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公开(公告)号:US09505775B2
公开(公告)日:2016-11-29
申请号:US14440085
申请日:2013-10-31
申请人: Carl Thibeault , Jean Rancourt , Pierre L. Beaulieu , Anne Décor , Chantal Grand-Maitre , Cyrille Kuhn , Elisia Villemure , Oliver Hucke , Simon Surprenant , Melissa Leblanc , Jean-Eric Lacoste , Benoit Moreau , Eric Jolicoeur
发明人: Carl Thibeault , Jean Rancourt , Pierre L. Beaulieu , Anne Décor , Chantal Grand-Maitre , Cyrille Kuhn , Elisia Villemure , Oliver Hucke , Simon Surprenant , Melissa Leblanc , Jean-Eric Lacoste , Benoit Moreau , Eric Jolicoeur
IPC分类号: C07D403/14 , C07D403/06 , C07D413/14 , C07D401/14 , C07D209/04 , A61K31/404 , A61K31/4178 , A61K31/4155 , A61K31/4192 , A61K31/4196 , A61K31/422 , A61K31/44 , A61K31/497 , C07D491/107 , C07D403/08 , C07D471/04 , C07D487/10 , C07D471/10
CPC分类号: C07D491/107 , C07D401/14 , C07D403/06 , C07D403/08 , C07D403/14 , C07D413/14 , C07D471/04 , C07D471/10 , C07D487/10
摘要: Compounds of Formula (I) wherein R1, R2, R3A, R3B, Y, Z1 and Z2 are defined herein, are useful for the treatment of cytomegalovirus disease and/or infection.
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公开(公告)号:US09315499B2
公开(公告)日:2016-04-19
申请号:US14390243
申请日:2013-04-03
申请人: Lee Fader , Olivier Lepage , Murray Bailey , Pierre Louis Beaulieu , Francois Bilodeau , Rebekah J. Carson , André Giroux , Cédrickx Godbout , Benoît Moreau , Julie Naud , Mathieu Parisien , Martin Poirier , Maude Poirier , Simon Surprenant , Carl Thibeault
发明人: Lee Fader , Olivier Lepage , Murray Bailey , Pierre Louis Beaulieu , Francois Bilodeau , Rebekah J. Carson , André Giroux , Cédrickx Godbout , Benoît Moreau , Julie Naud , Mathieu Parisien , Martin Poirier , Maude Poirier , Simon Surprenant , Carl Thibeault
IPC分类号: C07D471/04 , A61K31/4375 , C07D519/00 , A61K31/496 , A61K31/5513 , A61K31/506 , A61K31/553 , A61K31/4985 , A61K31/5377 , A61K31/541 , A61K31/501 , A61K45/06 , C12N7/00
CPC分类号: C07D471/04 , A61K31/4375 , A61K31/496 , A61K31/4985 , A61K31/501 , A61K31/506 , A61K31/5377 , A61K31/541 , A61K31/5513 , A61K31/553 , A61K45/06 , C07D519/00 , C12N7/00 , C12N2710/16163
摘要: Compounds of Formula (I) wherein n, m, R1, R2, R3, R4, R5 and R6 are defined herein, are useful for the treatment of cytomegalovirus disease and/or infection.
摘要翻译: 其中n,m,R 1,R 2,R 3,R 4,R 5和R 6在本文中定义的式(I)化合物可用于治疗巨细胞病毒疾病和/或感染。
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公开(公告)号:US08338441B2
公开(公告)日:2012-12-25
申请号:US12777406
申请日:2010-05-11
申请人: Christiane Yoakim , Murray Bailey , Francois Bilodeau , Rebekah Carson , Lee Fader , Stephen Kawai , Sebastien Morin , Carl Thibeault , Bruno Simoneau , Simon Surprenant , Youla Tsantrizos , Steven Laplante
发明人: Christiane Yoakim , Murray Bailey , Francois Bilodeau , Rebekah Carson , Lee Fader , Stephen Kawai , Sebastien Morin , Carl Thibeault , Bruno Simoneau , Simon Surprenant , Youla Tsantrizos , Steven Laplante
IPC分类号: A01N43/40 , A61K31/435
CPC分类号: C07D213/81 , A61K31/4375 , A61K31/44 , A61K31/4433 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K31/4709 , A61K31/4741 , A61K31/501 , A61K31/506 , A61K31/538 , A61K31/5383 , A61K45/06 , C07D213/55 , C07D401/12 , C07D405/10 , C07D405/14 , C07D411/10 , C07D413/10 , C07D413/14 , C07D417/10 , C07D471/04 , C07D491/06 , C07D498/06
摘要: Compounds of formula I: wherein a, R1, R2, R3, R4, R5 and R6 are defined herein, are useful as inhibitors of HIV replication.
