公开(公告)号：US08580780B2

公开(公告)日：2013-11-12

申请号：US13192707

申请日：2011-07-28

Applicant: John Gordon Allen ,  Karin Briner ,  Christopher Stanley Galka ,  Maria Angeles Martinez-Grau ,  Matthew Robert Reinhard ,  Michael John Rodriguez ,  Roger Ryan Rothhaar ,  Michael Wade Tidwell ,  Frantz Victor ,  Deyi Zhang ,  Steven Armen Boyd ,  Arundhati S. Deo ,  Wai-Man Lee ,  Christopher Stephen Siedem ,  Ajay Singh

Inventor： John Gordon Allen ,  Karin Briner ,  Christopher Stanley Galka ,  Maria Angeles Martinez-Grau ,  Matthew Robert Reinhard ,  Michael John Rodriguez ,  Roger Ryan Rothhaar ,  Michael Wade Tidwell ,  Frantz Victor ,  Deyi Zhang ,  Steven Armen Boyd ,  Arundhati S. Deo ,  Wai-Man Lee ,  Christopher Stephen Siedem ,  Ajay Singh

IPC: A61P3/04 ,  A61P25/22 ,  A61P25/24 ,  A61P25/30 ,  A61K31/55 ,  C07D223/16 ,  C07D401/12 ,  C07D417/12 ,  C07D413/12 ,  C07D403/12 ,  C07D409/12 ,  C07D405/12 ,  C07D413/14 ,  C07D417/06 ,  C07D403/06

CPC classification number: C07D223/16 ,  C07D401/12 ,  C07D403/06 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D413/14 ,  C07D417/06 ,  C07D417/12

Abstract: The present invention provides 6-substituted 2,3,4,5-tetrahydro-1H-benzo[d]azepines of Formula I as selective 5-HT2C receptor agonists for the treatment of 5-HT2C associated disorders including obesity, obsessive/compulsive disorder, depression, and anxiety: where: R6 is —S—R14; and other substituents are as defined in the specification.

Abstract translation: 本发明提供式I的6-取代2,3,4,5-四氢-1H-苯并[d]吖庚因作为选择性5-HT 2C受体激动剂，用于治疗5-HT 2C相关病症，包括肥胖，强迫症/强迫症 ，抑郁症和焦虑症：其中：R6为-S-R14; 和其它取代基如说明书中所定义。

公开(公告)号：US08541611B2

公开(公告)日：2013-09-24

申请号：US13535544

申请日：2012-06-28

Applicant: Gerhard Hamprecht ,  Michael Puhl ,  Bernd Wolf ,  Norbert Götz ,  Michael Keil ,  Robert Reinhard ,  Ingo Sagasser ,  Werner Seitz

Inventor： Gerhard Hamprecht ,  Michael Puhl ,  Bernd Wolf ,  Norbert Götz ,  Michael Keil ,  Robert Reinhard ,  Ingo Sagasser ,  Werner Seitz

IPC: C07C331/28

CPC classification number: C07D213/76 ,  C07C303/34 ,  C07C307/06 ,  C07C331/28 ,  C07C2601/14 ,  C07D207/20 ,  C07D211/18 ,  C07D211/70 ,  C07D295/26 ,  C07D307/52 ,  C07D319/06 ,  C07D333/20

Abstract: A process for preparing phenyl iso(thio)cyanates of the formula I in which a compound of the formula II or its HCl adduct is reacted with a phosgenating agent where W is oxygen or sulfur and Ar and A are as defined in claim 1 is described. Moreover, the invention relates to the use of the phenyl iso(thio)cyanates for preparing crop protection agents.

Abstract translation: 描述式I的苯基异（硫代）氰酸酯的方法，其中将式II化合物或其HCl加合物与W是氧或硫的光气反应剂和Ar和A如权利要求1中所定义的相同 。 此外，本发明涉及苯基异（硫代）氰酸酯用于制备作物保护剂的用途。

公开(公告)号：US20130102463A1

公开(公告)日：2013-04-25

申请号：US13805554

申请日：2011-06-21

Applicant: Thomas Ehrhardt ,  Klaus Grossmann ,  Johannes Hutzler ,  Anja Simon ,  Sylke Haremza ,  Michael Ishaque ,  Trevor William Newton ,  Robert Reinhard ,  Steven Bowe ,  Kyle Keller ,  Phil Munger

