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公开(公告)号:US20140288076A1
公开(公告)日:2014-09-25
申请号:US14295398
申请日:2014-06-04
申请人: Paul A. Barsanti , Cheng Hu , Jeff Jin , Robert Keyes , Robert Kucejko , Xiaodong Lin , Yue Pan , Keith B. Pfister , Martin Sendzik , James Sutton , Lifeng Wan
发明人: Paul A. Barsanti , Cheng Hu , Jeff Jin , Robert Keyes , Robert Kucejko , Xiaodong Lin , Yue Pan , Keith B. Pfister , Martin Sendzik , James Sutton , Lifeng Wan
IPC分类号: C07D409/14 , C07D401/14 , C07D405/14 , C07D401/04
CPC分类号: A61K31/497 , C07D213/74 , C07D241/20 , C07D401/04 , C07D401/12 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14
摘要: The present invention provides a compound of formula (I): and pharmaceutically acceptable salts, enantiomers, stereoisomers, rotamers, tautomers, diastereomers, or racemates thereof. Also provided is a method of treating a disease or condition mediated by CDK9.
摘要翻译: 本发明提供式(I)化合物及其药学上可接受的盐,对映体,立体异构体,旋转异构体,互变异构体,非对映体或其外消旋物。 还提供了治疗由CDK9介导的疾病或病症的方法。
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公开(公告)号:US20110028492A1
公开(公告)日:2011-02-03
申请号:US12843494
申请日:2010-07-26
申请人: Paul A. Barsanti , Cheng Hu , Jeff Jin , Robert Keyes , Robert Kucejko , Xiaodong Lin , Yue Pan , Keith B. Pfister , Martin Sendzik , James Sutton , Lifeng Wan
发明人: Paul A. Barsanti , Cheng Hu , Jeff Jin , Robert Keyes , Robert Kucejko , Xiaodong Lin , Yue Pan , Keith B. Pfister , Martin Sendzik , James Sutton , Lifeng Wan
IPC分类号: A61K31/497 , C07D213/02 , C07D401/04 , A61K31/444 , A61K31/506 , A61P31/18 , A61P35/00
CPC分类号: A61K31/497 , C07D213/74 , C07D241/20 , C07D401/04 , C07D401/12 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14
摘要: The present invention provides a compound of formula (I): and pharmaceutically acceptable salts, enantiomers, stereoisomers, rotamers, tautomers, diastereomers, or racemates thereof. Also provided is a method of treating a disease or condition mediated by CDK9.
摘要翻译: 本发明提供式(I)化合物及其药学上可接受的盐,对映体,立体异构体,旋转异构体,互变异构体,非对映体或其外消旋物。 还提供了治疗由CDK9介导的疾病或病症的方法。
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公开(公告)号:US08415381B2
公开(公告)日:2013-04-09
申请号:US12843494
申请日:2010-07-26
申请人: Paul A. Barsanti , Cheng Hu , Jeff Jin , Robert Keyes , Robert Kucejko , Xiaodong Lin , Yue Pan , Keith B. Pfister , Martin Sendzik , James Sutton , Lifeng Wan
发明人: Paul A. Barsanti , Cheng Hu , Jeff Jin , Robert Keyes , Robert Kucejko , Xiaodong Lin , Yue Pan , Keith B. Pfister , Martin Sendzik , James Sutton , Lifeng Wan
CPC分类号: A61K31/497 , C07D213/74 , C07D241/20 , C07D401/04 , C07D401/12 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14
摘要: The present invention provides a compound of formula (I): and pharmaceutically acceptable salts, enantiomers, stereoisomers, rotamers, tautomers, diastereomers, or racemates thereof. Also provided is a method of treating a disease or condition mediated by CDK9.
摘要翻译: 本发明提供式(I)化合物及其药学上可接受的盐,对映体,立体异构体,旋转异构体,互变异构体,非对映体或其外消旋物。 还提供了治疗由CDK9介导的疾病或病症的方法。
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