Pyrroles possessing insecticidal activity
    2.
    发明授权
    Pyrroles possessing insecticidal activity 失效
    PYRROLES POSSESSING INSECTICIDAL活动

    公开(公告)号:US5164409A

    公开(公告)日:1992-11-17

    申请号:US661399

    申请日:1991-02-26

    CPC分类号: C07D207/333 A01N53/00

    摘要: All possible stereoisomers and mixtures of a compound of the formula ##STR1## wherein X and Y are different and are selected from the group consisting of hydrogen, halogen, --CN, alkyl and haloalkyl of 1 to 8 carbon atoms and phenyl optionally substituted by at least one member of the group consisting of halogen and alkyl and alkoxy of 1 to 8 carbon atoms, R.sub.1 is selected from the group consisting of hydrogen, methyl, --CN and ethynyl, ##STR2## A and B are individually selected from the group consisting of hydrogen, halogen, alkyl of 1 to 8 carbon atoms and aryl of 6 to 14 carbon atoms and the --CF.sub.3 is in the 2-, 4- or 5-position of the pyrrole ring having pesticidal activity.

    摘要翻译: 式(I)化合物的所有可能的立体异构体和混合物,其中X和Y不同,并且选自氢,卤素,-CN,具有1至8个碳原子的烷基和卤代烷基,以及任选的苯基 被至少一个由卤素和1至8个碳原子的烷基和烷氧基组成的组取代,R 1选自氢,甲基,-CN和乙炔基,A和B分别选自 由氢,卤素,碳原子数1〜8的烷基和碳原子数为6〜14的芳基构成的基团,在具有杀虫活性的吡咯环的2-,4-或5-位。

    Novel pyrethrinoids
    8.
    发明授权
    Novel pyrethrinoids 失效
    新型拟除虫菊酯类

    公开(公告)号:US4925862A

    公开(公告)日:1990-05-15

    申请号:US221948

    申请日:1988-07-20

    摘要: All stereoisomeric forms and mixtures thereof of a compound of the formula ##STR1## wherein X is --O-- or --S--, Y is --C.dbd.O, ##STR2## or --CH.sub.2 --, R.sub.1 is selected from the group consisting of hydrogen, halogen, optionally unsaturated alkyl of 1 to 8 carbon atoms and optionally unsaturated cycloalkyl of 3 to 8 carbon atoms, the latter two being optionally substituted with one or more halogen and aryl of 6 to 14 carbon atoms, R.sub.2 is selected from the group consisting of hydrogen, --CF.sub.3, --NO.sub.2, --CN, halogen, alkoxy of 1 to 8 carbon atoms, aryl of 6 to 14 carbon atoms, an ester, optionally unsaturated alkyl of 1 to 8 carbon atoms and optionally unsaturated cycloalkyl of 3 to 8 carbon atoms the latter two being optionally substituted with one or more halogen, R.sub.3 is selected from the group consisting of hydrogen, alkyl of 1 to 3 carbon atoms, --CN and --C.tbd.CH and A is the residue of an ACOOH pyrethrinoid acid having pesticidal properties.

    摘要翻译: 其中X为-O-或-S-,Y为-C = O, - 或 - 2-的式I化合物的所有立体异构形式及其混合物选自: 氢,卤素,1〜8个碳原子的任选不饱和的烷基和3〜8个碳原子的任选的不饱和环烷基,后两个任选被一个或多个6-14个碳原子的卤素和芳基取代,R2选自 由氢,-CF 3,-NO 2,-CN,卤素,1至8个碳原子的烷氧基,6至14个碳原子的芳基,酯,任选不饱和的1至8个碳原子的烷基和任选的不饱和的环烷基3至 8个碳原子,后两个任选被一个或多个卤素取代,R 3选自氢,1至3个碳原子的烷基,-CN和-C 3 C CH,A是ACOOH拟除虫菊酯酸的残基 具有杀虫性。

    Ribose-substituted aromatic amides, method for the production and use thereof as medicaments
    10.
    发明授权
    Ribose-substituted aromatic amides, method for the production and use thereof as medicaments 失效
    核糖取代的芳族酰胺,其生产和使用方法作为药物

    公开(公告)号:US06579902B1

    公开(公告)日:2003-06-17

    申请号:US09980728

    申请日:2002-01-09

    IPC分类号: A61K3135

    CPC分类号: C07H17/075

    摘要: Compounds of formula (I); wherein R1=alkyl, alkenyl or alkynyl, O-alkyl, O-alkenyl or optionally substituted, optionally interrupted O-alkynyl; R2=hydrogen or halogen; R3=hydrogen, alkyl or halogen; R4=NHR′ or NHOR″, R′ or R″ are identical or different and represent hydrogen, alkyl, alkenyl or alkynyl, aryl; R5=hydrogen or O-alkyl; R6=alkyl or CH2—O-alkyl; R7=hydrogen or alkyl or R6 et R7 form a cycle together with the carbon carrying them in addition to the addition salts thereof with bases. The compounds of formula (I) have antibiotic properties.

    摘要翻译: 式(I)化合物; 其中R 1 =烷基,烯基或炔基,O-烷基,O-烯基或任选取代的任选中断的O-炔基; R2 =氢或卤素; R3 =氢,烷基或卤素; R4 = NHR'或NHOR“,R'或R”相同或不同,表示氢,烷基,烯基或炔基,芳基; R5 =氢或O-烷基; R6 =烷基或CH2-O-烷基; R7 =氢或烷基或R6和R7与携带它们的碳以及与碱的加成盐一起形成一个循环。 式(I)化合物具有抗生素特性。