Inventor： Thomas Ehrhardt ,  Klaus Grossmann ,  Johannes Hutzler ,  Anja Simon ,  Sylke Haremza ,  Michael Ishaque ,  Trevor William Newton ,  Robert Reinhard ,  Steven Bowe ,  Kyle Keller ,  Phil Munger

IPC: A01N43/54

CPC classification number: A01N43/54 ,  A01N25/22 ,  A01N61/00 ,  A01N33/22 ,  A01N43/653 ,  A01N43/84 ,  A01N2300/00

Abstract: The present invention relates to herbicidal compositions comprising as herbicide A at least one protoporphyrinogen-IX oxidase inhibitor (PPO inhibitor), and at least one light detoxifying compound B, compositions comprising them and their use as herbicides, i.e. for controlling harmful plants, and also a method for controlling unwanted vegetation which comprises allowing a herbicidal effective amount of said herbicidal composition to act on plants, their seed and/or their habitat.

Abstract translation: 本发明涉及包含除草剂A至少一种原卟啉原-Ⅸ氧化酶抑制剂（PPO抑制剂）和至少一种轻解毒化合物B，包含它们的组合物及其作为除草剂的用途，即用于防治有害植物的除草组合物，以及 一种防治有害植物的方法，包括使除草有效量的所述除草组合物作用于植物，其种子和/或其栖息地。

公开(公告)号：US07820846B2

公开(公告)日：2010-10-26

申请号：US10532931

申请日：2003-10-29

Applicant: Gerhard Hamprecht ,  Michael Puhl ,  Bernd Wolf ,  Norbert Götz ,  Michael Keil ,  Robert Reinhard ,  Ingo Sagasser ,  Werner Seitz

Inventor： Gerhard Hamprecht ,  Michael Puhl ,  Bernd Wolf ,  Norbert Götz ,  Michael Keil ,  Robert Reinhard ,  Ingo Sagasser ,  Werner Seitz

IPC: C07C255/50

CPC classification number: C07D213/76 ,  C07C303/34 ,  C07C307/06 ,  C07C331/28 ,  C07C2601/14 ,  C07D207/20 ,  C07D211/18 ,  C07D211/70 ,  C07D295/26 ,  C07D307/52 ,  C07D319/06 ,  C07D333/20

Abstract: A process for preparing phenyl iso(thio)cyanates of the formula I in which a compound of the formula II or its HCl adduct is reacted with a phosgenating agent where W is oxygen or sulfur and Ar and A are as defined in claim 1 is described. Moreover, the invention relates to the use of the phenyl iso(thio)cyanates for preparing crop protection agents.

Abstract translation: 描述式I的苯基异（硫代）氰酸酯的方法，其中将式II化合物或其HCl加合物与W是氧或硫的光气反应剂和Ar和A如权利要求1中所定义的相同 。 此外，本发明涉及苯基异（硫代）氰酸酯用于制备作物保护剂的用途。

公开(公告)号：US20100167933A1

公开(公告)日：2010-07-01

申请号：US12663756

申请日：2008-06-20

Applicant: Eike Hupe ,  Thomas Seitz ,  Matthias Witschel ,  Dschun Song ,  William Karl Moberg ,  Liliana Parra Rapado ,  Frank Stelzer ,  Andrea Vescovi ,  Trevor William Newton ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt ,  Michael Rack ,  Elmar Kibler

Inventor： Eike Hupe ,  Thomas Seitz ,  Matthias Witschel ,  Dschun Song ,  William Karl Moberg ,  Liliana Parra Rapado ,  Frank Stelzer ,  Andrea Vescovi ,  Trevor William Newton ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt ,  Michael Rack ,  Elmar Kibler

IPC: A01N43/60 ,  C07D241/04 ,  A01P13/00

CPC classification number: C07D239/54 ,  A01N43/60 ,  A01N43/90 ,  C07D239/22 ,  C07D239/49 ,  C07D239/58 ,  C07D239/70 ,  C07D401/06 ,  C07D401/10 ,  C07D403/04 ,  C07D403/10 ,  C07D405/04 ,  C07D413/10 ,  C07D417/10 ,  C07D471/14 ,  C07D487/04 ,  C07D491/10

Abstract: The present invention relates to piperazine compounds of the general formula I defined below and to their use as herbicides. Moreover, the invention relates to compositions for crop protection and to a method for controlling unwanted vegetation. In formula I, A1, A2 independently of one another are aryl or heteroaryl, where Ra is attached in the ortho-position to the point of attachment of A1 to a carbon atom or a nitrogen atom of A1, Y1, Y2 are oxygen, sulfur or a group NRy1, and the variables Ra, Rb, Rc, Rd, Re, Rf, R1, R2, R3, R4, R5, R6, R7, and R8 have the meanings mentioned in the claims and the description.