摘要翻译: 式I化合物:其中a,R 1,R 2,R 3,R 4,R 5和R 6在本文中定义,可用作HIV复制的抑制剂。
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公开(公告)号:US20100292227A1
公开(公告)日:2010-11-18
申请号:US12777406
申请日:2010-05-11
申请人: CHRISTIANE YOAKIM , MURRAY BAILEY , FRANCOIS BILODEAU , REBEKAH CARSON , LEE FADER , STEPHEN KAWAI , SEBASTIEN MORIN , CARL THIBEAULT , BRUNO SIMONEAU , SIMON SURPRENANT , YOULA TSANTRIZOS , STEVEN LAPLANTE
发明人: CHRISTIANE YOAKIM , MURRAY BAILEY , FRANCOIS BILODEAU , REBEKAH CARSON , LEE FADER , STEPHEN KAWAI , SEBASTIEN MORIN , CARL THIBEAULT , BRUNO SIMONEAU , SIMON SURPRENANT , YOULA TSANTRIZOS , STEVEN LAPLANTE
IPC分类号: A61K31/5383 , C07D405/02 , A61K31/4433 , C07D401/14 , A61K31/444 , C07D401/10 , A61K31/4439 , A61K31/506 , A61K31/501 , C07D413/12 , C07D417/02 , C07D413/02 , A61K31/538 , A61K31/4741 , C07D491/16 , C07D401/02 , A61K31/4709 , C07D417/12 , C07D498/16 , A61P31/18
CPC分类号: C07D213/81 , A61K31/4375 , A61K31/44 , A61K31/4433 , A61K31/4436 , A61K31/4439 , A61K31/444 , A61K31/4709 , A61K31/4741 , A61K31/501 , A61K31/506 , A61K31/538 , A61K31/5383 , A61K45/06 , C07D213/55 , C07D401/12 , C07D405/10 , C07D405/14 , C07D411/10 , C07D413/10 , C07D413/14 , C07D417/10 , C07D471/04 , C07D491/06 , C07D498/06
摘要: Compounds of formula I: wherein a, R1, R2, R3, R4, R5 and R6 are defined herein, are useful as inhibitors of HIV replication.
摘要翻译: 式I化合物:其中a,R 1,R 2,R 3,R 4,R 5和R 6在本文中定义,可用作HIV复制的抑制剂。
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公开(公告)号:US20150274744A1
公开(公告)日:2015-10-01
申请号:US14440085
申请日:2013-10-31
申请人: Carl THIBEAULT , Jean RANCOURT , Pierre L. BEAULIEU , Anne DECOR , Chantal GRAND-MAITRE , Cyille KUHN , Elisia VILLEMURE , Melissa LEBLANC , Jene-Eric LACOSTE , Benoit MOREAU , Eric JOLICOEUR , Simon SURPRENANT , Oliver HUCKE
发明人: Carl Thibeault , Jean Rancourt , Pierre L. Beaulieu , Anne Décor , Chantal Grand-Maitre , Cyrille Kuhn , Elisia Villemure , Oliver Hucke , Simon Surprenant , Melissa Leblanc , Jean-Eric Lacoste , Benoit Moreau , Eric Jolicoeur
IPC分类号: C07D491/107 , C07D401/14 , C07D471/10 , C07D413/14 , C07D403/14 , C07D403/06
CPC分类号: C07D491/107 , C07D401/14 , C07D403/06 , C07D403/08 , C07D403/14 , C07D413/14 , C07D471/04 , C07D471/10 , C07D487/10
摘要: Compounds of Formula (I) wherein R1, R2, R3A, R3B, Y, Z1 and Z2 are defined herein, are useful for the treatment of cytomegalovirus disease and/or infection.
摘要翻译: 其中R1,R2,R3A,R3B,Y,Z1和Z2在本文中定义的式(I)化合物可用于治疗巨细胞病毒疾病和/或感染。
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公开(公告)号:US20100069353A1
公开(公告)日:2010-03-18
申请号:US12517310
申请日:2007-12-03
申请人: Christiane Yoakim , Patrick Deroy , Martin Duplessis , Alexandre Gagnon , Sylvie Goulet , Oliver Huecke , Christopher Lemke , Simon Surprenant
发明人: Christiane Yoakim , Patrick Deroy , Martin Duplessis , Alexandre Gagnon , Sylvie Goulet , Oliver Huecke , Christopher Lemke , Simon Surprenant
IPC分类号: A61K31/397 , C07D401/14 , A61K31/4439 , C07D403/02 , A61K31/4184 , C07D413/14 , A61K31/5377 , C07D403/14 , A61K31/496 , A61P31/18
CPC分类号: C07D409/14 , C07D405/14 , C07D413/14 , C07D417/14
摘要: The present invention relates to compounds of formula (I) wherein R1, R2, R3 and R4 are as defined herein, compositions and uses thereof for treating human immunodeficiency virus (HIV) infection. In particular, the present invention provides novel inhibitors of HIV replication, pharmaceutical compositions containing such compounds and methods for using these compounds in the treatment of HIV infection.
摘要翻译: 本发明涉及其中R 1,R 2,R 3和R 4如本文所定义的式(I)化合物,其用于治疗人类免疫缺陷病毒(HIV)感染的组合物和用途。 特别地,本发明提供HIV复制的新型抑制剂,含有这些化合物的药物组合物和使用这些化合物治疗HIV感染的方法。
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