/00
摘要: The invention provides gidA1 polypeptides and polynucleotides encoding gidA1 polypeptides and methods for producing such polypeptides by recombinant techniques. Also provided are methods for utilizing gidA1 polypeptides to screen for antibacterial compounds.
摘要翻译: 本发明提供gidA1多肽和编码gidA1多肽的多核苷酸以及通过重组技术产生此类多肽的方法。 还提供了利用gidA1多肽筛选抗菌化合物的方法。
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公开(公告)号:US06228364B1
公开(公告)日:2001-05-08
申请号:US09360682
申请日:1999-07-26
IPC分类号: A61K3902
CPC分类号: C07K14/295 , A61K39/00 , A61K48/00
摘要: The invention provides gidA1 polypeptides and DNA (RNA) encoding gidA1 polypeptides and methods for producing such polypeptides by recombinant techniques. Also provided are methods for utilizing gidA1 polypeptides to screen for antibacterial compounds.
摘要翻译: 本发明提供了gidA1多肽和编码gidA1多肽的DNA(RNA)以及通过重组技术产生此类多肽的方法。 还提供了利用gidA1多肽筛选抗菌化合物的方法。
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