Abstract translation: 本发明涉及下面定义的通式I的哌嗪化合物及其作为除草剂的用途。 此外，本发明涉及用于作物保护的组合物和用于防治不想要的植物的方法。 式Ⅰ中，A 1，A 2彼此独立地为芳基或杂芳基，其中R a与A1连接的位置与A1的碳原子或氮原子的邻位相连，Y 1，Y 2为氧，硫 或NRy1基团，变量Ra，Rb，Rc，Rd，Re，Rf，R1，R2，R3，R4，R5，R6，R7和R8具有权利要求书和说明书中提及的含义。

公开(公告)号：US20090137396A1

公开(公告)日：2009-05-28

申请号：US12159686

申请日：2007-01-04

Applicant: Eike Hupe ,  Cyrill Zagar ,  Matthias Witschel ,  Toralf Kuehn ,  William Karl Moberg ,  Liliana Parra Rapado ,  Frank Stelzer ,  Andrea Vescovi ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt

Inventor： Eike Hupe ,  Cyrill Zagar ,  Matthias Witschel ,  Toralf Kuehn ,  William Karl Moberg ,  Liliana Parra Rapado ,  Frank Stelzer ,  Andrea Vescovi ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt

IPC: A01N43/84 ,  A01N43/60 ,  C07D241/04 ,  A01P21/00 ,  C07D413/08

CPC classification number: C07D241/18 ,  A01N43/60 ,  A01N43/653 ,  A01N43/713 ,  A01N43/80 ,  A01N55/00 ,  C07D241/08 ,  C07D403/06 ,  C07D409/06 ,  C07D413/06 ,  C07D417/06

Abstract: The present invention relates to the use of piperazine compounds of the formula I or of the agriculturally useful salts of piperazine compounds of the formula I as herbicides, where in formula I the variables are as defined in the claims and the description.Moreover, the invention relates to compositions comprising, in addition to auxiliaries customary for formulating crop protection agents, piperazine compounds of the formula I or agriculturally useful salts of I, and to a process for preparing these compositions. Furthermore, the invention relates to certain piperazine compounds of the formula I, a process for preparing piperazine compounds of the formula I and a method for controlling unwanted vegetation which comprises treating plants, their seeds and/or their habitat with at least one piperazine compound of the formula I.

Abstract translation: 本发明涉及式I的哌嗪化合物或式I的哌嗪化合物的农业上可用的盐作为除草剂的用途，其中在式I中，变量如权利要求和说明书所定义。 此外，本发明涉及除了常规用于配制作物保护剂的助剂，式I的哌嗪化合物或I的农业上有用的盐以及制备这些组合物的方法之外，本发明涉及组合物。 此外，本发明涉及式I的某些哌嗪化合物，一种制备式I的哌嗪化合物的方法和一种防治有害植物的方法，其包括用至少一种哌嗪化合物处理植物，其种子和/或其栖息地 公式一

公开(公告)号：US20090054240A1

公开(公告)日：2009-02-26

申请号：US12279425

申请日：2007-02-07

Applicant: Matthias Witschel ,  Cyrill Zagar ,  Eike Hupe ,  Toralf Kuhn ,  William Karl Moberg ,  Liliana Parra Rapado ,  Frank Stelzer ,  Andrea Vescovi ,  Michael Rack ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt

Inventor： Matthias Witschel ,  Cyrill Zagar ,  Eike Hupe ,  Toralf Kuhn ,  William Karl Moberg ,  Liliana Parra Rapado ,  Frank Stelzer ,  Andrea Vescovi ,  Michael Rack ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt

IPC: A01N43/56 ,  C07D231/14 ,  C07D333/24 ,  C07D307/68 ,  A01N43/10 ,  C07D405/02 ,  A01P13/00

CPC classification number: C07D231/12 ,  C07D333/06 ,  C07D401/12 ,  C07D403/12 ,  C07D407/12

Abstract: The present invention relates to heteroaroyl-substituted alanines of the formula I in which the variables A and R1 to R7 are as defined in the description, and to their agriculturally useful salts, to processes and intermediates for their preparation, and to the use of these compounds or of compositions comprising these compounds for controlling unwanted plants.

