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    2-Amino-3-acylamino-6-benzylamino-pyridine-derivative having antiepileptic action
    1.
    发明授权
    2-Amino-3-acylamino-6-benzylamino-pyridine-derivative having antiepileptic action 失效
    具有抗癫痫作用的2-氨基-3-酰基氨基-6-苄基氨基 - 吡啶衍生物

    公开(公告)号：US4554281A

    公开(公告)日：1985-11-19

    申请号：US545930

    申请日：1983-10-27

    申请人： Walter vonBebenburg, deceased ,  Joachim Heese ,  Jurgen Engel ,  Kurt Thiele

    发明人： Walter vonBebenburg, deceased ,  Joachim Heese ,  Jurgen Engel ,  Kurt Thiele

    IPC分类号： C07D213/74 ,  A61K31/44 ,  A61P25/08 ,  C07D213/75

    CPC分类号： C07D213/75

    摘要： Compounds of the formula ##STR1## where R is a C.sub.1 -C.sub.4 alkyl group, a C.sub.1 -C.sub.4 alkoxy group, a phenoxy group or a phenyl-C.sub.1 -C.sub.2 -alkoxy group, R.sub.1 is hydrogen or a C.sub.1 -C.sub.4 -alkyl group and R.sub.5 is hydrogen or a C.sub.1 -C.sub.4 -alkyl group and the groups R.sub.2, R.sub.3, and R.sub.4 are the same or different and are hydrogen, halogen atoms, C.sub.1 -C.sub.4 alkyl groups, C.sub.1 -C.sub.4 -alkylcarbonyl group, the aminosulfonyl group, the trifluoromethyl group and their acid addition salts are effective as antiepileptics.

    摘要翻译： 其中R是C 1 -C 4烷基，C 1 -C 4烷氧基，苯氧基或苯基-C 1 -C 2 - 烷氧基的式Ⅺ化合物，R 1是氢或C 1 -C 4 - 烷基 并且R 5为氢或C 1 -C 4烷基，基团R 2，R 3和R 4相同或不同，为氢，卤素原子，C 1 -C 4烷基，C 1 -C 4烷基羰基，氨基磺酰基， 三氟甲基及其酸加成盐作为抗癫痫药有效。