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公开(公告)号:US06589934B1
公开(公告)日:2003-07-08
申请号:US09581386
申请日:2000-06-13
申请人: Dulce Garrido Bubacz , Iain David Dukes , Ed Williams McLean , Robert Anderson Noe , Andrew James Peat , Jerzy Ryszard Szewczyk , Stephen Andrew Thomson , Jennings Franklin Worley, III
发明人: Dulce Garrido Bubacz , Iain David Dukes , Ed Williams McLean , Robert Anderson Noe , Andrew James Peat , Jerzy Ryszard Szewczyk , Stephen Andrew Thomson , Jennings Franklin Worley, III
IPC分类号: A61K31395
CPC分类号: G01N33/6872 , C07D471/08 , G01N33/5008 , G01N33/502 , G01N33/507 , G01N33/5088 , G01N2333/705
摘要: The invention relates to methods of treatment of non insulin dependent diabetes mellitus, antagonists of the delayed rectifier potassium channel Kv2.1, methods of using and preparing the antagonists and assays for identifying such antagonists.
摘要翻译: 本发明涉及治疗非胰岛素依赖性糖尿病的方法,延迟整流钾通道Kv2.1的拮抗剂,使用和制备拮抗剂的方法以及用于鉴定此类拮抗剂的测定法。