Abstract translation: 本发明涉及式I的杂芳酰基取代的丙氨酸，其中变量A和R 1至R 7如说明书中所定义，并且其农业上有用的盐，其制备方法和中间体以及这些 化合物或包含这些化合物的组合物以控制不想要的植物。

公开(公告)号：US20090042727A1

公开(公告)日：2009-02-12

申请号：US11908635

申请日：2006-03-16

Applicant: Richard R. Evans ,  Rex Liebl ,  Robert Reinhard ,  Helmut Walter ,  Cyrill Zagar

Inventor： Richard R. Evans ,  Rex Liebl ,  Robert Reinhard ,  Helmut Walter ,  Cyrill Zagar

IPC: A01N43/80 ,  A01P13/00

CPC classification number: A01N43/54 ,  A01N43/80 ,  A01N43/84 ,  A01N2300/00

Abstract: A herbicidal composition comprising a) at least one 3-phenyluracils of formula I wherein the variables R1 to R7 are as defined in the specification; and b) at least one 3-sulfonylisoxazoline of formula II wherein the variables R8 and R9 are as defined in the specification; and c) optionally at least one safener III selected from the group as defined in the specification.

Abstract translation: 一种除草组合物，其包含a）至少一种式I的3-苯基尿嘧啶，其中变量R1至R7如说明书中所定义; 和b）至少一种式II的3-磺酰基异恶唑啉，其中变量R8和R9如说明书中所定义; 和c）任选的至少一种安全剂III，其选自说明书中定义的基团。

公开(公告)号：US20090036311A1

公开(公告)日：2009-02-05

申请号：US12279351

申请日：2007-02-07

Applicant: Matthias Witschel ,  Cyrill Zagar ,  Eike Hupe ,  Toralf Kuhn ,  William Karl Moberg ,  Liliana Parra Rapado ,  Frank Stelzer ,  Andrea Vescovi ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt

Inventor： Matthias Witschel ,  Cyrill Zagar ,  Eike Hupe ,  Toralf Kuhn ,  William Karl Moberg ,  Liliana Parra Rapado ,  Frank Stelzer ,  Andrea Vescovi ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt

IPC: A01N37/18 ,  C07C237/34 ,  C07C229/34 ,  A01N37/44 ,  A01P13/00

CPC classification number: C07D307/14 ,  C07C237/22 ,  C07C271/22 ,  C07C275/16 ,  C07C311/06 ,  C07C311/58 ,  C07C335/08 ,  C07C335/10 ,  C07D309/04 ,  C07D309/20

Abstract: The present invention relates to benzoyl-substituted alanines of the formula I in which the variables R1 to R12 are as defined in the description, and to their agriculturally useful salts, to processes and intermediates for their preparation, and to the use of these compounds or of compositions comprising these compounds for controlling unwanted plants.

Abstract translation: 本发明涉及式I的苯甲酰基取代的丙氨酸，其中变量R1至R12如说明书中所定义，及其农业上有用的盐，其制备方法和中间体以及这些化合物或 包含这些化合物的组合物用于防治有害植物。

公开(公告)号：US20050239655A1

公开(公告)日：2005-10-27

申请号：US10522095

申请日：2003-07-22

Applicant: Michael Puhl ,  Gerhard Hamprecht ,  Robert Reinhard ,  Ingo Sagasser ,  Werner Seitz ,  Cyrill Zagar ,  Andreas Landes

Inventor： Michael Puhl ,  Gerhard Hamprecht ,  Robert Reinhard ,  Ingo Sagasser ,  Werner Seitz ,  Cyrill Zagar ,  Andreas Landes

IPC: A01N25/30 ,  A01N43/38 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/64 ,  A01N43/653 ,  A01N43/90 ,  C07D213/61 ,  C07D213/65 ,  C07D231/16 ,  C07D231/18 ,  C07D237/14 ,  C07D237/22 ,  C07D239/54 ,  C07D251/38 ,  A01N43/46

CPC classification number: C07D251/38 ,  C07D213/61 ,  C07D213/65 ,  C07D231/16 ,  C07D231/18 ,  C07D237/14 ,  C07D237/22 ,  C07D239/54

Abstract: Disclosed are 3-heterocyclyl substituted benzoic acid derivatives of general formula (I), in which the variables R1 to R8 and X have the meanings indicated in claim 1, and the use thereof as herbicides or for desiccating/defoliating plants.

Abstract translation: 公开了通式（I）的3-杂环基取代的苯甲酸衍生物，其中变量R 1至R 8和X具有权利要求1所示的含义，和 其用作除草剂或用于干燥/脱叶植物。